Herbicidal sulfonamides

ABSTRACT

Tetrazole-substituted benzenesulfonamides are useful as agricultural chemicals and, in particular, as growth regulants and herbicides.

RELATED APPLICATION

This application is a continuation-in-part of copending application U.S. Ser. No. 934,118, filed Nov. 24, 1986, now U.S. Pat. No. 4,746,353, which in turn is a continuation-in-part of copending application U.S. Ser. No. 849,618, filed Apr. 11, 1986, now abandoned which in turn is a continuation-in-part of copending application U.S. Ser. No. 739,214, filed May 30, 1985, now abandoned.

BACKGROUND OF THE INVENTION

This invention relates to tetrazole-substituted benzene sulfonamides which are useful as agricultural chemicals such as growth regulants and herbicides.

U.S. Pat. No. 4,127,405 and U.S. Pat. No. 4,169,719 disclose herbicidal benzenesulfonylureas.

EP-A-No. 165,753, published Dec. 27, 1985, discloses herbicidal thiophenesulfonamides of formula ##STR1## wherein Q is optionally substituted phenyl or an optionally substituted saturated or unsaturated 5- or 6-membered heterocyclic ring containing one to three heteroatoms.

EP-A-No. 83,975 (published July 20, 1983) discloses herbicidal benzenesulfonamides of formula ##STR2## wherein Q is selected from various five or six-membered aromatic or partially unsaturated heterocyclic rings containing 2 or 3 heteroatoms selected from O, S or NR.

EP-A-No. 85,476 (published Aug. 10, 1983) discloses herbicidal benzenesulfonamides of formulae ##STR3## wherein Q is selected from various 5-membered aromatic heterocycles, and their dihydro and tetrahydro analogs, which contain one heteroatom selected from O, S or NR, or Q is a saturated or partially unsaturated 6-membered ring containing one heteroatom selected from O or S; and

Q¹ is a 6-membered aromatic heterocycle containing one to three N atoms.

South African patent application 83/8416 (published May 12, 1984) discloses herbicidal benzenesulfonamides of formula ##STR4## wherein A is an unsaturated or only partially saturated 5- or 6-membered heterocyclic ring system which is bonded through a carbon atom and contains 1, 2 or 3 heteroatoms.

EP-A-No. 116,518, published Aug. 22, 1984, discloses herbicidal sulfonamides of formula ##STR5## wherein X is NR₆ R₇, N(SO₂ R₉)₂ or ##STR6## A is CO, SO₂, CONR₂₃ or CO₂ ; B is C₁ -C₄ alkyl or C₂ -C₄ alkenyl; and

C is CO, CR₂₁ R₂₂ or SO₂.

U.S. Pat. No. 4,475,944 discloses herbicidal sulfamates, possessing an ortho-heterocyclic ring, such as those of formula ##STR7## wherein W is O, S or NR₁.

EP-A-No. 164,268, published Dec. 11, 1985, discloses herbicidal benzylsulfonamides of formula ##STR8## wherein Q is a saturated, 5- or 6-membered ring containing 1 to 2 heteroatoms selected from 0-2 S or 0-2 O or an unsaturated 5- or 6-membered ring containing 1 to 3 heteroatoms selected from 0-S, 0-1 O or 0-3 N and Q may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₁ -C₂ haloalkoxy, C₃ -C₄ alkenylthio, C₁ -C₂ haloalkylthio or SCH₂ CN.

EP-A-No. 165,753, published Dec. 27, 1985, discloses herbicidal pyridinesulfonamides of formula ##STR9## wherein Q is phenyl optionally substituted with Cl, CH₃ O or CH₃, a saturated 5-membered ring containing 1 heteroatom selected from O or S, or an unsaturated 5- or 6-membered ring containing 1 to 3 heteroatoms selected from 0-1 S, 0-1 O or 0-3 N and when Q is an unsaturated 5- or 6-membered ring, it may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₃ -C₄ alkenylthio, C₁ -C₂ haloalkoxy or C₁ -C₂ haloalkylthio.

EP-A-No. 176,304, published Apr. 11, 1986, discloses herbicidal pyrazolesulfonamides such as those of formula ##STR10## wherein Q is a saturated 5- or b 6-membered ring containing 1 heteroatom selected from 0-1 S or 0-1 O or an unsaturated 5- or 6-membered ring containing 1-3 heteroatoms selected from 0-1 S, 0-1 O or 0-3 N and Q may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₃ -C₄ alkenylthio, C₃ -C₄ alkenyloxy, C₁ -C₂ haloalkoxy, C₁ -C₂ haloalkylthio, C₂ -C₄ cyanoalkylthio or C₁ -C₂ alkoxycarbonylmethylthio.

EP-A-No. 141,777, published May 15, 1985, discloses ortho-benzyl-substituted sulfonylureas of the formula ##STR11## wherein Y is O or S; and

R¹⁷ is a 5- to 6-membered unsaturated heterocyclic radical including ##STR12## U.S. Pat. No. 4,602,936 carrying part of this disclosure, issued July 29, 1986.

South African patent application No. 83/0441, published July 25, 1983, discloses herbicidal benzenesulfonamides of formula ##STR13## wherein R₁ is H, halogen, NO₂, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₅ alkenyl or C₁ -C₄ alkoxycarbonyl;

R₂ is C₁ -C₃ alkyl or C₁ -C₃ alkoxy, each unsubstituted or substituted by 1 to 3 halogen atoms;

R₃ is halogen, H, NR₄ R₅, C₁ -C₃ alkyl, unsubstituted or substituted by 1 to 3 alkoxy, unsubstituted or substituted by methoxy, ethoxy, or 1 to 3 halogen atoms;

A is C₁ -C₄ alkylene or C₂ -C₄ alkenylene, each unsubstituted or substituted by C₁ -C₄ alkyl;

m is 0 or 1;

E is N or CH;

X is oxygen, sulfur, SO or SO₂ ; and

Q is, in part, a 5- or 6-membered heterocyclic ring bound through carbon or nitrogen, such heterocycles including furan, pyrane, thiophene, triazole, pyridine, pyrroline, oxaxole, isooxazole, thiazole, isothiazole, thiadiaxole, oxathiole, pyrrole, imidazole, pyrazole, pyrazine, pyrimidine, pyridazine, symmetrical and assymetrical triazines, oxdiazole, oxazine, furazane, pyridine-N-oxide, thiophene-S-oxide, benzthiophene, benzofuran, isobenzofuran, chromene, chromane, indole, isoindole, indazole, quinoline, isoquinoline, phthalazine, quinoxaline, quinazoline, quinoline, benzthiazole and benzimidiazole, and partially or completely hydrogenated and fused homoglogues thereof.

South African patent application No. 85/2646, published Oct. 11, 1985, discloses herbicidal benzenesulfonamides of formula ##STR14## wherein R₁ is H, halogen, NO₂, alkyl, alkoxy, alkoxycarbonyl or haloalkyl;

X is O, S, SO or SO₂ ;

Y is O or S;

E is CH or N;

R₂ and R₃ are independently alkyl, alkoxy or alkoxyalkyl;

A is alkylene or alkenylene;

m is 0 or 1;

Q is, in part, ##STR15## each of which is optionally substituted and/or optionally partially hydrogenated; and

X' is O, S or NR.

The presence of undesired vegetation causes substantial damage to useful crops, especially agricultural products that satisfy man's basic food needs, such as corn, soybeans, wheat and the like. The current population explosion and concomitant world food shortage demand improvements in the efficiency of producing these crops. Prevention or minimization of the loss of a portion of valuable crops by killing or inhibiting the growth of undesired vegetation is one way of improving this efficiency.

A wide variety of materials, useful for killing, or inhibiting (controlling) the growth of undesired vegetation is available. Such materials are commonly referred to as herbicides. The need exists, however, for still more effective herbicides that destroy or retard weeds without causing significant damage to useful crops.

SUMMARY OF THE INVENTION

This invention relates to novel compounds of Formula I, agriculturally suitable compositions containing them, and their method-of-use as preemergent or postemergent herbicides or as plant growth regulants. ##STR16## wherein J is ##STR17## W is O, S or NR_(X) ; R_(X) is H, OH, C₁ -C₃ alkyl, C₁ -C₃ alkoxy, allyloxy, propargyloxy, C₁ -C₃ haloalkyl, C₁ -C₃ haloalkoxy or NR_(Y) R_(Z) ;

R_(Y) is H or C₁ -C₃ alkyl;

R_(Z) is C₁ -C₃ alkyl;

G is O, S, SO or SO₂ ;

m is 0 or 1;

n is 0, 1 or 2;

R is H or CH₃ ;

E is a single bond, CH₂ or O;

Q is ##STR18## R₁ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR_(a) R_(b), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, SCN, CO₂ R_(c), C₁ -C₃ haloalkoxy, C₁ -C₃ haloalkylthio, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ haloalkoxy, C₁ -C₂ alkylthio, C₁ -C₂ haloalkylthio or CN;

R₂ is H, C₁ -C₃ alkyl, allyl or phenyl;

R₃ is H, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, CH₂ -(C₂ -C₅ alkenyl), CH₂ (C₂ -C₅ haloalkenyl), CH₂ (C₂ -C₅ alkynyl), CH₂ (C₂ -C₅ haloalkynyl), C₆ H₅ or C₁ -C₄ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, C₁ -C₂ alkylsulfinyl or C₁ -C₂ alkylsulfonyl;

R₄ is H, halogen, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, C₂ -C₆ alkenyl, C₂ -C₆ haloalkenyl, C₂ -C₆ alkynyl, C₃ -C₆ haloalkynyl, C₆ H₅, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, OCH₂ CH₂ O-(C₁ -C₂ alkyl) or di(C₁ -C₃ alkyl)amino;

R₅ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, allyl or propargyl;

R_(a) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy;

R_(b) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or

R_(a) and R_(b) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --;

R_(c) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ haloalkyl, C₁ -C₂ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or C₂ -C₄ alkoxyalkyl;

A is ##STR19## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkyl, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, halogen, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₃ -C₅ cycloalkyl;

Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₂ -C₅ alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, C₁ -C₄ haloalkyl, C₂ -C₄ alkynyl, azido, cyano, ##STR20## or --N(OCH₃)CH₃ ; p is 2 or 3;

L₁ and L₂ are independently O or S;

R₆ is H or CH₃ ;

R₇ and R₈ are independently C₁ -C₃ alkyl;

Z is CH, N, CCH₃, CC₂ H₅, CCl or CBr;

Y₁ is O or CH₂ ;

X₁ is CH₃, OCH₃, OC₂ H₅ or OCF₂ H;

X₂ is CH₃, C₂ H₅ or CH₂ CF₃ ;

Y₂ is OCH₃, OC₂ H₅, SCH₃, SC₂ H₅, CH₃ or CH₂ CH₃ ;

X₃ is CH₃ or OCH₃ ;

Y₃ is H or CH₃ ;

X₄ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl;

Y₄ is CH₃, OCH₃, OC₂ H₅ or Cl; and

Z¹ is CH or N;

and their agriculturally suitable salts; provided that

(a) when X is Cl, F, Br or I, then Z is CH and Y is OCH₃, OC₂ H₅, N(OCH₃)CH₃, NHCH₃, N(CH₃)₂ or OCF₂ H;

(b) when X or Y is C₁ haloalkoxy, then Z is CH;

(c) when J is J-9 and n is O, then Q is Q-1 or Q-2;

(d) when E is O, then J is J-1;

(e) when W is S, then A is A-1, R is H, and Y is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH(OCH₃)₂ or ##STR21## (f) when the total number of carbon atoms in X and Y is greater than 4, then the carbon content of R₁, R₃, R₄ and R₅ must each be less than or equal to 2;

(g) X₄ and Y₄ cannot simultaneously be Cl;

(h) when J is J-1 and m is 0, then n is 0; and

(i) when n is 0 and m is 1, then Q is Q-1 or Q-2.

In the above definitions, the term "alkyl" used either alone or in compound words such as "alkylthio" or "haloalkyl", denotes straight chain or branched alkyl, e.g., methyl, ethyl, n-propyl, isopropyl or the different butyl, pentyl or hexyl isomers.

Alkoxy denotes methoxy, ethoxy, n-propoxy, isopropoxy and the different butyl isomers.

Alkenyl denotes straight chain or branched alkenes, e.g., vinyl, 1-propenyl, 2-propenyl, 3-propenyl and the different butenyl, pentenyl or hexenyl isomers.

Alkynyl denotes straight chain or branched alkynes, e.g., ethynyl, 1-propynyl, 2-propynyl and the different butynyl, pentynyl and hexynyl isomers.

Alkylsulfonyl denotes methylsulfonyl, ethylsulfonyl or the different propylsulfonyl isomers.

Alkylthio, alkylsulfinyl, alkylamino, etc. are defined in an analogous manner.

Cycloalkyl denotes cyclopropyl, cyclobutyl, cyclopentyl and cyclohexyl.

The term "halogen", either alone or in compound words such as "haloalkyl", denotes fluorine, chlorine, bromine or iodine.

In terms such as C₂ -C₃ alkylthioalkyl, the specified number of carbon atoms is meant to define the total number of carbon atoms in that substituent group. For example, C₂ -C₃ alkylthioalkyl would designate CH₂ SCH₃, CH₂ SC₂ H₅, CH₂ CH₂ SCH₃ or CH(CH₃)SCH₃, and C₂ -C₅ alkoxyalkoxy would represent OCH₂ OCH₃ through O(CH₂)₄ OCH₃ or OCH₂ O(CH₂)₃ CH₃ and the various structural isomers embraced therein.

Preferred for reasons of increased ease of synthesis and/or greater herbicidal efficacy are:

(1) Compounds of Formula I where E is a single bond.

(2) Compounds of Formula I where E is CH₂.

(3) Compounds of Formula I where E is O.

(4) Compounds of Preferred 1 where

m is 0; and

W is O.

(5) Compounds of Preferred 4 where

X is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, cyclopropyl, Cl, F, Br, I, OCF₂ H, CH₂ F, CF₃, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and

Y is H, C₁ -C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH₂ SCH₃, ##STR22## OCF₂ H, SCF₂ H, OCF₂ Br, C.tbd.CH or C.tbd.CCH₃.

(6) Compounds of Preferred 5 where

R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; and

n is 0.

(7) Compounds of Preferred 6 where

R₃ is H, C₁ -C₃ alkyl, C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; and

R₄ is H, C₁ -C₃ alkyl, C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, N(CH₃)₂, allyl, propargyl of C₁ -C₂ alkyl substituted with 1-3 atoms of F, Cl or Br.

(8) Compounds of Preferred 7 where J is J-1.

(9) Compounds of Preferred 8 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(10) Compounds of Preferred 9 where Q is Q₁.

(11) Compounds of Preferred 9 where Q is Q₂.

(12) Compounds of Preferred 9 where Q is Q₃.

(13) Compounds of Preferred 9 where Q is Q₄.

(14) Compounds of Preferred 9 where Q is Q₅.

(15) Compounds of Preferred 9 where Q is Q₆.

(16) Compounds of Preferred 9 where Q is Q₇.

(17) Compounds of Preferred 7 where J is J-2. (18) Compounds of Preferred 17 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(19) Compounds of Preferred 18 where Q is Q₁.

(20) Compounds of Preferred 18 where Q is Q₂.

(21) Compounds of Preferred 18 where Q is Q₃.

(22) Compounds of Preferred 18 where Q is Q₄.

(23) Compounds of Preferred 18 where Q is Q₅.

(24) Compounds of Preferred 18 where Q is Q₆.

(25) Compounds of Preferred 18 where Q is Q₇.

(26) Compounds of Preferred 7 where J is J-3.

(27) Compounds of Preferred 26 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(28) Compounds of Preferred 27 where Q is Q₁.

(29) Compounds of Preferred 27 where Q is Q₂.

(30) Compounds of Preferred 27 where Q is Q₃.

(31) Compounds of Preferred 27 where Q is Q₄.

(32) Compounds of Preferred 27 where Q is Q₅.

(33) Compounds of Preferred 27 where Q is Q₆.

(34) Compounds of Preferred 27 where Q is Q₇.

(35) Compounds of Preferred 7 where J is J-4.

(36) Compounds of Preferred 35 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(37) Compounds of Preferred 36 where Q is Q₁.

(38) Compounds of Preferred 36 where Q is Q₂.

(39) Compounds of Preferred 36 where Q is Q₃.

(40) Compounds of Preferred 36 where Q is Q₄.

(41) Compounds of Preferred 36 where Q is Q₅.

(42) Compounds of Preferred 36 where Q is Q₆.

(43) Compounds of Preferred 36 where Q is Q₇.

(44) Compounds of Preferred 7 where J is J-5.

(45) Compounds of Preferred 44 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(46) Compounds of Preferred 45 where Q is Q₁.

(47) Compounds of Preferred 45 where Q is Q₂.

(48) Compounds of Preferred 45 where Q is Q₃.

(49) Compounds of Preferred 45 where Q is Q₄.

(50) Compounds of Preferred 45 where Q is Q₅.

(51) Compounds of Preferred 45 where Q is Q₆.

(52) Compounds of Preferred 45 where Q is Q₇.

(53) Compounds of Preferred 7 where J is J-6.

(54) Compounds of Preferred 53 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(55) Compounds of Preferred 54 where Q is Q₁.

(56) Compounds of Preferred 54 where Q is Q₂.

(57) Compounds of Preferred 54 where Q is Q₃.

(58) Compounds of Preferred 54 where Q is Q₄.

(59) Compounds of Preferred 54 where Q is Q₅.

(60) Compounds of Preferred 54 where Q is Q₆.

(61) Compounds of Preferred 54 where Q is Q₇.

(62) Compounds of Preferred 7 where J is J-7.

(63) Compounds of Preferred 62 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ H₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(64) Compounds of Preferred 63 where Q is Q₁.

(65) Compounds of Preferred 63 where Q is Q₂.

(66) Compounds of Preferred 63 where Q is Q₃.

(67) Compounds of Preferred 63 where Q is Q₄.

(68) Compounds of Preferred 63 where Q is Q₅.

(69) Compounds of Preferred 63 where Q is Q₆.

(70) Compounds of Preferred 63 where Q is Q₇.

(71) Compounds of Preferred 7 where J is J-8.

(72) Compounds of Preferred 71 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(73) Compounds of Preferred 72 where Q is Q₁.

(74) Compounds of Preferred 72 where Q is Q₂.

(75) Compounds of Preferred 72 where Q is Q₃.

(76) Compounds of Preferred 72 where Q is Q₄.

(77) Compounds of Preferred 72 where Q is Q₅.

(78) Compounds of Preferred 72 where Q is Q₆.

(79) Compounds of Preferred 72 where Q is Q₇.

(80) Compounds of Preferred 7 where J is J-9.

(81) Compounds of Preferred 80 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(82) Compounds of Preferred 81 where Q is Q₁.

(83) Compounds of Preferred 81 where Q is Q₂.

(84) Compounds of Preferred 81 where Q is Q₃.

(85) Compounds of Preferred 81 where Q is Q₄.

(86) Compounds of Preferred 81 where Q is Q₅.

(87) Compounds of Preferred 81 where Q is Q₆.

(88) Compounds of Preferred 81 where Q is Q₇.

(89) Compounds of Preferred 7 where J is J-10.

(90) Compounds of Preferred 89 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(91) Compounds of Preferred 90 where Q is Q₁.

(92) Compounds of Preferred 90 where Q is Q₂.

(93) Compounds of Preferred 90 where Q is Q₃.

(94) Compounds of Preferred 90 where Q is Q₄.

(95) Compounds of Preferred 90 where Q is Q₅.

(96) Compounds of Preferred 90 where Q is Q₆.

(97) Compounds of Preferred 90 where Q is Q₇.

(98) Compounds of Preferred 7 where J is J-11.

(99) Compounds of Preferred 98 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(100) Compounds of Preferred 99 where Q is Q₁.

(101) Compounds of Preferred 99 where Q is Q₂.

(102) Compounds of Preferred 99 where Q is Q₃.

(103) Compounds of Preferred 99 where Q is Q₄.

(104) Compounds of Preferred 99 where Q is Q₅.

(105) Compounds of Preferred 99 where Q is Q₆.

(106) Compounds of Preferred 99 where Q is Q₇.

(107) Compounds of Preferred 7 where J is J-12.

(108) Compounds of Preferred 107 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(109) Compounds of Preferred 108 where Q is Q₁.

(110) Compounds of Preferred 108 where Q is Q₂.

(111) Compounds of Preferred 108 where Q is Q₃.

(112) Compounds of Preferred 108 where Q is Q₄.

(113) Compounds of Preferred 108 where Q is Q₅.

(114) Compounds of Preferred 108 where Q is Q₆.

(115) Compounds of Preferred 108 where Q is Q₇.

(116) Compounds of Preferred 7 where J is J-13.

(117) Compounds of Preferred 116 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(118) Compounds of Preferred 117 where Q is Q₁.

(119) Compounds of Preferred 117 where Q is Q₂.

(120) Compounds of Preferred 117 where Q is Q₃.

(121) Compounds of Preferred 117 where Q is Q₄.

(122) Compounds of Preferred 117 where Q is Q₅.

(123) Compounds of Preferred 117 where Q is Q₆.

(124) Compounds of Preferred 117 where Q is Q₇.

(125) Compounds of Preferred 2 where

m is 0;

n is 0;

J is J-1, J-2, J-3, J-8, J-10 or J-11;

W is O;

R is H;

R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H;

R₃ is H, C₁ -C₃ alkyl, CH₂ CH₃ OCH₃, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, alyl or propargyl;

R₄ is H or C₁ -C₃ alkyl;

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; and

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(126) Compounds of Preferred 3 where

m is 0;

R is H;

R₁ is H;

R₃ is H or C₁ -C₃ alkyl;

R₄ is H or C₁ -C₃ alkyl;

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; and

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

Specifically preferred for reasons of greatest ease of synthesis and/or greatest herbicidal efficiency are:

N-[(4-chloro-6-methoxypyrimidin-2-yl)aminocarbonyl]-2-(1-ethyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 223°-225° C.;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-methyl-6-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 178°-189° C.;

N-[(4-chloro-6-methoxypyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 225°-227° C.;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 207°-210° C.;

N-[(4,6-dimethylpyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 224°-226° C.;

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole-5-sulfonamide, m.p. 181°-183° C.;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole-5-sulfonamide, m.p. 171°-173° C.;

N-[[N-4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide, m.p. 180°-182° C.; and

N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide, sodium salt, NMR (CDCl₃) δ 8.4-8.13 (m, 1H), 7.70-7.40 (m, 1H), 7.25-7.00 (m, 1H), 3.85 (s, 6H), 3.19 (s, 3H), 2.32 (s, 3H).

DETAILED DESCRIPTION OF THE INVENTION Synthesis

Compounds of Formula I can be synthesized by one or both of the methods shown below in Equation 1 and 2.

Equation 1 illustrates the reaction of sulfonyl isocyanates and isothiocyanates of Formula II with the appropriate heterocyclic amines of Formula III to give the desired sulfonylureas and sulfonylthioureas of Formula I. ##STR23## wherein J, W, R, and A are as previously defined.

The reaction of Equation 1 is best carried out in an inert aprotic solvent such as methylene chloride, tetrahydrofuran or acetonitrile at a temperature between 0° and 82° C. A catalytic amount of 1,4-diazabicyclo[2,2,2]octane (DABCO®) may be used to accelerate the reaction. In cases in which the products are insoluble in the reaction solvent, they may be isolated by simple filtration. When the products are soluble, they can be isolated by evaporation of the solvent and trituration of the residue with solvents such as 1-chlorobutane, diethyl ether or ethyl acetate, and filtration.

Compounds of Formula I can be prepared as shown below in Equation 2 by the reaction of sulfonamides IV with the phenyl ester of the appropriate carbamic acid or thiocarbamic acid of Formula V, in the presence of an equimolar quantity of a tertiary amine base such as 1,8-diazabicyclo[5,4,0]undec-7-ene (DBU). ##STR24## wherein J, R, W and A are as previously defined.

The reaction shown in Equation 2 is best carried out at 25° C. in a solvent such as dioxane or acetonitrile for 1-2 hours under an inert atmosphere as described in European Patent Application No. 70,804 (published Jan. 26, 1983). The desired products of Formula I can be conveniently isolated by acidifying the reaction solution with aqueous hydrochloric acid. Alternatively, the aqueous layer can be extracted with a solvent such as methylene chloride or ethyl acetate. Drying and evaporation of the solvent affords the desired products.

The phenylcarbamates and phenylthiocarbamates of Formula V can be prepared by methods, or modifications thereof known to those skilled in the art, described in South African Patent Application No. 82/5671 and South African Patent Application No. 82/5045.

A judicious choice of the appropriate methods for preparing compounds of Formula I must take into account the nature of the substituents contained within the J values (J₁ -J₆), namely Q and R₁, and their chemical compatibility with the reactive conditions of Equations 1 and 2.

Sulfonyl isocyanates of Formula II can be prepared as shown in Equation 3 by the reaction of sulfonamides of the general structure IV with phosgene in the presence of n-butyl isocyanate and a catalytic amount of 1,4-diazabicyclo[2.2.2]octane (DABCO). ##STR25## wherein J is as previously defined, provided E is not oxygen.

The reaction depicted in Equation 3 is best carried out according to the procedure described in U.S. Pat. No. 4,238,621.

Alternatively, sulfonyl isocyanates II can be prepared via phosgenation of the preformed n-butylureas of Formula VI as represented in Equation 4. ##STR26## wherein J is as previously defined, provided E is not oxygen.

The compounds of Formula VI are conveniently prepared by stirring a mixture of the appropriate sulfonamide IV, anhydrous potassium carbonate, and n-butyl isocyanate in a suitable solvent such as acetone or methyl ethyl ketone at 25° to 80° C. until all of the isocyanate has reacted. The products are isolated by quenching in dilute aqueous acid and recrystallizing the insoluble solid. The n-butylureas VI are then treated with phosgene and a catalytic amount of DABCO in refluxing xylenes or chlorobenzene in a manner analogous to that described in the reference cited for Equation 3.

Alternatively, treatment of the sulfonamides of Formula IV with thionyl chloride gives intermediate N-sulfinylsulfonamides VII, which afford sulfonylisocyanates II (where W is O) upon exposure to phosgene in the presence of a catalytic amount of pyridine. ##STR27##

The reaction of Equation 5 can best be performed according to the procedure of H. Ulrich, B. Tucker and A. Sayigh, J. Org. Chem., 34, 3200 (1969).

Sulfonyl isothiocyanates II (where W is S) are known in the art and are prepared from the corresponding sulfonamides (IV) by reaction with carbon disulfide and potassium hydroxide followed by treatment of the resulting dipotassium salt with phosgene. Such a procedure is described in Arch. Pharm. 299, 174 (1966).

A judicious choice of the appropriate method for preparing compounds of Formula II must taken into account the nature of the substituents contained within the J values (J₁ -J₆), namely Q and R₁, and their chemical compatability with the reaction conditions of Equations 3-5.

The required sulfonamides of Formula IV can be synthesized by one or more of the methods shown below.

Equation 6 depicts the reaction of sulfonyl chlorides of Formula VIII with ammonia to give sulfonamides of Formula IVa. ##STR28## wherein J is as previously defined, provided E is not oxygen.

The amination of Equation 6 can be effected by adding at least two molar equivalents of either anhydrous ammonia or concentrated ammonium hydroxide to a solution of the sulfonyl chloride VIII in a solvent such as diethyl ether, methylene chloride, or tetrahydrofuran at temperatures between -30° and 25° C. The sulfonamides of Formula IVa are isolated either by filtration, in which case the ammonium chloride byproduct is removed by washing with water, or extraction into an organic solvent such as methylene chloride. Drying and evaporation of the solvent afford the sulfonamides IVa, which are usually sufficiently pure to be carried directly on to the next step.

Sulfonyl chlorides of Formula VIII can be prepared by one or more of the methods shown below in Equations 7, 8 and 9.

The reaction of an appropriately substituted N-arylhydroxylamine of Formula IX, as shown in Equation 7, and subsequent displacement with sulfur dioxide in the presence of cupric or cuprous chloride yields the desired sulfonyl chloride of Formula VIII. ##STR29##

The reaction of Equation 7 can be carried out by combining the appropriate arylhydroxylamine with aqueous concentrated hydrochloric acid and acetic acid and adding an aqueous solution of sodium nitrite at -10° to 10° C. After being stirred for 10 minutes to two hours the reaction mixture is added to a mixture of acetic acid, a catalytic amount of cuprous or cupric chloride and excess sulfur dioxide at -5° to 20° C. After being stirred for 0.5 to 24 hours the mixture is diluted with cold water and the product is extracted into a solvent such as methylene chloride or ethyl ether.

The solution of sulfonyl chloride thus obtained can be treated as in Equation 6 to prepare the desired sulfonamide IVa.

Diazotization of appropriately substituted amine derivatives of Formula X, as shown in Equation 8, and subsequent reaction with sulfur dioxide in the presence of either cupric or cuprous chloride gives the desired products of Formula VIII. ##STR30##

The reaction of Equation 8 can be effected by methods analogous to those described in EP-A-Nos. 83,975 and 85,476 (published Aug. 10, 1983). In Equation 8, a substituted amine X, in concentrated hydrochloric acid is treated with a solution of sodium nitrite in water at -5° to 5° C. After being stirred for 10 minutes to one hour at about 0° C., the solution is added to a mixture of excess sulfur dioxide and a catalytic amount of cupric or cuprous chloride in acetic acid at about 10° C. After being stirred for 0.25 to 24 hours at temperatures between 10° to 25° C., the solution is poured into a large excess of ice water. The sulfonyl chloride VIII can be isolated by filtration, or by extraction into a solvent such as methylene chloride or ether, followed by drying and evaporation of the solvent.

Alternatively, diazotization of appropriately substituted amine hydrochloride salts of Formula Xa can be effected under anhydrous conditions, as shown in Equation 8a, and subsequent reaction with sulfur dioxide and cupric chloride gives the desired products of Formula VIII. ##STR31##

The amine hydrochloride salts Xa are diazotized with an alkylnitrite in a suitable solvent such as acetonitrile or acetone, and the resulting diazonium salts are reacted with sulfur dioxide and cupric chloride to give sulfonyl chlorides VIII. M. Doyle, in J. Org. Chem. 42, 2426, 2431 (1977), decribes conditions for conducting similar Meerwein reactions.

Sulfonyl chlorides can also be prepared as shown below in Equation 9 by metal halogen exchange or directed lithiation of appropriately substituted aryl or heterocyclic substrates XI, and trapping with sulfuryl chloride. ##STR32## wherein J is as previously described provided that R₁ is not CO₂ R_(c), C₁ -C₃ haloalkyl, Br, nitro, C₁ -C₃ alkylsulfonyl or CN.

The lithiation shown in Equation 9 can be performed according to the procedure of S. H. Bhattacharya, et al., J. Chem. Soc. (C), 1265 (1968) or by procedures reviewed by H. Gschwind and H. Rodriquez in Organic Reactions, Vol. 26, Wiley, New York, 1979, and references cited within.

Compounds of Formula VIII can be prepared via oxidative chlorination of the appropriate thioethers or mercaptans of Formula XII as represented in Equation 10. ##STR33## wherein J is as previously defined, R₁₅ is H, C₂ -C₄ alkyl or benzyl, R₁ is not C₁ -C₃ alkylthio or C₁ -C₃ alkylsulfinyl, and R₄ is not C₁ -C₄ alkylthio or C₁ -C₄ alkylsulfinyl.

The reaction of Equation 10 can be carried out by treating a solution of the thioether XII in a solvent such as acetic acid in the presence of at least 2.5 equivalents of water and at least 3.0 equivalents of chlorine at 0°-30° C. for 0.25 to 5 hours. The raction is poured into ice-water and the product is isolated by extraction with a suitable solvent such as methylene chloride, dried, and the solvent evaporated to yield a product sufficiently pure to be carried directly on to the next step.

Arylmethanesulfonyl chlorides of Formula VIIIb can be prepared from appropriately substituted benzyl chlorides or bromides of Formula XIII by a simple two-step procedure outlined in Equation 11. ##STR34## wherein J'CH₂ is defined as for J-1 through J-6 where E is CH₂ ;

R₁, R₄ and Q are as previously defined except R₁ is not C₁ -C₃ alkylthio or C₁ -C₃ alkylsulfinyl, and R₄ is not C₁ -C₄ alkylthio or C₁ -C₄ alkylsulfinyl; and

M is Cl or Br.

The conversion of alkylhalides of Formula XIII to isothiouronium salts of Formula XIV can be carried out by the procedure or T. B. Johnson and J. M. Sprague, J. Am. Chem. Soc., 58, 1348 (1936); 59 1837 and 2439 (1937); 61 176 (1939). Oxidative chlorination of isothouronium salts such as XIV to afford sulfonyl chlorides of Formula VIIIb is best carried out according to the procedure of Johnson as described in J. Am. Chem. Soc., 61 2548 (1939).

The requisite tetrazole substituted intermediates can be prepared by various methods depending on the nature of the aromatic ring in J (J-1 to J-6) systems on which the tetrazole is substituted and the nature of the other substituents present on J (J-1 to J-6). These intermediates can be prepared by one skilled in the art by the methods referred to in the following reviews on tetrazole chemistry: F. R. Benson, "Heterocyclic Compounds" (R. C. Elderfield, Ed.) 8, 1-104, John Wiley and Sons, New York, (1967); R. N. Butler, "Advances in Heterocyclic Chem.", 21, 323-436, Academic Press (1977); R. N. Butler, "Comprehensive Heterocyclic Chem.", (K. T. Potts, Ed.) 5, 791-838, Pergamon Press (1984) and F. R. Benson, "High Nitrogen Compounds", John Wiley and Sons, New York (1983).

The heterocyclic amines of Formula III in Equation 1 above can be prepared by methods known in the literature, or simple modifications thereof, by those skilled in the art. For instance, EP-A-No. 84,224 (published July 27, 1983) and W. Braker et al., J. Am. Chem. Soc., 69, 3072 (1947) describes methods for preparing aminopyridines and triazines substituted by acetal groups such as dialkoxymethyl or 1,3-dioxolan-2-yl, among other groups. Also, for example, South African patent application Nos. 82/5045 and 82/5671 describe methods for preparing aminopyridines and triazines substituted by haloalkyl or haloalkylthio groups such as OCH₂ CH₂ F, OCH₂ CF₃, SCF₂ H, or OCF₂ H, among other groups. South African patent application No. 83/7434 (published Oct. 5, 1983) describes methods for the synthesis of cycopropylpyrimidines and triazines substituted by such groups as alkyl, haloalkyl, alkoxy, haloalkoxy, alkylamino, dialkylamino or alkoxyalkyl.

The 5,6-dihydrofuro[2,3-d]pyrimidin-2-amines, the cyclopenta[d]pyrimidin-2-amines (III, A is A-2) and the 6,7-dihydro-5H-pyrano[2,3-d]pyrimidin-2-amines (III, A is A-3) can be prepared as described in EP-A-No. 15,683. The furo[2,3-d]pyrimidin-2-amines (III, A is A-4) are described in EP-A-No. 46,677.

Compounds of Formula III, where A is A-5, are described in EP-A-No. 73,562. Compounds of Formula III, where A is A-6 are described in EP-A-No. 94,260.

In addition, general methods for preparing aminopyridimidines and triazines have been reviewed in the following publications:

"The Chemistry of Heterocyclic Compounds", a series published by Interscience Publishers, Inc., New York and London;

"Pyrimidines", Vol. 16 of the same series by D. J. Brown;

"s-Triazines and Derivatives", Vol. 13 of the same series by E. M. Smolin and L. Rappoport; and

F. C. Schaefer, U.S. Pat. No. 3,154,547 and K. R. Huffman and F. C. Schaefer, J. Org. Chem., 28, 1812 (1963), which describes the synthesis of triazines.

Agriculturally suitable salts of compounds of Formula I are also useful herbicides and can be prepared in a number of ways known to the art. For example, metal salts can be made by contacting compounds of Formula I with a solution of an alkali or alkaline earth metal salt having a sufficiently basic anion (e.g., hydroxide, alkoxide or carbonate). Quaternary amine salts can be made by similar techniques.

A particularly useful process for preparing salts of compounds of Formula I involves reaction of a solution of the sulfonylurea in a water-immiscible halogenated hydrocarbon solvent with the appropriate alkali or alkaline earth metal hydroxide as described in copending application, U.S. Ser. No. 086,867 filed on Aug. 19, 1987.

Salts of compounds of Formula I can also be prepared by exchange of one cation for another. Cationic exchange can be effected by direct contact of an aqueous solution of a salt of a compound of Formula I (e.g. alkali or quaternary amine salt) with a solution containing the cation to be exchanged. This method is most effective when the desired salt containing the exchange cation is insoluble in water and can be separated by filtration.

Exchange may also be effected by passing an aqueous solution of a salt of a compound of Formula I (e.g., an alkali metal or quaternary amine salt) through a column packed with a cation exchange resin containing the cation to be exchanged for that of the original salt and the desired product is eluted from the column. This method is particularly useful when the desired salt is water-soluble, e.g. a potassium, sodium or calcium salt.

Acid addition salts, useful in this invention, can be obtained by reacting a compound of Formula I with a suitable acid, e.g., p-toluenesulfonic acid, trichloroacetic acid or the like.

The preparation of the compounds of this invention is further illustrated by the following specific examples.

EXAMPLE 1 1-(2-Chlorosulfonylphenyl)-5-methyl-1H-tetrazole

To 5 g of 1-(2-hydroxylaminophenyl)-5-methyl-1H-tetrazole in 12 mL of 37% hydrochloric acid and 5 mL of acetic acid at 0°-5° C. was added 2.3 g of sodium nitrite in 10 mL of water. The resultant solution was stirred at -5° to +5° C. for one hour and then added portionwise, with stirring, to a mixture of 25 mL of acetic acid, 0.5 g of cupric chloride and 5 mL of liquified sulfur dioxide at below 5° C. After stirring for two hours, during which time the mixture was allowed to warm to room temperature, it was poured into 150 mL of ice and water and extracted twice with 150 mL of methylene chloride. The methylene chloride solution was washed three times with 100 mL portions of water, two times with 100 mL of saturated aqueous sodium bicarbonate followed by single washes with 100 mL of saturated aqueous sodium chloride and 100 mL of water. The methylene chloride solution was then dried over magnesium sulfate and filtered to yield a solution containing the desired sulfonylchloride. This solution was used without further work-up to prepare the sulfonamide of Example 2.

EXAMPLE 2 1-(2-Aminosulfonylphenyl)-5-methyl-1H-tetrazole

Twenty-five mL of 28% ammonium hydroxide was added to the methylene chloride solution obtained from Example 2 and the mixture was stirred for two hours and concentrated in vacuo to yield a mixture of an oil and a solid. The solid product was separated by filtration and washed with water to yield 2.2 g of the desired product, which melted at 141°-148° C. Infrared absorption peaks at 3260 and 3360 cm⁻¹ were consistent for NH₂ and 1160 and 1350 cm⁻¹ consistent for the SO₂ of the desired product. Elem. anal. calc'd for C₈ H₉ N₅ O₂ S:C, 40.15; H, 3.79; N, 29.26, S, 13.39. Found: C, 40.43; H, 3.84; N, 29.61; S, 13.04.

EXAMPLE 3 5-(2-Chlorosulfonylphenyl)-2-methyl-2H-tetrazole and 5-(2-chlorosulfonylphenyl)-1-methyl-1H-tetrazole

To 5 g of a mixture of 5-(2-hydroxylaminophenyl)-2-methyl-2H-tetrazole and 5-(2-hydroxyaminophenyl)-1-methyl-1H-tetrazole dissolved in 12 mL of 37% hydrochloric acid and 5 mL of acetic acid was added with stirring 2.3 g of sodium nitrite dissolved in 10 mL of water at -5° to 5° C. After one hour this solution was added, at 0°-5° C., portionwise to a mixture of 25 mL of acetic acid, 0.5 g of cupric chloride and 5 mL of liquified sulfur dioxide. After the addition was completed the cooling bath was removed and the reaction mixture was allowed to warm to 31° C. whereupon the cooling bath was reapplied and the stirring was continued until two and one half hours after completion of the addition. The mixture was then poured into ice and worked up as described in Example 1 except that the desired methylene chloride solution was concentrated in vacuo to yield an oil which solidified. This product, (3.28 g) which was a mixture of the desired sulfonylchlorides, was of sufficient purity for the preparation of the sulfonamides of Example 4.

EXAMPLE 4 5-(2-Aminosulfonylphenyl)-2-methyl-2H-tetrazole and 5-(2-aminosulfonylphenyl)-1-methyl-1H-tetrazole

The solid product obtained in Example 3 was dissolved in 50 mL of tetrahydrofuran and added portionwise to 20 mL of 28% ammonium hydroxide. The mixture was stirred for one hour and concentrated in vacuo. Water was added to the residue, the mixture filtered and the solid washed with a small amount of cold water to yield 1.3 g of the isomer mixture. Infrared absorption spectra showed peaks at 3260 and 3360 cm⁻¹ consistent for NH₂ and 1160 and 1330 consistent for the SO₂ group of the desired product. Elem. anal. calc'd. for C₈ H₉ N₅ O₂ S:C, 40.15; H, 3.79; N, 29.26; S, 13.39. Found: C, 40.49; H, 3.86; N, 29.99; S, 13.75.

EXAMPLE 5 5-(2-Aminosulfonylphenyl)-1-methyl-1H-tetrazole

To 4.4 g of 5-(2-ethylthiophenyl)-1-methyl-1H-tetrazole in 40 mL of propionic acid and 1.08 g of water at -10° C. was added slowly, dropwise, 5.2 mL, of liquid chlorine (1.367 g/mL). After the addition the mixture was allowed to warm to room temperature, and was then poured into approximately 100 g of ice. The resultant sulfonyl chloride was extracted with methylene chloride, washed with water and the methylene chloride solution added to 45 mL of concentrated aqueous ammonium hydroxide while maintaining the reaction temperature below 25° C. with ice bath cooling. Evaporation of the methylene chloride yielded a solid product which was removed by filtration from the aqueous residue and washed with water. The product, 3.72 g, melted at 176°-179° C. and showed absorption peaks by infrared spectroscopy at 3210 and 3300 cm⁻¹, consistent for the desired sulfonamide.

EXAMPLE 6 5-(2-Aminosulfonyl-4-methylphenyl)-1-methyl-1H-tetrazole

To a mixture of 4.68 g of 5-(4-methyl-2-propylthiophenyl)-1-methyl-1H-tetrazole, 40 mL of propionic acid and 1.08 g of water cooled to -10° C. was added dropwise 5.2 mL (liquified) of chlorine while maintaining the reaction temperature at -10° to 0° C. After one-half hour the reaction mixture was allowed to warm to room temperature and stirred for one hour. It was then poured into 200 mL of ice and water and extracted with methylene chloride. The methylene chloride solution was added to 45 mL of concentrated ammonium hydroxide at 10° C. and stirred overnight. The mixture was concentrated in vacuo to an oil residue which was taken up in 100 mL of methylene chloride washed with three 100 mL portions of water and 100 mL of saturated aqueous sodium hydroxide. The methylene chloride solution was then dried over magnesium sulfate, filtereed, and the filtrate evaporated to yield 4.1 g of the desired product melting at 161°-171° C.

NMR (CDCl₃): δ 2.56 (s, CH₃ on phenyl); 3.99 (s, CH₃ on tetrazole); 5.6 (s, w, NH₂); and 7.3-8.1 (m, 3CH on phenyl).

EXAMPLE 7 5-(2-Aminosulfonyl-3-methylphenyl)-1-methyl-1H-tetrazole

To a mixture of 14.6 mL of concentrated (12M) hydrochloric acid, 6.1 mL of acetic acid, 25 mL of ethyl ether and 6.91 g of 5-(2-amino-3-methylphenyl)-1-methyl-1H-tetrazole at 0° C. was added dropwise 2.8 g of sodium nitrite dissolved in 12.2 mL of water while maintaining the reaction temperature at below 10° C. Stirring was continued for one hour after the addition was completed. This mixture was then added slowly to 30.5 mL of acetic acid containing 0.6 g of cupric chloride and 6.1 mL of liquified sulfur dioxide. After stirring for two hours at ambient temperature, the mixture was poured into 200 mL of ice-water and extracted twice with 125 mL of methylene chloride. The organic phase was then washed twice with 200 ml of water, once with 200 mL saturated aqueous sodium chloride, once with 200 mL aqueous sodium bicarbonate followed by 200 mL of water and 200 mL saturated aqueous sodium chloride. The organic phase was then added dropwise to 25 mL of concentrated aqueous ammonium hydroxide and the mixture stirred overnight and evaporated to a solid, which was washed with water and dried. The crude product thus obtained melted at 140°-161° C., yield 6.26 g. Mass spectral analysis showed a molecular weight of 253 (calc. 253) for the product.

EXAMPLE 8 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(2-methyl-2H-tetrazol-5-yl)benzenesulfonamide

To 25 mL of acetonitrile was added at ambient temperature and pressure 0.48 g of 5-(2-aminosulfonylphenyl)-2-methyl-2H-tetrazole and 0.54 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate followed by 0.3 mL of DBU. After being stirred for three hours the reaction mixture was added to 25 g of ice and acidified to pH 3 with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried to yield 0.66 g of the desired product, m.p. 214°-222° C. Infrared absorptions at 1720, 1600 and 1580 cm⁻¹ were consistent with the desired structure.

NMR(CDCl₃): δ 3.91 (s, 2×CH₃ O), 5.82 (s, CH, pyrimidin), 4.43 (s, CH₃ on N-2 of tetrazole), 4.38 (s, CH₃ on N-1 of tetrazole).

Integration of the peaks at 4.43 d and 4.38 d total one CH₃ indicating a ratio of 2-methyl-2H-tetrazole to 1-methyl-1H-tetrazole of 2:1. This mixture is suitable for purposes of this invention. If desired, the isomer mixture obtained in Example 6 can be separated by chromatography into its component parts.

EXAMPLE 9 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide

To 0.48 g of 1-(2-aminosulfonylphenyl)-5-methyl 1H-tetrazole in 25 mL of acetonitrile was added at ambient temperature and pressure 0.54 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate and 0.3 mL of DBU. The reaction mixture was stirred for three hours, added to 25 g of ice and acidified to pH 3 with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried to yield 0.74 g of the desired product, melting point at 213°-216° C. Infrared absorption spectra showed peaks at 1710, 1605 and 1570 cm⁻¹, consistent for the desired product.

NMR(CDCl₃): δ2.48 (s, CH₃ on tetrazole), 3.82 (s, 2×CH₃ O), 5.81 (s, CH-pyrimidin).

EXAMPLE 10 N-[(4-Methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide

To 0.48 g of 1-(2-aminosulfonylphenyl)-5-methyl-1H-tetrazole and 0.52 g of phenyl N-(4-methoxy-6-methyl-1,3,5-triazin-2-yl)carbamate in 25 mL of acetonitrile at ambient temperature and pressure was added 0.3 mL of DBU. The mixture was stirred for three hours and then added to 25 g of ice and acidified with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried in vacuo to yield 0.65 g of the desired product melting at 207°-209° C. Infrared absorption spectra showed absorption at 1700, 1600 and 1550 cm⁻¹, consistent for the desired structure.

EXAMPLE 11 N-[(4-chloro-6-methoxypyrimidine-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide

To 0.48 g of 5-(2-aminosulfonylphenyl)-1-methyl-1H-tetrazole and 0.56 g of phenyl N-(4-chloro-6-methoxypyrimidine-2-yl)carbamate in 20 mL of dry acetonitrile at ambient temperature was added, with stirring, 0.3 mL of DBU. After stirring 16 hours the mixture was then poured into 25 g of ice followed by the addition of 10 mL of 2N hydrochloric acid. The precipitate thus formed was removed by filtration, washed with water and dried to yield 0.74 g of the desired product, m.p. 225°-227° C.

NMR (CDCl₃): δ 3.88 (s, CH₃ on tetrazole); 3.95 (s, CH₃ O); 6.52 (s, CH of pyrimidine); 7.2-7.5 (m, CH of phenyl and NH); 7.84 (m, 2CH of phenyl); 8.6 (m, CH of phenyl); and 11.96 (s, NH).

EXAMPLE 12 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-5-chloro-2-(4-methyl-5-oxo-1H,4H-tetrazol-5-yl)-benzenesulfonamide

To a stirred solution of 0.29 g of 1-(2-aminosulfonyl-5-chlorophenyl)-4-methyl-1H-tetrazol-5[4H]-one and 0.27 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate in 10 mL of acetonitrile at ambient temperature was added 0.1 mL of DBU. The mixture was stirred for two hours, poured into 20 g of ice and acidified with 2N hydrochloric acid. The precipitate was removed by filtration, washed with water and dried to yield 0.37 g of product, m.p. 178°-180° C.

NMR (CDCl₃): δ 3.63 (s, CH₃ on tetrazole); 3.92 (s, 2×CH₃ O); 5.81 (s, CH of pyrimidine); 7.4-8.6 (m, 3CH of phenyl); and 12.6 (s, w, NH).

EXAMPLE 13 3-(2-Methyl-2H-tetrazole-5-yl)-1-phenyl-1H-pyrazole-5-sulfonamide

To a mixture of 3.1 mL of 12N hydrochloric acid, 12.5 mL of acetic acid, 3.7 mL of formic acid and 4.5 g of 5-amino-1-phenyl-3-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole was added dropwise 1.4 g of sodium nitrite in 2.5 mL of water at -8° to -6° C. The mixture was stirred for 15 minutes and then added to 20 mL of acetic acid containing 3.7 mL (liquid) of sulfur dioxide and 0.75 g of cupric chloride dihydrate. After stirring for thirty minutes and allowing to warm to room temperature, the mixture was poured into an ice and water mixture and the precipitate removed by filtration. After washing with water the solid was dissolved in tetrahydrofuran, cooled to -78° C., and ammonia (liquified, 1.0 mL) was added dropwise. The mixture was allowed to stand overnight at ambient temperature and filtered to yield a brown solid. This solid showed peaks at 3300 and 3200 cm⁻¹, consistent for NH₂, and 1370, 1185 and 1170 cm⁻¹, consistent for SO₂.

EXAMPLE 14 N-[[N-(4,6-Dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)-benzenesulfonamide

To 0.22 g of 2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide (compound of Example 2, 0.32 g) and 0.32 g of phenyl (4,6-dimethoxy-1,3,5-triazin-2-yl)(methyl)carbamate in 4 ml of dry acetonitrile was added at room temperature 0.2 ml of DBU. The reaction mixture was allowed to stand for four days, then diluted with 4 ml of water, several ice chips and 4 ml of diethyl ether. After stirring this solution for one minute, the ether layer was removed by pipet and the remaining mixture was acidified by dropwise addition of 1N HCl. The resulting precipitate was filtered, washed with water and dried to give 0.32 g of a white solid, m.p. 180°-182° C. (d).

EXAMPLE 15 Preparation of the sodium salt of N-[[N-(4,6-Dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)-benzenesulfonamide

To a stirred suspension of the compound of Example 14 (16.87 g, 38.7 mmol) and sodium carbonate (36 g) in methylene chloride (400 g), was added 1.79 g of sodium hydroxide (powder, 44.7 mmol). The suspension was allowed to stir at ambient temperature (20°-25° C. ) for 16 hours before it was filtered. The filtrate was evaporated under reduced pressure using a rotary evaporator. A colorless solid (17.8 g, 38.7 mmol, 100% yield) was isolated;

NMR (90 MHz, CDCl₃): δ 8.4-8.13 (m, 1H); 7.70-7.40 (m, 1H); 7.25-7.00 (m, 1H); 3.85 (s, 6H); 3.19 (s, 3H); 2.32 (s, 3H).

By using the procedures described in the foregoing equations and examples or modifications thereof, one skilled in the art can prepare the compounds shown in the following tables. ##STR35##

                                      TABLE I                                      __________________________________________________________________________     General Structure 1                                                            R.sub.1  E  Q  R.sub.3    W     R  X      Y          Z  m.p.                   __________________________________________________________________________                                                             (°C.)           H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 224-226                H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH 222-224                H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 207-210                H        -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 225-227                H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N  196-198                H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  172-187                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              CH.sub.3   CH 200-207                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  CH 203-205                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  CH 214-217                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  Cl     OCH.sub.3  CH 223-225                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3 N  193-200                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  N  192-196                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  N  192-195                H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               cyclopentyl                                                                               O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               cyclopentyl                                                                               O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               cyclopentyl                                                                               O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               cyclopentyl                                                                               O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               cyclopentyl                                                                               O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               cyclopentyl                                                                               O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub. 2 Cl                                                            O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               (CH.sub.2 ).sub.2 SCH.sub.2 CH.sub.3                                                      O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 235-238                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH 233-234                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 213-216                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 217-219                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N  200-205                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  195-198                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 192-197                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  201-206                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   N  159-173                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH 219-222                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 223-226                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 181-186                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3 N  187-190                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   N  179-186                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 214-218                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH 225-229                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  191-196                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 182- 196               4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 140-150                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3 N  152-160                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  197-200                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   N  198-202                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 178-180                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH 180-183                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 213-215                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 196-199                5-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 221-223                5-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH 207-210                5-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 214-216                5-Cl     -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 203-205                5-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N  191-193                5-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  175-180                5-Cl     -- Q-1                                                                               CH.sub.3   O     H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3 N  144-158                5-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH(OCH.sub.3).sub.2                                                                       CH 180-183                5-Br     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-Br     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-Br     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-Br     -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        5-Br     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-Br     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 198-200                5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH 218-219                5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 205-207                5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 185-188                5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         6-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 159-164                6-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH 196-199                6-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 153-156                6-Cl     -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 166-170                6-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N  187-189                6-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  202-205                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 181-186                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub. 3  O     H  OCH.sub.3                                                                             CH.sub.3   CH 205-209                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 174-181                5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  Cl     OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub. 3                                                                            OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.3   S     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.3   S     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   S     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   S     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   S     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.3   S     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.3   O     H  H      OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H  H      OC.sub.2 H.sub.5                                                                          CH                        H        -- Q-1                                                                               CH.sub.3   O     H  H      OCF.sub.2 H                                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CF.sub.3   CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              SCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.2 OCH.sub.3                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.2 OCH.sub.3                                                                       CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              NHCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                         CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        O  Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        O  Q-1                                                                               CH.sub. 3  O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        O  Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        O  Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        O  Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        O  Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        O  Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        O  Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        H        O  Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        O  Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.3   O     H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H  H      OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H  H      OC.sub.2 H.sub.5                                                                          CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CF.sub.3   CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              SCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2   O     H  CH.sub.3                                                                              CH.sub.2 OCH.sub.3                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              NHCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                         CH                        H        -- Q-1                                                                               CH.sub.3   O     H  H      OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.3   O     H  H      OC.sub.2 H.sub.5                                                                          N                         H        -- Q-1                                                                               CH.sub.3   O     H  H      OCF.sub.2 H                                                                               N                         H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.2 OCH.sub.3                                                                        N                         H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              NHCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                         N                         3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CH.sub.2 CH.sub.2 Cl                                                                  -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CH.sub.2 CH.sub.2 Cl                                                                  -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        6-SO.sub.2 N(CH.sub.3).sub.2                                                            -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        6-SO.sub.2 N(CH.sub.3).sub.2                                                            -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        6-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        6-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        6-SCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        6-SCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        6-SOCH.sub.3                                                                            -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        6-SOCH.sub.3                                                                            -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        6-SO.sub.2 CH.sub.3                                                                     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        6-SO.sub.2 CH.sub.3                                                                     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CN     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CN     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CO.sub.2 CH.sub.3                                                                     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CO.sub.2 CH.sub.3                                                                     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-OCH.sub.2 CH.sub.2 Cl                                                                 -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-OCH.sub.2 CH.sub.2 Cl                                                                 -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-OCH.sub.2 CF.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-OCH.sub.2 CF.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-SCH.sub.2 CF.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-SCH.sub.2 CF.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-NH.sub.2                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-NH.sub.2                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-NHC.sub.2 H.sub.5                                                                     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-NHC.sub.2 H.sub.5                                                                     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-N(CH.sub.3).sub.2                                                                     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-N(CH.sub.3).sub.2                                                                     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-C.sub.2 H.sub.4 OCH.sub.3                                                             -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-C.sub.2 H.sub.4 OCH.sub.3                                                             -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-C.sub.2 H.sub.4 OC.sub.2 H.sub.5                                                      -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-C.sub.2 H.sub.4 OC.sub.2 H.sub.5                                                      -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CH.sub.2 OC.sub.2 H.sub.4 Cl                                                          -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CH.sub.2 OC.sub.2 H.sub.4 Cl                                                          -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CH.sub.2 OCH.sub.2 CF.sub.3                                                           -- Q-1                                                                               CH.sub. 3  O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CH.sub.2 OCH.sub.2 CF.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CH.sub.2 SCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CH.sub.2 SCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CH.sub.2 SC.sub.2 H.sub.4 Cl                                                          -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        5-CH.sub.2 SC.sub.2 H.sub.4 Cl                                                          -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CH.sub.2 CN                                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-CH.sub.2 CN                                                                           -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.2 CH.sub.2 CH.sub.2                                                    CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.2 CH.sub.2 Cl                                                                     CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.2 CH.sub.2 CH.sub.2                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             SCH.sub.2 CH.sub.2 Cl                                                                     CH                        H        -- Q-1                                                                               CH.sub. 3  O     H  OCH.sub.3                                                                             SCHF.sub.2 CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             SCH.sub.2 CH.sub.3                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             C.sub.2 H.sub.4 OC.sub.2                                                       H.sub.5    CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OC.sub.2 H.sub.4 OC.sub.2                                                      H.sub.5    CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.2 CH═CH.sub.2                                                                 CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.2 C.tbd.CH                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.2 SCH.sub.3                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             C.sub.2 H.sub.4 SCH.sub.3                                                                 CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             C.sub.2 H.sub.4 SC.sub.2                                                       H.sub.5    CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.2 SO.sub.2 CH.sub.3                                                                CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             C.sub.2 H.sub.4 SO.sub.2                                                       CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             C.sub.2 H.sub.4 SOCH.sub.3                                                                CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.2 CH.sub.2 CH.sub.2                                                                CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.2 C.tbd.CH                                                                         CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             N.sub.3    CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CN         CH                        H        -- Q-l                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             COCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             C(CH.sub.3)(OCH.sub.3).sub.2                                                              CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             2-methyldi-                                                                               CH                                                                  oxolan-2-yl                          H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             N(OCH.sub.3)CH.sub.3                                                                      CH                        H        -- Q-1                                                                               CH.sub.3   O     H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3 N  204-208                H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 214-222                H        -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-2                                                                               CH(CH.sub.3).sub. 2                                                                       O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H  Cl     OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCF.sub.2 H                                                                               CH 160-165                H        -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCF.sub.2 H                                                                               CH 195-198                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCF.sub.2 H                                                                               CH 168-172                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCF.sub.2 H                                                                               CH  90-93                 H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-OCF.sub. 2 H                                                                          -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         6-Cl     -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        6-Cl     -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        6-Cl     -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   CH                        6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              CH.sub.3   CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  Cl     OCH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  CH.sub.3                                                                              OCH.sub.3  N                         5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                          CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                          Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-2                                                                               CH.sub.3   S     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-2                                                                               CH.sub.3   S     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   S     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   S     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   S     H  CH.sub.3                                                                              OCH.sub.3  N                         H        -- Q-2                                                                               CH.sub.3   S     H  OCH.sub.3                                                                             OCH.sub.3  N                         H        -- Q-2                                                                               CH.sub.3   O     H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.3   O     H  H      OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H  H      OC.sub.2 H.sub.5                                                                          CH                        H        -- Q-2                                                                               CH.sub.3   O     H  H      OCF.sub.2 H                                                                               CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              SCF.sub.2 H                                                                               CH                        H        -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.2 OCH.sub.3                                                                        CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.2 OCH.sub.3                                                                       CH                        H        -- Q-2                                                                               CH.sub.3   O     H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.3   O     H  H      OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H  H      OC.sub.2 H.sub.5                                                                          CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CF.sub.3   CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              SCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.2 OCH.sub.3                                                                        CH                        H        -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.2 OCH.sub.3                                                                       CH                        H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OC.sub.2 H.sub.5                                                                          N                         H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH(CH.sub.3).sub.2                                                                       N                         H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.2 CF.sub.3                                                                        N                         H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CF.sub.3   N                         H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             O(CH.sub.2).sub.2 OCH.sub.3                                                               N                         H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             C.tbd.C--CH.sub.3                                                                         N                         H        -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             N(CH.sub.3)OCH.sub.3                                                                      N                         H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H  CH.sub.3                                                                              CH.sub.3   CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H  Cl     OCH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H  CH.sub.3                                                                              OCH.sub.3  N                         6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH                        6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH                        6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH                        6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.3   N                         6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  Br     OCH.sub.3  CH 196-198 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3  CH 199-200 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3  N   49-56                 6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  H      CH.sub.3   CH 196-199 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  H      OCH.sub.3  CH 163-166 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  C.sub.2 H.sub.5                                                                       OCH.sub.3  CH 160-164                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  C.sub.2 H.sub.5                                                                       OCH.sub.3  N  179-180 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3  N                         6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  cyclopropyl                                                                           OCH.sub.3  N  222-223 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OC.sub.2 H.sub.5                                                                          CH                        6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             CH.sub.2 OC.sub.2 H.sub.5                                                                 CH 189-190 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.2 CF.sub.3                                                                        CH 140-145 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OC.sub.2 H.sub.5                                                                          N  159-164 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCF.sub.2 H                                                                               CH 168-172                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCF.sub.2 H                                                                               CH  90-93                 H        -- Q-1                                                                               CH.sub.3   NH    H  OCH.sub.3                                                                             OCH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   NOCH.sub.3                                                                           H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   NOH   H  CH.sub.3                                                                              OCH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           NNHCH.sub.3                                                                          H  OCH.sub.3                                                                             OCH.sub.3  CH                        3-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  199-202                3-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N  206-209                3-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 143-162                3-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH 226-227                3-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 221-223 dec.           3-Cl     -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 189-192                5-F      -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  CH 209-212                5-F      -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 199-201                5-F      -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  187-190                5-F      -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N  196-201                5-F      -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              CH.sub.3   CH 233-236                5-F      -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  CH 164-168                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H  OCH.sub.3                                                                             OCF.sub.2 H                                                                               CH  87-94                 6-Cl     -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCF.sub.2 H                                                                               CH  93-95                 6-Cl     -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCF.sub.2 H                                                                               CH 118-120                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N  194-197                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N  172-182                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH 206-209                6-Cl     -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        6-Cl     -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         6-Cl     -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  Cl     OCH.sub.3  CH                        6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  OCH.sub.3                                                                             OCH.sub.3  N                         6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H  CH.sub.3                                                                              OCH.sub.3  N                         __________________________________________________________________________

                                      TABLE Ia                                     __________________________________________________________________________     General Structure 1                                                            R.sub.1                                                                               E  Q  R.sub.4 W R  X      Y       Z  m.p. (°C.)                  __________________________________________________________________________     H      -- Q-3                                                                               H       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 214 dec.                           H      -- Q-3                                                                               H       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 204-205                            H      -- Q-3                                                                               H       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 187-188                            H      -- Q-3                                                                               H       O H  Cl     OCH.sub.3                                                                              CH 195-196                            H      -- Q-3                                                                               H       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  199-202                            H      -- Q-3                                                                               H       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  191-192                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3                                                                             N  167-200 dec.                       H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 221-223                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 213-216                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH 208- 210                           H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  207-209                            H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  209-216                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 217-220                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 224-228                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 193-196                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  Cl     OCH.sub.3                                                                              CH 200-204                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  174-179                            H      -- Q-3                                                                               C.sub.2 H.sub.5                                                                        O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  194-197                            H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH(CH.sub.3).sub.2                                                                     O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               cyclopropyl                                                                            O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               cyclopropyl                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               cyclopropyl                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               cyclopropyl                                                                            O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               cyclopropyl                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               cyclopropyl                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 Cl                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CF.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CF.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CF.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 195-196                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 175-177                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 188-189                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH 200-201                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  189-190                            H      -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  180                                H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 199-200 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 197-198 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 200-201 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH 184-185 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  170-173 dec.                       H      -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  178-180 dec.                       H      -- Q-3                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               N(CH.sub.3).sub.2                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 177-186                            5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH 207-208                            5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  200-202                            5-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 227-230                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 173-180                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 216-220                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH 227-230                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  188-195                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  192-194                            5-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OC.sub. 2 H.sub.5                                                                     NHCH.sub.3                                                                             N  181-185                            5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              H                                     5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OCF.sub.2 H                                                                         -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub. 3                                                                             CH                                    5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-CF.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-SCH.sub.3                                                                           -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-CH.sub.2 OCH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    5-OCH.sub.2 CH.sub.3                                                                  -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OCH.sub.2 CH.sub. 3                                                                 -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 OCH.sub.3                                                                     O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.2 OCH.sub.3                                                                     O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 OCH.sub.3                                                                     O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 OCH.sub.3                                                                     O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3 OCH.sub.3                                                                     O H  OCH.sub.3                                                                             CH.sub.3                                                                               N                                     H      -- Q-3                                                                               CH.sub.3 OCH.sub.3                                                                     O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               O H  cyclopropyl                                                                           OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             N.sub.3 CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CN      CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             C(O)CH.sub.3                                                                           CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CH(OCH.sub.3).sub.2                                                                    CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             1,3-dioxo-                                                                             CH                                                                     lan-2-yl                                      H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             1,3-diox-                                                                              CH                                                                     an-2-yl                                       H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      CH.sub.2                                                                          Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      O  Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      O  Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      O  Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      O  Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      O  Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      O  Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               S H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               S H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               S H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub. 3                                                                              S H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               S H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               S H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.3                                                                               O CH.sub.3                                                                          OCH.sub.3                                                                             OCH.sub.3                                                                              N  180-182(d)                         H      -- Q-3                                                                               CH.sub.3                                                                               O H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3                                                                             CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  H      OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  H      OC.sub.2 H.sub.5                                                                       CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  H      OCF.sub.2 H                                                                            CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              SCF.sub.2 H                                                                            CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.2 OCH.sub.3                                                                     CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OC.sub.2 H.sub.5                                                                       CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CF.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             O(CH.sub.2).sub.2 OCH.sub.3                                                            CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             SCF.sub.2 H                                                                            CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             C.tbd.CH                                                                               CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             C.tbd.C--CH.sub.3                                                                      CH                                    H      -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             N(OCH.sub.3)CH.sub.3                                                                   CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               SCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               SCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               SCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               N(CH.sub.2).sub. 4                                                                     O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               N(CH.sub.2).sub.4                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  OCH.sub.3                                                                             CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               C.sub.6 H.sub.5                                                                        O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CF.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               CF.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CF.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CF.sub.3                                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               N                                     H      -- Q-4                                                                               CF.sub.3                                                                               O H  OC.sub.2 H.sub.5                                                                      NHCH.sub.3                                                                             N                                     H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-4                                                                               CH.sub.2 CH═CH.sub. 2                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               N                                     6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               N                                     6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             CH.sub.3                                                                               CH                                    6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 170-171                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 171-173                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 176-178                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  Cl     OCH.sub.3                                                                              CH 163-167                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  148-152                            H      -- Q-3                                                                               OC.sub.3 H.sub.7                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  158-160                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 181-184                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 188-190                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 166-168                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH 182-184                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  184-186                            5-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  175-178                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 180-181                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 188-191                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub. 5                                                                      O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 198-199                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH 184-186                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  204-206                            5-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  175-179                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH 192-193                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH 182-184                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH 181-183                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH 172-175                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N  167-170                            5-OCH.sub.3                                                                           -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N  174-176                            H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               OCF.sub.2 H                                                                            O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH                                    3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     3-CH.sub.3                                                                            -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    5-OC.sub. 2 H.sub.5                                                                   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH                                    5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-OC.sub.2 H.sub.5                                                                    -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub. 3                                                                             N                                     5-Br   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  Cl     OCH.sub.3                                                                              CH                                    5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     5-Br   -- Q-3                                                                               OC.sub.2 H.sub.5                                                                       O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SOCH.sub.3                                                                             O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               SO.sub.2 CH.sub.3                                                                      O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-3                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     6-CH.sub.3                                                                            -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                    6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              CH                                    6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              CH.sub.3                                                                               CH                                    6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  Cl     OCH.sub.3                                                                              CH                                    6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     6-Cl   -- Q-3                                                                               OCH.sub.3                                                                              O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     6-CH.sub.3                                                                            -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  CH.sub.3                                                                              OCH.sub.3                                                                              N                                     6-Cl   -- Q-3                                                                               CH.sub.3                                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  Cl     OCH.sub.3                                                                              CH                                    H      -- Q-4                                                                               CH.sub.2 CH═CH.sub.2                                                               O H  OCH.sub.3                                                                             OCH.sub.3                                                                              N                                     __________________________________________________________________________

                                      TABLE Ib                                     __________________________________________________________________________     General Structure 1                                                            R.sub.1                                                                              E Q  R.sub.5 W R X   Y    Z  m.p. (°C.)                           __________________________________________________________________________     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N  199-201                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 213-218                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H CH.sub.3                                                                           CH.sub.3                                                                            CH 185-189                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H CH.sub.3                                                                           OCH.sub.3                                                                           CH 201-206                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 191-209                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H Cl  OCH.sub.3                                                                           CH 196-199                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H CH.sub.3                                                                           OCH.sub.3                                                                           N  194-198                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H OCH.sub.3                                                                          OCH.sub.3                                                                           N  166-169                                     H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub. 5                                                                       O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N  202                                         H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 178-180                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH 134-140                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N  202                                         5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCF.sub.2 H                                                                         CH 196-198                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCF.sub.2 H                                                                         CH 162-166                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH 125-128                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N  70-112                                      5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N  190-194                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 153-157                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH 170-173                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH 141-143                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub. 3                                                                              O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              __________________________________________________________________________

                                      TABLE II                                     __________________________________________________________________________     General Structure 2                                                            R.sub.1                                                                             E Q  R.sub.3    W R X.sub.1                                                                             Y.sub.1                                                                           m.p. (°C.)                             __________________________________________________________________________     H    --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub. 5                                                                          O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OC.sub.2 H.sub.5                                                                    CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCF.sub.2 H                                                                         CH.sub.2                                         H    --                                                                               Q-1                                                                               (CH.sub.2).sub.5 CH.sub.3                                                                 O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               CH.sub.2 CH═CH--CH.sub.2 Cl                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-CN --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CN --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-2                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    CH.sub.2                                         H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-C.sub.2 H.sub.5                                                                   --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         __________________________________________________________________________

                  TABLE IIa                                                        ______________________________________                                         General Structure 2                                                                                                            m.p.                           R.sub.1                                                                               E     Q       R.sub.4                                                                              W   R    X.sub.1                                                                               Y.sub.1                                                                             (°C.)                   ______________________________________                                         H      --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   H      --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   H      --    Q-3     CH.sub.3                                                                             O   H    OC.sub.2 H.sub.5                                                                      O                                   H      --    Q-3     CH.sub.3                                                                             O   H    OCF.sub.2 H                                                                           O                                   H      --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              CH.sub.2                            H      --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             CH.sub.2                            H      --    Q-3     CH.sub.3                                                                             O   H    OC.sub.2 H.sub.5                                                                      CH.sub.2                            H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    CH.sub.3                                                                              O                                   H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    OCH.sub.3                                                                             O                                   H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    OC.sub.2 H.sub.5                                                                      O                                   H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    CH.sub.3                                                                              CH.sub.2                            H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    OCH.sub.3                                                                             CH.sub.2                            H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    OC.sub.2 H.sub.5                                                                      CH.sub.2                            H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    OCF.sub.2 H                                                                           CH.sub.2                            H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    OCH.sub.3                                                                             O                                   H      --    Q-3     C.sub.2 H.sub.5                                                                      O   H    OCH.sub.3                                                                             O                                   5-CH.sub.3                                                                            --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-CH.sub.3                                                                            --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             CH.sub.2                            5-Cl   --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-Cl   --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-Cl   --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   5-OCH.sub.3                                                                           --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-OCH.sub.3                                                                           --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   5-OC.sub.2 H.sub.5                                                                    --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-OC.sub.2 H.sub.5                                                                    --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   5-SCH.sub.3                                                                           --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-SCH.sub.3                                                                           --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   5-SC.sub.2 H.sub.5                                                                    --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-SC.sub.2 H.sub.5                                                                    --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   5-OCF.sub.2 H                                                                         --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-OCF.sub.2 H                                                                         --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   5-SCF.sub.2 H                                                                         --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   5-SCF.sub.2 H                                                                         --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   H      --    Q-4     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   H      --    Q-4     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   H      --    Q-4     CH.sub.3                                                                             O   H    OC.sub.2 H.sub.5                                                                      O                                   H      --    Q-4     CH.sub.3                                                                             O   H    OCF.sub.2 H.sub.5                                                                     O                                   H      --    Q-4     CH.sub.3                                                                             O   H    CH.sub.3                                                                              CH.sub.2                            H      --    Q-4     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             CH.sub.2                            H      --    Q-4     CH.sub.3                                                                             O   H    OC.sub.2 H.sub.5                                                                      CH.sub.2                            H      --    Q-4     CH.sub.3                                                                             O   H    OCF.sub.2 H                                                                           CH.sub.2                            H      --    Q-4     C.sub.2 H.sub.5                                                                      O   H    CH.sub.3                                                                              O                                   H      --    Q-4     C.sub.2 H.sub.5                                                                      O   H    OCH.sub.3                                                                             O                                   H      --    Q-4     C.sub.2 H.sub.5                                                                      O   H    OC.sub.2 H.sub.5                                                                      O                                   H      --    Q-4     C.sub.2 H.sub.5                                                                      O   H    OCF.sub.2 H                                                                           O                                   H      --    Q-4     C.sub.2 H.sub.5                                                                      O   H    CH.sub.3                                                                              CH.sub.2                            H      --    Q-4     C.sub.2 H.sub.5                                                                      O   H    OCH.sub.3                                                                             CH.sub.2                            H      --    Q-4     C.sub.2 H.sub.5                                                                      O   H    OC.sub.2 H.sub.5                                                                      CH.sub.2                            H      --    Q-4     C.sub.2 H.sub.5                                                                      O   H    OCF.sub.2 H                                                                           CH.sub.2                            6-CH.sub.3                                                                            --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             CH.sub.2                            6-CH.sub.3                                                                            --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   6-CH.sub.3                                                                            --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   6-Cl   --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             CH.sub.2                            6-Cl   --    Q-3     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   6-Cl   --    Q-3     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   6-CH.sub.3                                                                            --    Q-4     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             CH.sub.2                            6-CH.sub.3                                                                            --    Q-4     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   6-CH.sub.3                                                                            --    Q-4     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   6-Cl   --    Q-4     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             CH.sub.2                            6-Cl   --    Q-4     CH.sub.3                                                                             O   H    OCH.sub.3                                                                             O                                   6-Cl   --    Q-4     CH.sub.3                                                                             O   H    CH.sub.3                                                                              O                                   H      --    Q-3     H     O   H    OCH.sub.3                                                                             O                                   H      --    Q-3     H     O   H    CH.sub.3                                                                              O                                   H      --    Q-3     H     O   H    OCH.sub.3                                                                             CH.sub.2                            H      --    Q-3     H     O   H    CH.sub.3                                                                              CH.sub.2                            H      --    Q-3     OCH.sub.3                                                                            O   H    OCH.sub.3                                                                             O                                   H      --    Q-3     OCH.sub.3                                                                            O   H    CH.sub.3                                                                              O                                   H      --    Q-3     OCH.sub.3                                                                            O   H    OCH.sub.3                                                                             CH.sub.2                            H      --    Q-3     OCH.sub.3                                                                            O   H    CH.sub.3                                                                              CH.sub.2                            H      --    Q-3     OC.sub.2 H.sub.5                                                                     O   H    OCH.sub.3                                                                             O                                   H      --    Q-3     OC.sub.2 H.sub.5                                                                     O   H    CH.sub.3                                                                              O                                   H      --    Q-3     OC.sub.2 H.sub.5                                                                     O   H    OCH.sub.3                                                                             CH.sub.2                            H      --    Q-3     OC.sub.2 H.sub.5                                                                     O   H    CH.sub.3                                                                              CH.sub.2                            H      --    Q-3     SCH.sub.3                                                                            O   H    OCH.sub.3                                                                             O                                   H      --    Q-3     SCH.sub.3                                                                            O   H    CH.sub.3                                                                              O                                   H      --    Q-3     SCH.sub.3                                                                            O   H    OCH.sub.3                                                                             CH.sub.2                            H      --    Q-3     SCH.sub.3                                                                            O   H    CH.sub.3                                                                              CH.sub.2                            ______________________________________                                    

                  TABLE IIb                                                        ______________________________________                                         General Structure 2                                                            R.sub.1                                                                               E      Q      R.sub.5                                                                             W   R   X.sub.1                                                                              Y.sub.1                                                                             m.p. (°C.)                 ______________________________________                                         H      --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      H      --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               H      --     Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      H      --     Q-5    C.sub.2 H.sub.5                                                                     O   H   OCH.sub.3                                                                            O                                      H      --     Q-5    C.sub.2 H.sub.5                                                                     O   H   OCH.sub.3                                                                            CH.sub.2                               H      --     Q-5    C.sub.2 H.sub.5                                                                     O   H   CH.sub.3                                                                             O                                      5-CH.sub.3                                                                            --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      5-CH.sub.3                                                                            --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               5-CH.sub.3                                                                            --     Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      5-Cl   --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      5-Cl   --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               5-Cl   --     Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      6-CH.sub.3                                                                            --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      6-CH.sub.3                                                                            --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               6-CH.sub.3                                                                            --     Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      6-Cl   --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      6-Cl   --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               6-Cl   --     Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      5-F    --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      5-F    --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               5-F    --     Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      5-OCH.sub.3                                                                           --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            O                                      5-OCH.sub.3                                                                           --     Q-5    CH.sub.3                                                                            O   H   OCH.sub.3                                                                            CH.sub.2                               5-OCH.sub.3                                                                           --     Q-5    CH.sub.3                                                                            O   H   CH.sub.3                                                                             O                                      ______________________________________                                    

                  TABLE III                                                        ______________________________________                                         General Structure 3                                                                                                             m.p.                          R.sub.1                                                                              E     Q      R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                             W   R   X.sub.1                                                                              (°C.)                  ______________________________________                                         H     --    Q-1    CH.sub.3                                                                            --    --   O   H   CH.sub.3                            H     --    Q-1    CH.sub.3                                                                            --    --   O   H   OCH.sub.3                           H     --    Q-1    CH.sub.3                                                                            --    --   O   H   OC.sub.2 H.sub.5                    H     --    Q-1    CH.sub.3                                                                            --    --   O   H   OCF.sub.2 H                         H     --    Q-1    C.sub.2 H.sub.5                                                                     --    --   O   H   CH.sub.3                            H     --    Q-1    C.sub.2 H.sub.5                                                                     --    --   O   H   OCH.sub.3                           H     --    Q-1    C.sub.2 H.sub.5                                                                     --    --   O   H   OC.sub.2 H.sub.5                    H     --    Q-2    CH.sub.3                                                                            --    --   O   H   CH.sub.3                            H     --    Q-2    CH.sub.3                                                                            --    --   O   H   OCH.sub.3                           H     --    Q-2    CH.sub.3                                                                            --    --   O   H   OC.sub.2 H.sub.5                    H     --    Q-2    C.sub.2 H.sub.5                                                                     --    --   O   H   OCH.sub.3                           H     --    Q-2    C.sub.2 H.sub.5                                                                     --    --   O   H   CH.sub.3                            H     --    Q-3    --   CH.sub.3                                                                             --   O   H   OC.sub.2 H.sub.5                    H     --    Q-3    --   CH.sub.3                                                                             --   O   H   OCH.sub.3                           H     --    Q-3    --   CH.sub.3                                                                             --   O   H   CH.sub.3                            H     --    Q-3    --   C.sub.2 H.sub.5                                                                      --   O   H   CH.sub.3                            H     --    Q-3    --   C.sub.2 H.sub.5                                                                      --   O   H   OCH.sub.3                           6-CH.sub.3                                                                           --    Q-1    CH.sub.3                                                                            --    --   O   H   OCH.sub.3                           6-CH.sub.3                                                                           --    Q-1    CH.sub.3                                                                            --    --   O   H   CH.sub.3                            6-Cl  --    Q-1    CH.sub.3                                                                            --    --   O   H   CH.sub.3                            6-Cl  --    Q-1    CH.sub.3                                                                            --    --   O   H   OCH.sub.3                           H     --    Q-4    --   CH.sub.3                                                                             --   O   H   OCH.sub.3                           H     --    Q-5    --   --    CH.sub.3                                                                            O   H   OCH.sub.3                           H     --    Q-5    --   --    CH.sub.3                                                                            O   H   CH.sub.3                            H     --    Q-6    --   --    CH.sub.3                                                                            O   H   OCH.sub.3                           H     --    Q-7    --   --    CH.sub.3                                                                            O   H   OCH.sub.3                           H     --    Q-3    --   H     --   O   H   OCH.sub.3                           H     --    Q-3    --   H     --   O   H   CH.sub.3                            H     --    Q-3    --   OCH.sub.3                                                                            --   O   H   OCH.sub.3                           H     --    Q-3    --   OCH.sub.3                                                                            --   O   H   CH.sub.3                            H     --    Q-3    --   OC.sub.2 H.sub.5                                                                     --   O   H   OCH.sub.3                           H     --    Q-3    --   OC.sub.2 H.sub.5                                                                     --   O   H   CH.sub.3                            H     --    Q-3    --   SCH.sub.3                                                                            --   O   H   OCH.sub.3                           H     --    Q-3    --   SCH.sub.3                                                                            --   O   H   CH.sub.3                            ______________________________________                                    

                                      TABLE IV                                     __________________________________________________________________________     General Structure 4                                                            R.sub.1                                                                            E  Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W  R X.sub.1                                                                            Y.sub.3                                                                            m.p. (°C.)                             __________________________________________________________________________     H   -- Q-1                                                                               CH.sub.3                                                                          --  -- O  H CH.sub.3                                                                           H                                                 H   -- Q-1                                                                               CH.sub.3                                                                          --  -- O  H OCH.sub.3                                                                          H                                                 H   -- Q-1                                                                               CH.sub.3                                                                          --  -- O  H OC.sub.2 H.sub.5                                                                   H                                                 H   -- Q-1                                                                               CH.sub.3                                                                          --  -- O  H CH.sub.3                                                                           CH.sub.3                                          H   -- Q-1                                                                               CH.sub.3                                                                          --  -- O  H OCH.sub.3                                                                          CH.sub.3                                          H   -- Q-1                                                                               CH.sub.3                                                                          --  -- O  H OCF.sub.2 H                                                                        CH.sub.3                                          H   -- Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O  H CH.sub.3                                                                           H                                                 H   -- Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O  H OCH.sub.3                                                                          H                                                 H   -- Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O  H CH.sub.3                                                                           CH.sub.3                                          H   -- Q-2                                                                               CH.sub.3                                                                          --  -- O  H OCH.sub.3                                                                          CH.sub.3                                          H   -- Q-2                                                                               CH.sub.3                                                                          --  -- O  H OCH.sub.3                                                                          H                                                 H   -- Q-2                                                                               CH.sub.3                                                                          --  -- O  H CH.sub.3                                                                           H                                                 H   -- Q-2                                                                               CH.sub.3                                                                          --  -- O  H OCH.sub.3                                                                          CH.sub.3                                          H   -- Q-2                                                                               CH.sub.3                                                                          --  -- O  H CH.sub.3                                                                           CH.sub.3                                          H   -- Q-3                                                                               -- CH.sub.3                                                                           -- O  H OCH.sub.3                                                                          CH.sub.3                                          H   -- Q-3                                                                               -- CH.sub.3                                                                           -- O  H OCH.sub.3                                                                          CH.sub.3                                          H   -- Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O  H CH.sub.3                                                                           CH.sub.3                                          H   -- Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O  H OCH.sub.3                                                                          H                                                 H   -- Q-4                                                                               -- CH.sub.3                                                                           -- O  H OCH.sub.3                                                                          H                                                 H   -- Q-5                                                                               -- --  CH.sub.3                                                                          O  H OCH.sub.3                                                                          H                                                 H   -- Q-5                                                                               -- --  CH.sub.3                                                                          O  H OCH.sub.3                                                                          CH.sub.3                                          H   -- Q-5                                                                               -- --  CH.sub.3                                                                          O  H CH.sub.3                                                                           H                                                 5-Cl                                                                               -- Q-5                                                                               -- --  CH.sub.3                                                                          O  H CH.sub.3                                                                           H                                                 6-CH.sub.3                                                                         -- Q-5                                                                               -- --  CH.sub.3                                                                          O  H OCH.sub.3                                                                          H                                                 H   -- Q-3                                                                               -- H   -- O  H CH.sub.3                                                                           H                                                 H   -- Q-3                                                                               -- H   -- O  H OCH.sub.3                                                                          H                                                 H   -- Q-3                                                                               -- OCH.sub.3                                                                          -- O  H CH.sub.3                                                                           CH.sub.3                                          H   -- Q-3                                                                               -- OCH.sub.3                                                                          -- O  H OCH.sub.3                                                                          CH.sub.3                                          H   -- Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O  H CH.sub.3                                                                           H                                                 H   -- Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O  H OCH.sub.3                                                                          H                                                 H   -- Q-3                                                                               -- SCH.sub.3                                                                          -- O  H CH.sub.3                                                                           CH.sub.3                                          H   -- Q-3                                                                               -- SCH.sub.3                                                                          -- O  H OCH.sub.3                                                                          CH.sub.3                                          __________________________________________________________________________

                                      TABLE V                                      __________________________________________________________________________     General Structure 5                                                            R.sub.1                                                                            E Q  R.sub.3                                                                              R.sub.4                                                                            R.sub.5                                                                           W R X.sub.2                                                                             Y.sub.2                                                                            m.p. (°C.)                           __________________________________________________________________________     H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.2 CF.sub.3                                                                   OCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SC.sub.2 H.sub.5                                H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                      --  -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                      --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-2                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-2                                                                               CH(CH.sub.3).sub.2                                                                   --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SC.sub.2 H.sub.5                                H   --                                                                               Q-3                                                                               --    C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CF.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       6-CH.sub.3                                                                         --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       6-Cl                                                                               --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-5                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-6                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-7                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       6-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SCH.sub.3                                       5-Cl                                                                               --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    H   -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    H   -- O H C.sub.2 H.sub.5                                                                     OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    OCH.sub.3                                                                          -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    OCH.sub.3                                                                          -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                H   --                                                                               Q-3                                                                               --    SCH.sub.3                                                                          -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    SCH.sub.3                                                                          -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                __________________________________________________________________________

                  TABLE VI                                                         ______________________________________                                         General Structure 6                                                                                                              m.p.                         R.sub.1                                                                              E     Q      R.sub.3                                                                             R.sub.4 R.sub.5                                                                             W   R   X.sub.3                                                                             (°C.)                 ______________________________________                                         H     --    Q-1    CH.sub.3                                                                            --      --   O   H   CH.sub.3                          H     --    Q-1    CH.sub.3                                                                            --      --   O   H   OCH.sub.3                         H     --    Q-1    C.sub.2 H.sub.5                                                                     --      --   O   H   CH.sub.3                          H     --    Q-1    C.sub.2 H.sub.5                                                                     --      --   O   H   OCH.sub.3                         H     --    Q-2    CH.sub.3                                                                            --      --   O   H   CH.sub.3                          H     --    Q-2    C.sub.2 H.sub.5                                                                     --      --   O   H   CH.sub.3                          H     --    Q-3    --   CH.sub.3                                                                               --   O   H   CH.sub.3                          H     --    Q-3    --   CH.sub.3                                                                               --   O   H   OCH.sub.3                         H     --    Q-3    --   C.sub.2 H.sub.5                                                                        --   O   H   CH.sub.3                          H     --    Q-3    --   C.sub.2 H.sub.5                                                                        --   O   H   OCH.sub.3                         H     --    Q-3    --   CH(CH.sub.3).sub.2                                                                     --   O   H   OCH.sub.3                         H     --    Q-3    --   CH.sub.2 Cl                                                                            --   O   H   OCH.sub.3                         H     --    Q-3    --   CF.sub.3                                                                               --   O   H   OCH.sub.3                         H     --    Q-4    --   CH.sub.3                                                                               --   O   H   OCH.sub.3                         6-CH.sub.3                                                                           --    Q-1    CH.sub.3                                                                            --      --   O   H   OCH.sub.3                         6-Cl  --    Q-1    CH.sub.3                                                                            --      --   O   H   OCH.sub.3                         5-Cl  --    Q-1    CH.sub.3                                                                            --      --   O   H   OCH.sub.3                         H     --    Q-5    --   --      CH.sub.3                                                                            O   H   OCH.sub.3                         H     --    Q-5    --   --      CH.sub.3                                                                            O   H   CH.sub.3                          H     --    Q-6    --   --      CH.sub.3                                                                            O   H   OCH.sub.3                         H     --    Q-6    --   --      CH.sub.3                                                                            O   H   CH.sub.3                          H     --    Q-7    --   --      CH.sub.3                                                                            O   H   OCH.sub.3                         H     --    Q-3    --   H       --   O   H   CH.sub.3                          H     --    Q-3    --   H       --   O   H   OCH.sub.3                         H     --    Q-3    --   OCH.sub.3                                                                              --   O   H   CH.sub.3                          H     --    Q-3    --   OCH.sub.3                                                                              --   O   H   OCH.sub.3                         H     --    Q-3    --   OC.sub.2 H.sub.5                                                                       --   O   H   CH.sub.3                          H     --    Q-3    --   OC.sub.2 H.sub.5                                                                       --   O   H   OCH.sub.3                         H     --    Q-3    --   SCH.sub.3                                                                              --   O   H   CH.sub.3                          H     --    Q-3    --   SCH.sub.3                                                                              --   O   H   OCH.sub.3                         ______________________________________                                    

                                      TABLE VII                                    __________________________________________________________________________     General Structure 7                                                            R.sub.1                                                                             E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X.sub.4                                                                              Y.sub.4                                                                            Z.sup.1                                                                           m.p. (°C.)                         __________________________________________________________________________     H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    CH.sub.3                                                                           N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    OCH.sub.3                                                                          N                                            H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    CH.sub.3                                                                           CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    OCH.sub.3                                                                          CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OC.sub.2 H.sub.5                                                                   CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            Cl  CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OC.sub.2 H.sub.5                                                                   CH                                           H    --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             Cl  CH                                           6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           6-CH.sub.3                                                                          --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           6-CH.sub.3                                                                          --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            5-Cl --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           5-Cl --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           5-OCH.sub.3                                                                         --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           5-OCH.sub.3                                                                         --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           5-OCH.sub.3                                                                         --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           H    --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-6                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-7                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          N                                            H    --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                           H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                           H    --                                                                               Q-3                                                                               -- H   -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- H   -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           N                                            H    --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            H    --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                           H    --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H OCH.sub. 3                                                                           CH.sub.3                                                                           N                                            H    --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                           H    --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                            __________________________________________________________________________

                                      TABLE VIII                                   __________________________________________________________________________     General Structure 8                                                            R.sub.1                                                                            n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W    R  X   Y    Z  m.p.(°C.)                    __________________________________________________________________________     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub.3                                                                          CH.sub. 3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N                                      H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N                                      H   0 --                                                                               Q-3                                                                               -- H     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            N                                      H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q 4                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               O-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub. 3                                                                          N                                      4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4 Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub. 3                                                                           -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    CH.sub.3                                                                          CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- NCH.sub.3                                                                           H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- NOCH.sub.3                                                                          H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    CH.sub.3                                                                          CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     __________________________________________________________________________

                                      TABLE IX                                     __________________________________________________________________________     General Structure 9                                                            R.sub.1 n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                            W  R  X   Y   Z  m.p. (°C.)                 __________________________________________________________________________     H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --  O  H  CH.sub. 3                                                                          CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --  O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --  O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --  O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --  O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub. 3                                                                         OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-1                                                                               CH.sub. 3                                                                         --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  Cl  OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --  O  H  OCH.sub. 3                                                                         OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           N                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --  O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                           O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                           O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                           O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                           O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                           O  H  Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                           O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                           O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     --  C  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub. 3                                                                         CH                                   4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            O   H  CH.sub.3                                                                          OCH.sub.3                                                                          N                                        4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  H  CH.sub.3                                                                          OCH.sub.3                                                                          CH                                       4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-Br    0 --                                                                               Q-3                                                                               -- H     --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-3                                                                               -- H     --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-3                                                                               -- H     --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-Br    0 --                                                                               Q-3                                                                               -- H     --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-3                                                                               -- H     --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-Br    0 --                                                                               Q-3                                                                               -- H     --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  H  Cl OCH.sub.3                                                                          CH                                       4-SOCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-SOCH.sub. 3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  Cl  OCH.sub.3                                                                          CH                                   4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  S  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --  S  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                   H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --  O  CH.sub.3                                                                          Cl  OCH.sub.3                                                                          CH                                   H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                           NH H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                   H       1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --  O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                    H       1 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --  O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                   __________________________________________________________________________

                                      TABLE X                                      __________________________________________________________________________     General Structure 10                                                           R.sub.1                                                                           n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W     R  X   Y   Z  m.p. (°C.)                    __________________________________________________________________________     H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub. 3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub. 3                                                                           -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- S     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     CH.sub.3                                                                          CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- NNHCH.sub.3                                                                          H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  1 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      __________________________________________________________________________

                                      TABLE XI                                     __________________________________________________________________________     General Structure 11                                                           R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p. (°C.)               __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub. 6 H.sub.5                                                                    C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C H.sub.5                                                                           C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub. 3                                                                           CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub. 3                                                                           --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub. 3                                                                           --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub. 3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub. 3                                                                           -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                         CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub. 3                                                                           --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  __________________________________________________________________________

                                      TABLE XII                                    __________________________________________________________________________     General Structure 12                                                           R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y    Z  m.p. (°C.)              __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                          H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 232-233                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH 193-195                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH 195-198                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 165-170                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N  140-145                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  195-196                        H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub. 6 H.sub.5                                                                    --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 165-167                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH 125-127                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH 189-191                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N  166-170                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  160-172                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  180-183                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 171-173                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH 181-183                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH 178-180                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 200-202                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N  179-180                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 195                            H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 172-173                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH 152-156                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                           CH 170-171                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N  173-174                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  168-170                        H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub. 3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub. 3                                                                          CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                          N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH3                                                                               OCH.sub.3                                                                           N                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub. 3                                                                         CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q.2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 OCH.sub. 3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub. 3                                                                         CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub. 3                                                                         OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                           CH                                CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub. 3                                                                         OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub. 3                                                                         CH.sub.3                                                                            N                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                 CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                            CH 213-216                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           CH 186-189                        CH.sub.3                                                                            0 --                                                                               0.2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 207-208                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                           CH 170-173                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N  186-191                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                           N  141-144                        CH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           N  191-193                        H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N  179-183                        H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH 165-167                        __________________________________________________________________________

                                      TABLE XIII                                   __________________________________________________________________________     General Structure 13                                                           R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p. (°C.)               __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub. 2 H.sub.5                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub. 6 H.sub.5                                                                    CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub. 3                                                                         CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub. 3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub. 3                                                                           CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                         CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                         N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub. 3                                                                         CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                         N                                  CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub. 3                                                                           CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  __________________________________________________________________________

                  TABLE XIV                                                        ______________________________________                                         General Structure 14                                                                                                               m.p.                       R.sub.1                                                                            n E    Q      R.sub.3                                                                             R.sub.4                                                                            W   R   X     Y     Z    (°C.)               ______________________________________                                         H   0 --   Q-1    CH.sub.3                                                                            --  O   H   CH.sub.3                                                                             CH.sub.3                                                                             CH                              H   0 --   Q-1    CH.sub.3                                                                            --  O   H   OCH.sub.3                                                                            CH.sub.3                                                                             CH                              H   0 --   Q-1    CH.sub.3                                                                            --  O   H   Cl    OCH.sub.3                                                                            CH                              H   0 --   Q-1    CH.sub.3                                                                            --  O   H   CH.sub.3                                                                             OCH.sub.3                                                                            N                               H   0 --   Q-1    CH.sub.3                                                                            --  O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                               H   0 --   Q-1    C.sub.2 H.sub.5                                                                     --  O   H   OCH.sub.3                                                                            CH.sub.3                                                                             CH                              H   0 --   Q-1    C.sub.2 H.sub.5                                                                     --  O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                              H   0 --   Q-1    C.sub.2 H.sub.5                                                                     --  O   H   Cl    OCH.sub.3                                                                            CH                              H   0 --   Q-1    C.sub.2 H.sub.5                                                                     --  O   H   CH.sub.3                                                                             CH.sub.3                                                                             CH                              H   0 --   Q-1    C.sub.2 H.sub.5                                                                     --  O   H   CH.sub.3                                                                             OCH.sub.3                                                                            N                               H   0 --   Q-2    CH.sub.3                                                                            --  O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                               H   0 --   Q-2    CH.sub.3                                                                            --  O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                              H   0 --   Q-2    CH.sub.3                                                                            --  O   H   OCH.sub.3                                                                            CH.sub.3                                                                             CH                              H   0 --   Q-2    CH.sub.3                                                                            --  O   H   Cl    OCH.sub.3                                                                            CH                              H   0 --   Q-2    CH.sub.3                                                                            --  O   H   CH.sub.3                                                                             CH.sub.3                                                                             CH                              H   0 --   Q-2    CH.sub.3                                                                            --  O   H   OCH.sub.3                                                                            CH.sub.3                                                                             N                               H   0 --   Q-2    C.sub.2 H.sub.5                                                                     --  O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                               H   0 --   Q-2    C.sub.2 H.sub.5                                                                     --  O   H   CH.sub.3                                                                             CH.sub.3                                                                             CH                              H   0 --   Q-2    C.sub.2 H.sub.5                                                                     --  O   H   CH.sub.3                                                                             OCH.sub.3                                                                            CH                              H   0 --   Q-2    C.sub.2 H.sub.5                                                                     --  O   H   Cl    OCH.sub.3                                                                            CH                              H   0 --   Q-2    C.sub.2 H.sub.5                                                                     --  O   H   CH.sub.3                                                                             OCH.sub.3                                                                            N                               H   0 --   Q-2    C.sub.2 H.sub.5                                                                     --  O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                               ______________________________________                                    

                                      TABLE XV                                     __________________________________________________________________________     General Structure 15                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                             W R X   Y   Z  m.p. (°C.)                        __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --   O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --   O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH 138-143                                  H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --   O H OCH.sub.3                                                                          CH.sub.3                                                                           CH 155-159                                  H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --   O H Cl  OCH.sub.3                                                                          CH 157-158                                  H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH 135-140                                  H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --   O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                           H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N  75-78                                    H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --   O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --   O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                           H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --   O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                           H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --   O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                            O H CH.sub.3                                                                           CH.sub. 3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                            O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                            O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                            O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- H     --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- H     --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- H     --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- H     --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- H     --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- H     --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --   O H OCH.sub.3                                                                          OCH.sub. 3                                                                         CH                                          H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     --   O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --   O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --   O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --   O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             --   O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                            O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                            O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                     O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                     O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                     O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                     O H Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                     O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                     O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                           __________________________________________________________________________

                                      TABLE XVI                                    __________________________________________________________________________     General Structure 16                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                           R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                             __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                                H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                                H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H 0 --                                                                               Q-5                                                                               -- --CH.sub.3                                                                        O  H OCH.sub.3                                                                        OCH.sub.3                                                                          N                                                    __________________________________________________________________________

                                      TABLE XVII                                   __________________________________________________________________________     General Structure 17                                                           R.sub.1                                                                            E Q  G  n R.sub.3                                                                           W R X   Y   Z  m.p. (°C.)                              __________________________________________________________________________     H   --                                                                               Q-1                                                                               O  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               S  0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO 0 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO 1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               SO 2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               O  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               S  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               SO 2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 6-CH.sub.3                                                                         --                                                                               Q-1                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 5-Cl                                                                               --                                                                               Q-1                                                                               O  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                5-Cl                                                                               --                                                                               Q-1                                                                               S  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                5-Cl                                                                               --                                                                               Q-1                                                                               SO 1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 5-Cl                                                                               --                                                                               Q-1                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               S  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub. 3                                                                         N                                                 H   --                                                                               Q-2                                                                               SO.sub.2                                                                          0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                H   --                                                                               Q-2                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           N                                                 H   --                                                                               Q-2                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 __________________________________________________________________________

                                      TABLE XVIIa                                  __________________________________________________________________________     General Structure 17                                                           R.sub.1                                                                          E Q  G  n R.sub.4                                                                           W R X   Y   Z  m.p. (°C.)                                __________________________________________________________________________     H --                                                                               Q-3                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-3                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-3                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-3                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-3                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-3                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-3                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-3                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-4                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-4                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-4                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   __________________________________________________________________________

                  TABLE XVIIb                                                      ______________________________________                                         General Structure 17                                                                                                                 m.p.                     R.sub.1                                                                            E     Q      G    n   R.sub.5                                                                             W   R   X     Y     Z  (°C.)             ______________________________________                                         H   --    Q-5    O    1   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            CH                          H   --    Q-5    S    1   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                           H   --    Q-5    SO   1   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            N                           H   --    Q-5    SO.sub.2                                                                            1   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                          H   --    Q-5    O    2   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            N                           H   --    Q-5    S    2   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                          H   --    Q-5    SO   2   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            CH                          H   --    Q-5    SO.sub.2                                                                            2   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                           H   --    Q-6    O    1   CH.sub.3                                                                            O   H   CH.sub. 3                                                                            OCH.sub.3                                                                            N                           H   --    Q-6    S    1   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                          H   --    Q-6    SO   1   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            CH                          H   --    Q-6    SO.sub.2                                                                            1   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                           H   --    Q-6    O    2   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            CH                          H   --    Q-6    S    2   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                           H   --    Q-6    SO   2   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            N                           H   --    Q-6    SO.sub.2                                                                            2   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                          H   --    Q-7    O    1   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            CH                          H   --    Q-7    S    1   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                           H   --    Q-7    SO   1   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            N                           H   --    Q-7    SO.sub.2                                                                            1   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                          H   --    Q-7    O    2   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            CH                          H   --    Q-7    S    2   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            N                           H   --    Q-7    SO   2   CH.sub.3                                                                            O   H   CH.sub.3                                                                             OCH.sub.3                                                                            N                           H   --    Q-7    SO.sub.2                                                                            2   CH.sub.3                                                                            O   H   OCH.sub.3                                                                            OCH.sub.3                                                                            CH                          ______________________________________                                    

                                      TABLE XVIII                                  __________________________________________________________________________     General Structure 18                                                           R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p. (°C.)               __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub. 6 H.sub.5                                                                    --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub. 3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub. 3                                                                           --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub. 3                                                                           --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub. 3                                                                           -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub. 3                                                                         CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub. 3                                                                           --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub. 3                                                                         OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub. 3                                                                         CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                         CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub. 3                                                                           --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub. 3                                                                           -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  __________________________________________________________________________

                                      TABLE XIX                                    __________________________________________________________________________     General Structure 19                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                            __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub. 3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub. 5                                                                   -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               __________________________________________________________________________

                                      TABLE XX                                     __________________________________________________________________________     General Structure 20                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                            __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub. 3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               __________________________________________________________________________

Formulations

Useful formulations of the compounds of Formula I can be prepared in conventional ways. They include dusts, granules, pellets, solutions, suspensions, emulsions, wettable powders, eulsifiable concentrates and the like. Many of these may be applied directly. Sprayable formulations can be extended in suitable media and used at spray volumes of from a few liters to several hundred liters per hectare. High strength compositions are primarily used as intermediates for further formulation. The formulations, broadly, contain about 0.1% to 99% by weight of active ingredient(s) and at least one of (a) about 0.1% to 20% surfactant(s) and (b) about 1% to 99.9% solid or liquid inert diluent(s). More specifically, they will contain these ingredients in the following approximate proportions:

    ______________________________________                                                     Active  Weight Percent*                                                        Ingredient                                                                             Diluent(s)                                                                               Surfactant(s)                                    ______________________________________                                         Wettable Powders                                                                             20-90      0-74     1-10                                         Oil Suspensions,                                                                              3-50     40-95     0-15                                         Emulsions, Solutions,                                                          (including Emulsifiable                                                        Concentrates)                                                                  Aqueous Suspension                                                                           10-50     40-84     1-20                                         Dusts          1-25     70-99     0-5                                          Granules and Pellets                                                                         0.1-95      5-99.9  0-15                                         High Strength 90-99      0-10     0-2                                          Compositions                                                                   ______________________________________                                          *Active ingredient plus at least one of a Surfactant or a Diluent equals       100 weight percent.                                                      

Lower or higher levels of active ingredient can, of course, be present depending on the intended use and the physical properties of the compound. Higher ratios of surfactant to active ingredient are sometimes desirable, and are achieved by incorporation into the formulation or by tank mixing.

Typical solid diluents are described in Watkins, et al., "Handbook of Insecticide Dust Diluents and Carriers", 2nd Ed., Dorland Books, Caldwell, N.J., but other solids, either mined or manufactured, may be used. The more absorptive diluents are preferred for wettable powders and the denser ones for dusts. Typical liquid diluents and solvents are described in Marsden, "Solvents Guide," 2nd Ed., Interscience, New York, 1950. Solubility under 0.1% is preferred for suspension concentrates; solution concentrates are preferably stable against phase separation at 0° C. "McCutcheon's Detergents and Emulsifiers Annual", MC Publishing Corp., Ridgewood, N.J., as well as Sisely and Wood, "Encyclopedia of Surface Active Agents", Chemical Publishing Co., Inc., New York, 1964, list surfactants and recommended uses. All formulations can contain minor amounts of additives to reduce foaming, caking, corrosion, microbiological growth, etc.

The methods of making such compositions are well known. Solutions are prepared by simply mixing the ingredients. Fine solid compositions are made by blending and, usually, grinding as in a hammer or fluid energy mill. Suspensions are prepared by wet milling (see, for example, Littler, U.S. Pat. No. 3,060,084). Granules and pellets may be made by spraying the active material upon preformed granular carriers or by agglomeration techniques. See J. E. Browning, "Agglomeration", Chemical Engineering, Dec. 4, 1967, pp. 147ff. and "Perry's Chemical Engineer's Handbook", 5th Ed., McGraw-Hill, New York, 1973, pp. 8-57ff.

For further information regarding the art of formulation, see for example:

H. M. Loux, U.S. Pat. No. 3,235,361, Feb. 15, 1966, Col. 6, line 16 through Col. 7, line 19 and Examples 10 through 41;

R. W. Luckenbaugh, U.S. Pat. No. 3,309,192, Mar. 14, 1967, Col. 5, line 43 through Col. 7, line 62 and Examples 8, 12, 15, 39, 41, 52, 53, 58, 132, 138-140, 162-164, 166, 167 and 169-182;

H. Gysin and E. Knusli, U.S. Pat. No. 2,891,855, June 23, 1959, Col. 3, line 66 through Col. 5, line 17 and Examples 1-4;

G. C. Klingman, "Weed Control as a Science", John Wiley & Sons, Inc., New York, 1961, pp. 81-96; and

J. D. Fryer and S. A. Evans, "Weed Control Handbook", 5th Ed., Blackwell Scientific Publications, Oxford, 1968, pp. 101-103.

In the following examples, all parts are by weight unless otherwise indicated.

EXAMPLE 16 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       80%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    sodium alkylnaphthalenesulfonate                                                                            2%                                                sodium ligninsulfonate       2%                                                synthetic amorphous silica   3%                                                kaolinite                    13%                                               ______________________________________                                    

The ingredients are blended, hammer-milled until all the solids are essentially under 50 microns, reblended, and packaged.

EXAMPLE 17 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-                                                       50%                                               methyl-1H--tetrazol-1-yl)benzenesulfonamide                                    sodium alkylnaphthalenesulfonate                                                                             2%                                               low viscosity methyl cellulose                                                                               2%                                               diatomaceous earth           46%                                               ______________________________________                                    

The ingredients are blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in diameter. The product is reblended before packaging.

EXAMPLE 18 Granule

    ______________________________________                                         Wettable Powder of Example 17 (above)                                                                    5%                                                   attapulgite granules     95%                                                   (U.S.S. 20-40 mesh; 0.84-0.42 mm)                                              ______________________________________                                    

A slurry of wettable powder containing 25% solids is sprayed on the surface of attapulgite granules while tumbling in a double-cone blender. The granules are dried and packaged.

EXAMPLE 19 Extruded Pellet

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-                                                       25%                                               methyl-1H--tetrazol-1-yl)benzenesulfonamide                                    anhydrous sodium sulfate     10%                                               crude calcium ligninsulfonate                                                                                5%                                               sodium alkylnaphthalenesulfonate                                                                             1%                                               calcium/magnesium bentonite  59%                                               ______________________________________                                    

The ingredients are blended, hammer-milled and then moistened with about 12% water. The mixture is extruded as cylinders about 3 mm diameter which are cut to produce pellets about 3 mm long. These may be used directly after drying, or the dried pellets may be crushed to pass a U.S.S. No. 20 sieve (0.84 mm openings). The granules held on a U.S.S. No. 40 sieve (0.42 mm openings) may be packaged for use and the fines recycled.

EXAMPLE 20 Oil Suspension

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       25%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    polyoxyethylene sorbitol hexaoleate                                                                          5%                                               highly aliphatic hydrocarbon oil                                                                            70%                                               ______________________________________                                    

The ingredients are ground together in a sand mill until the solid particles have been reduced to under about 5 microns. The resulting thick suspension may be applied directly, but preferably after being extended with oils or emulsified in water.

EXAMPLE 21 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-                                                       20%                                               methyl-1H--tetrazol-1-yl)benzenesulfonamide                                    sodium alkylnaphthalenesulfonate                                                                            4%                                                sodium ligninsulfonate       4%                                                low viscosity methyl cellulose                                                                              3%                                                attapulgite                  69%                                               ______________________________________                                    

The ingredients are thoroughly blended. After grinding in a hammer-mill to produce particles essentially all below 100 microns, the material is reblended and sifted through a U.S.S. No. 50 sieve (0.3 mm opening) and packaged.

EXAMPLE 22 Low Strength Granule

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       1%                                                methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    N,N--dimethylformamide       9%                                                attapulgite granules         90%                                               (U.S.S. 20-40 sieve)                                                           ______________________________________                                    

The active ingredient is dissolved in the solvent and the solution is sprayed upon dedusted granules in a double cone blender. After spraying of the solution has been completed, the blender is allowed to run for a short period and then the granules are packaged.

EXAMPLE 23 Aqueous Suspension

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                        40%                                              methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    polyacrylic acid thickener   0.3%                                              dodecylphenol polyethylene glycol ether                                                                     0.5%                                              disodium phosphate             1%                                              monosodium phosphate         0.5%                                              polyvinyl alcohol            1.0%                                              water                        56.7%                                             ______________________________________                                    

The ingredients are blended and ground together in a sand mill to produce particles essentially all under 5 microns in size.

EXAMPLE 24 Solution

    ______________________________________                                         N--[(4,6,dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                        5%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide, Sodium                            Salt                                                                           water                        95%                                               ______________________________________                                    

The salt is added directly to the water with stirring to produce the solution, which may then be packaged for use.

EXAMPLE 25 Low Strength Granule

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                        0.1%                                             methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    attapulgite granules         99.9%                                             (U.S.S. 20-40 mesh)                                                            ______________________________________                                    

The active ingredient is dissolved in a solvent and the solution is sprayed upon dedusted granules in a doulbe-cone blender. After spraying of the solution has been completed, the material is warmed to evaporate the solvent. The material is allowed to cool and then packaged.

EXAMPLE 26 Granule

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       80%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    wetting agent                 1%                                               crude ligninsulfonate salt (containing                                                                      10%                                               5-20% of the natural sugars)                                                   attapulgite clay              9%                                               ______________________________________                                    

The ingredients are blended and milled to pass through a 100 mesh screen. This material is then added to a fluid bed granulator, the air flow is adjusted to gently fluidize the material, and a fine spray of water is sprayed onto the fluidized material. The fluidization and spraying are continued until granules of the desired size range are made. The spraying is stopped, but fluidization is continued, optionally with heat, until the water content is reduced to the desired level, generally less than 1%. The material is then discharged, screened to the desired size range, generally 14-100 mesh (1410-149 microns), and packaged for use.

EXAMPLE 27 High Strength Concentrate

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                        99%                                              methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    silica aerogel               0.5%                                              synthetic amorphous silica   0.5%                                              ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce a material essentially all passing a U.S.S. No. 50 screen (0.3 mm opening). The concentrate may be formulated further if necessary.

EXAMPLE 28 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                        90%                                              methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    dioctyl sodium sulfosuccinate                                                                               0.1%                                              synthetic fine silica        9.9%                                              ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce particles essentially all below 100 microns. The material is sifted through a U.S.S. No. 50 screen and then packaged.

EXAMPLE 29 Wettable Powder

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       40%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    sodium ligninsulfonate       20%                                               montmorillonite clay         40%                                               ______________________________________                                    

The ingredients are thoroughly blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in size. The material is reblended and then packaged.

EXAMPLE 30 Oil Suspension

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       35%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    blend of polyalcohol carboxylic                                                                              6%                                               esters and oil soluble petroleum                                               sulfonates                                                                     xylene                       59%                                               ______________________________________                                    

The ingredients are combined and ground together in a sand mill to produce particles essentially all below 5 microns. The product can be used directly, extended with oils, or emulsified in water.

EXAMPLE 31 Dust

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       10%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    attapulgite                  10%                                               Pyrophyllite                 80%                                               ______________________________________                                    

The active ingredient is blended with attapulgite and then passed through a hammer-mill to produce particles substantially all below 200 microns. The ground concentrate is then blended with powdered pyrophyllite until homogeneous.

EXAMPLE 32 Wettable Powder

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       50%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             sodium alkylnaphthalenesulfonate                                                                             2%                                               low viscosity methyl cellulose                                                                               2%                                               diatomaceous earth           46%                                               ______________________________________                                    

The ingredients are blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in diameter. The product is reblended before packaging.

EXAMPLE 33 Granule

    ______________________________________                                         Wettable Powder of Example 32 (above)                                                                    5%                                                   attapulgite granules     95%                                                   (U.S.S. 20-40 mesh; 0.84-0.42 mm)                                              ______________________________________                                    

A slurry of wettable powder containing 25% solids is sprayed on the surface of attapulgite granules while tumbling in a double-cone blender. The granules are dried and packaged.

EXAMPLE 34 Extruded Pellet

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       25%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             anhydrous sodium sulfate     10%                                               crude calcium ligninsulfonate                                                                                5%                                               sodium alkyulnaphthalenesulfonate                                                                            1%                                               calcium/magnesium bentonite  59%                                               ______________________________________                                    

The ingredients are blended, hammer-milled and then moistened with about 12% water. The mixture is extruded as cylinders about 3 mm diameter which are cut to produce pellets about 3 mm long. These may be used directly after drying, or the dried pellets may be crushed to pass a U.S.S. No. 20 sieve (0.84 mm openings). The granules held on a U.S.S. No. 40 sieve (0.42 mm openings) may be packaged for use and the fines recycled.

EXAMPLE 35 Oil Suspension

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       25%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             polyoxyethylene sorbitol hexaoleate                                                                          5%                                               highly aliphatic hydrocarbon oil                                                                            70%                                               ______________________________________                                    

The ingredients are ground together in a sand mill until the solid particles have been reduced to under about 5 microns. The resulting thick suspension may be applied directly, but preferably after being extended with oils or emulsified in water.

EXAMPLE 36 Wettable Powder

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       20%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             sodium alkylnaphthalenesulfonate                                                                            4%                                                sodium ligninsulfonate       4%                                                low viscosity methyl cellulose                                                                              3%                                                attapulgite                  69%                                               ______________________________________                                    

The ingredients are thoroughly blended. After grinding in a hammer-mill to produce particles essentially all below 100 microns, the material is reblended and sifted through a U.S.S. No. 50 sieve (0.3 mm opening) and packaged.

EXAMPLE 37 Low Strength Granule

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       1%                                                amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             N,N--dimethylformamide       9%                                                attapulgite granules         90%                                               ______________________________________                                    

The active ingredient is dissolved in the solvent and the solution is sprayed upon dedusted granules in a double cone blender. After spraying of the solution has been completed, the blender is allowed to run for a short period and then the granules are packaged.

EXAMPLE 38 Aqueous Suspension

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       40%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             polyacrylic acid thickener   0.3%                                              dodecylphenol polyethylene glycol ether                                                                     0.5%                                              disodium phosphate            1%                                               monosodium phosphate         0.5%                                              polyvinyl alcohol            1.0%                                              water                        56.7%                                             ______________________________________                                    

The ingredients are blended and ground together in a sand mill to produce particles essentially all under 5 microns in size.

EXAMPLE 39 Solution

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       5%                                                amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide, sodium salt                                                water                        95%                                               ______________________________________                                    

The salt is added directly to the water with stirring to produce the solution, which may then be packaged for use.

EXAMPLE 40 Low Strength Granule

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                        0.1%                                             amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             attapulgite granules         99.9%                                             (U.S.S. 20-40 mesh)                                                            ______________________________________                                    

The active ingredient is dissolved in a solvent and the solution is sprayed upon dedusted granules in a double-cone blender. After spraying of the solution has been completed, the material is warmed to evaporate the solvent. The material is allowed to cool and then packaged.

EXAMPLE 41 Granule

    ______________________________________                                         N--[[N--(4,6-dimethyoxy-1,3,5-triazin-2-yl)-N--methyl-                                                      80%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             wetting agent                1%                                                crude ligninsulfonate salt (containing                                                                      10%                                               5-20% of the natural sugars)                                                   attapulgite clay             9%                                                ______________________________________                                    

The ingredients are blended and milled to pass through a 100 mesh screen. This material is then added to a fluid bed granulator, the air flow is adjusted to gently fluidize the material, and a fine spray of water is sprayed onto the fluidized material. The fluidization and spraying are continued until granules of the desired size range are made. The spraying is stopped, but fluidization is continued, optionally with heat, until the water content is reduced to the desired level, generally less than 1%. The material is then discharged, screened to the desired size range, generally 14-100 mesh (1410-149 microns), and packaged for use.

EXAMPLE 42 High Strength Concentrate

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       99%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             silica aerogel               0.5%                                              synthetic amorphous silica   0.5%                                              ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce a material essentially all passing a U.S.S. No. 50 screen (0.3 mm opening). The concentrate may be formulated further if necessary.

EXAMPLE 43 Wettable Powder

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       90%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             dioctyl sodium sulfosuccinate                                                                               0.1%                                              synthetic fine silica        9.9%                                              ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce particles essentially all below 100 microns. The material is sifted through a U.S.S. No. 50 screen and then packaged.

EXAMPLE 44 Wettable Powder

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       40%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             sodium ligninsulfonate       20%                                               montmorillonite clay         40%                                               ______________________________________                                    

The ingredients are thoroughly blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in size. The material is reblended and then packaged.

EXAMPLE 45 Oil Suspension

    ______________________________________                                         N--[[N--(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                       35%                                               amino]carbonyl]-2-(5-methyl-1H--tetrazol-1-yl)-                                benzenesulfonamide                                                             blend of polyalcohol carboxylic                                                                              6%                                               esters and oil soluble petroleum                                               sulfonates                                                                     xylene                       59%                                               ______________________________________                                    

The ingredients are combined and ground together in a sand mill to produce particles essentially all below 5 microns. The product can be used directly, extended with oils, or emulsified in water.

EXAMPLE 46 Dust

    ______________________________________                                         N--[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       10%                                               methyl-1H--tetrazol-5-yl)benzenesulfonamide                                    attapulgite                  10%                                               Pyrophyllite                 80%                                               ______________________________________                                    

The active ingredient is blended with attapulgite and then passed through a hammer-mill to produce particles substantially all below 200 microns. The ground concentrate is then blended with powdered pyrophyllite until homogeneous.

Utility

Test results indicate that the compounds of the present invention are highly active preemergent or postemergent herbicides or plant growth regulants. They have utility for broad-spectrum pre- and/or post-emergence weed control in areas where complete control of all vegetation is desired, such as around fuel storage tanks, industrial storage areas, parking lots, drive-in theaters, around billboards, highway and railroad structures. Some of the compounds have utility for selective weed control in crops such as corn, rice, wheat, barley, soybean and rape. Alternatively, many of the subject compounds are useful to modify plant growth.

The rates of application for the compounds of the invention are determined by a number of factors, including their use as plant growth modifiers or as herbicides, the crop species involved, the types of weeds to be controlled, weather and climate, formulations selected, mode of application, amount of foliage present, etc. In general terms, the subject compounds should be applied at levels of about 0.001 to 10 kg/ha, the lower rates being suggested for use on lighter soils and/or those having a low organic matter content, for plant growth modification or for situations where only short-term persistence is required.

The compounds of the invention may be used in combination with any other commercial herbicide, examples of which are those of the triazine, triazole, uracil, urea, amide, diphenylether, carbamate phenoxyacetic acid and bipyridylium types, as well as other sulfonylureas. They are particularly useful in combination with the following herbicides.

    ______________________________________                                                 Chemical Name                                                          ______________________________________                                         Common Name                                                                    alachlor  2-chloro-2',6'-diethyl-N--(methoxymethyl)-                                     acetanilide                                                          atrazine  2-chloro-4-(ethylamino)-6-(isopropyl-                                          amino)- .sub.-s-triazine                                             butylate  S--ethyl-diisobutylthiocarbamate                                     cyanazine 2-[[4-chloro-6-(ethylamino)- .sub.-s-triazin-2-                                yl]amino]-2-methylpropionitrile                                      dicamba   3,6-dichloro- .sub.-o-anisic acid                                    EPTC      S--ethyl dipropylthiocarbamate                                       glyphosate                                                                               N--(phosphonomethyl)glycine                                          linuron   3-(3,4-dichlorophenyl)-1-methoxy-1-                                            methylurea                                                           metolachlor                                                                              2-chloro-N--(2-ethyl-6-methylphenyl)-N--                                       (2-methoxy-1-methylethyl)acetamide                                   metribuzin                                                                               4-amino-6-tert-butyl-3-(methylthio)-as-                                        triazine-5(4H)-one                                                   tridiphane                                                                               2-(3,5-dichlorophenyl)-2-(2,2,2-tri-                                           chloroethyl)oxirane                                                  2,4-D     (2,4-dichlorophenoxy)acetic acid                                     thiobencarb                                                                              S--4-chlorobenzyldiethylthiocarbamate                                molinate  S--ethyl N,N--hexamethylenethiocarbamate                             butachlor N--(butoxymethyl)-2-chloro-2',6'-di-                                           ethylacetanilide                                                     naproanilide                                                                             N--phenyl-2-(1-naphthyloxy)propionamide                              paraquat  1,1'-dimethyl-4,4'-bipyridinium ion                                  pyrazolate                                                                               4-(2,4-dichlorobenzoyl)-1,3-dimethyl-                                          pyrazol-5-yl-4-toluenesulfonate                                      pretilachlor                                                                             2-chloro-2',6'-diethyl-N--( .sub.-n-propoxy-                                   ethyl)acetanilide                                                    oxidiazon 3-[2,4-dichloro-5-(1-methylethoxy)-                                            phenyl]-5-(1,1-dimethylethyl)-1,3,4-                                           oxadiazol-2(3H)-one                                                  Trade Name or                                                                  Code Number                                                                    Harmony ®                                                                            3-[[(4-methoxy-6-methyl-1,3,5-triazin-                                         2-yl)aminocarbonyl]aminosulfonyl]-2-                                           thiophenecarboxylic acid, methyl ester                               Cinch ®                                                                              exo-1-methyl-4-(1-methylethyl)-2-[(2-                                          methylphenyl)methoxy]-7-oxabicyclo-                                            [2.2.1]heptane                                                       MY-93     S--(1-methyl-1-phenethyl)piperidine-1-                                         carbothioate                                                         CH-83     S--(2-methylpropyl)-hexanhydro-1H--aze-                                        pine-1-carbothioic acid, ester                                       X-52      2,4-dichlorophenyl-3-methoxy-4-nitro-                                          phenyl ether                                                         SC-2957   S--benzyl-N--ethyl-N--propylthiocarbamate                            HW-52     N--(2,3-dichlorophenyl)-4-(ethoxy-                                             methoxy)benzamide                                                    NTN-801   2-(benzothiazol-2-yl)-N--methyl-N--                                            phenylacetamide                                                      SL-49     2-[4-[(2,4-dichlorophenyl)carbonyl]-                                           1,3-dimethyl-1H--pyrazol-5-yloxy]-1-                                           phenylethanone                                                       BAS-514   3,7-dichloro-8-quinoline carboxylic                                            acid                                                                 Assure ®                                                                             ethyl 2-[4-(6-chloro-2-quinoxalinyloxy)-                                       phenoxy]-propionate                                                  DPX-L5300 2-[[N--(4-methoxy-6-methyl-1,3,5-tria-                               (Express ®)                                                                          zine-2-yl)-N--methylaminocarbonyl]-                                            aminosulfonyl]benzoic acid, methyl                                             ester                                                                ______________________________________                                    

Some of the compounds of this invention may particularly be useful in combination with the following herbicides for use as pre- or post-emergent treatments for control of weeds in soybeans:

    ______________________________________                                         Common Name Tradename  Chemical Name                                           ______________________________________                                         acifluorfen Blazer ®                                                                              5-[2-chloro-4-(trifluoro-                                                      methyl)phenoxy] -2-ni-                                                         trobenzoic acid                                         alachlor    Lasso ®                                                                               2-chloro-2',6'-diethyl-                                                        N--(methoxymethyl)acet-                                                        anilide                                                 bentazon    Basagran ®                                                                            3-isopropyl-1H--2,1,3-                                                         benzothiadiazin-4(3H)--                                                        one 2,2-dioxide                                         chloramben  Amiben ®                                                                              3-amino-2,5-dichloro-                                                          benzoic acid                                            fluazifop-  Fusilade ®                                                                            butyl 2-[4-[5-(trifluoro-                               butyl                  methyl)-2-pyridinyl-                                                           oxy]phenoxy]propanoate                                  linuron     Lorox ®                                                                               3-(3,4-dichlorophenyl)-1-                                                      methoxy-1-methylurea                                    metolachlor Dual ® 2-chloro-N--(2-ethyl-6-                                                        methylphenyl)-N--(2-                                                           methoxy-1-methylethyl)-                                                        acetamide                                               metribuzin  Lexone ®                                                                              4-amino-6-tert-butyl-3-                                                        (methylthio)-as-tri-                                                           azin-5(4H)one                                           pendimethalin                                                                              Prowl ®                                                                               N--(1-ethylpropyl)-3,4-                                                        dimethyl-2,6-dinitro-                                                          benzeneamine                                            sethoxydim  Poast ®                                                                               2-[1-(ethoxyimino)butyl]-                                                      5-[2-(ethylthio)-                                                              propyl]-3-hydroxy-2-                                                           cyclohexene-1-one                                       trifluralin Treflan ®                                                                             α,α,α-trifluoro-2,6-di-                                      nitro-N,N--dipropyl- -p                                                        toluidine                                               AC 252,214  --         2-(4,5-dihydro-4-methyl-                                                       4-(1-methylethyl)-5-                                                           oxo-1H--imidazol-2-yl)-                                                        3-quinolinecarboxylic                                                          acid                                                    FMC 57020   --         2-(2'-chlorophenyl)-                                                           methyl-4,4 dimethyl-                                                           3-isoxazolidinone                                       fomesafen   Flex ® 5-(2-chloro-4-trifluoro-                                                       methylphenoxy)-N--                                                             methylsulfonyl-2-nitro-                                                        benzamide                                               lactofen    --         1'-(carboethoxy)ethyl-5-                                                       (2-chloro-4-(trifluoro-                                                        methyl)phenoxy)-2-                                                             nitrobenzoate                                           DOWCO 453 ME           2-(4-(3-chloro-5-tri-                                                          fluoromethylpyridin-2-                                                         yloxy)phenoxy)propanoic                                                        acid, methyl ester                                      fenoxaprop ethyl                                                                           Whip ® ethyl 2-(4-(6-chloro-2-                                                        benzoxazolyloxy)phen-                                                          oxy)propanoate                                          CGA 82725   Topik ®                                                                               2-(4-(3,5-dichloropyri-                                                        din-2-yloxy)phenoxy-                                                           propanoic acid, propyn-                                                        yl ester                                                chlorimuron ethyl                                                                          Classic ®                                                                             2-[[(4-chloro-6-methoxy-                                                       pyrimidin-2-yl)amino-                                                          carbonyl]aminosul-                                                             fonyl]benzoic acid                                                             ethyl ester                                             cinmethylin Cinch ®                                                                               exo-1-methyl-4-(1-methyl-                                                      ethyl)-2-[(2-methyl-                                                           phenyl)methoxy]-7-oxa-                                                         bicyclo[2.2.1]heptane                                   AC 263,499  Pursuit ®                                                                             2-[4,5-dihydro-4-methyl-                                                       4-(1-methylethyl)-5-                                                           oxo-1H--imidazol-2-yl)]-                                                       5-ethyl-3-pyridine-                                                            carboxylic acid                                         AC 252,214  Scepter ®                                                                             2-[4,5-dihydro-4-methyl-                                                       4-(1-methylethyl)-5-                                                           oxo-1H--imidazol-2-yl]-                                                        3-quinolinecarboxylic                                                          acid                                                    ______________________________________                                    

The herbicidal properties of the subject compounds were discovered in a number of green house tests. The test procedures and results follow.

    __________________________________________________________________________     COMPOUNDS                                                                      General Structures for Compounds 1-58                                           ##STR36##                                                                      ##STR37##                                                                     Compound                                                                             Q  R.sub.1                                                                            R.sub.3                                                                             R.sub.4                                                                             R.sub.5                                                                           X    Y     Z                                         __________________________________________________________________________      1    Q-3                                                                               H   --   CH.sub.3                                                                            -- OCH.sub.3                                                                           CH.sub.3                                                                             N                                          2    Q-3                                                                               H   --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         3    Q-1                                                                               H   CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         4    Q-3                                                                               H   --   CH.sub.3                                                                            -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         5    Q-3                                                                               H   --   CH.sub.3                                                                            -- Cl   OCH.sub.3                                                                            CH                                         6    Q-3                                                                               H   --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          7    Q-3                                                                               H   --   CH.sub.3                                                                            -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                          8    Q-3                                                                               H   --   H    -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          9    Q-3                                                                               H   --   H    -- Cl   OCH.sub.3                                                                            CH                                        10    Q-3                                                                               H   --   H    -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        11    Q-3                                                                               H   --   H    -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        12    Q-3                                                                               H   --   H    -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         13    Q-3                                                                               H   --   H    -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        14    Q-3                                                                               5-CH.sub.3                                                                         --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        15    Q-3                                                                               5-CH.sub.3                                                                         --   CH.sub.3                                                                            -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         16    Q-3                                                                               5-CH.sub.3                                                                         --   CH.sub.3                                                                            -- Cl   OCH.sub.3                                                                            CH                                        17    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        18    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        19    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        20    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- Cl   OCH.sub.3                                                                            CH                                        21    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         22    Q-3                                                                               H   --   CH.sub.2 CH.sub.3                                                                   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         23    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        24    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        25    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         26    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         27    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        28    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- Cl   OCH.sub.3                                                                            CH                                        29    Q-3                                                                               5-Cl                                                                               --   CH.sub.3                                                                            -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                         30    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         31    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         32    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        33    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        34    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        35    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- Cl   OCH.sub.3                                                                            CH                                        36    Q-1                                                                               H   CH.sub.2 CH.sub.3                                                                   --   -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                         37    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         38    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         39    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        40    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub. 3                                                                           CH                                        41    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        42    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- Cl   OCH.sub.3                                                                            CH                                        43    Q-1                                                                               3-CH.sub.3                                                                         CH.sub.3                                                                            --   -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                         44    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         45    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         46    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        47    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        48    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        49    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- Cl   OCH.sub.3                                                                            CH                                        50    Q-1                                                                               4-CH.sub.3                                                                         CH.sub.3                                                                            --   -- NHCH.sub.3                                                                          OCH.sub.2 CH.sub.3                                                                   N                                         51    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         52    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            N                                         53    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        54    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        55    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- CH.sub.3                                                                            CH.sub.3                                                                             CH                                        56    Q-1                                                                               6-CH.sub.3                                                                         CH.sub.3                                                                            --   -- Cl   OCH.sub.3                                                                            CH                                        57    Q-5                                                                               H   --   --   CH.sub.3                                                                          OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        58    Q-5                                                                               H   --   --   CH.sub.3                                                                          CH.sub.3                                                                            OCH.sub.3                                                                            N                                         __________________________________________________________________________

    ______________________________________                                         General Structures for Compounds 59- 63                                         ##STR38##                                                                     Compound     X          Y          Z                                           ______________________________________                                         59           OCH.sub.3  OCH.sub.3  CH                                          60           CH.sub.3   OCH.sub.3  CH                                          61           CH.sub.3   CH.sub.3   CH                                          62           OCH.sub.3  OCH.sub.3  N                                           63           Cl         OCH.sub.3  CH                                          ______________________________________                                    

    __________________________________________________________________________     General Structures for Compounds 64- 179                                        ##STR39##                                                                      ##STR40##                                                                     Compound                                                                             Q  R  R.sub.1                                                                             R.sub.3                                                                             R.sub.4 R.sub.5                                                                             X      Y       Z                            __________________________________________________________________________      64   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             65   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             66   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            67   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            68   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            69   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                            70   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             71   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             72   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            73   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            74   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            75   Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub. 3                                                                             CH                            76   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            77   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            78   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            79   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   Cl     OCH.sub.3                                                                              CH                            80   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             81   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             82   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            83   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            84   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            85   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                            86   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             87   Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub. 3                                                                             OCH.sub.3                                                                              N                             88   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            89   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                            90   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   CH.sub.3                                                                              CH.sub.3                                                                               CH                            91   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   Cl     OCH.sub.3                                                                              CH                            92   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                             93   Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   CH.sub.3                                                                              OCH.sub.3                                                                              N                             94   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                            95   Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                            96   Q-1                                                                               H  H    CH.sub.2 CH.sub.3                                                                   --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                            97   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                            98   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                            99   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           100   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   Cl     OCH.sub.3                                                                              CH                           101   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              CH.sub.3                                                                               CH                           102   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           103   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           104   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           105   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           106   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           107   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           108   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           109   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           110   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                           111   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            112   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            113   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            114   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            115   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           116   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           117   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            118   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              N                            119   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           120   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            121   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           122   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            123   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           124   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           125   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           126   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            127   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           128   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              N                            129   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   Cl     OCH.sub.3                                                                              CH                           130   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              CH.sub.3                                                                               CH                           131   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           132   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           133   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           134   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                           135   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub. 3                                                                             --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            136   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            137   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   Br     OCH.sub.3                                                                              CH                           138   Q-1                                                                               CH.sub.3                                                                          6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           139   Q-1                                                                               CH.sub.3                                                                          6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            140   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              H       CH                           141   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             H       CH                           142   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              CH                           143   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              N                            144   Q-1                                                                               CH.sub.3                                                                          6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            145   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   cyclopropyl                                                                           OCH.sub.3                                                                              N                            146   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                     CH                           147   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             CH.sub.2 OCH.sub.2 CH.sub.3                                                            CH                           148   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.2 CF.sub.3                                                                     N                            149   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                     N                            150   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            151   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            152   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           153   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           154   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           155   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           156   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                             N                            157   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             CH(OCH.sub.3).sub.2                                                                    CH                           158   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           159   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            CH.sub.3                                                                              OCH.sub.3                                                                              CH                           160   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            CH.sub.3                                                                              OCH.sub.3                                                                              N                            161   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           162   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           163   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           164   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           165   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           166   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           167   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            168   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            169   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                             N                            170   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           171   Q-5                                                                               H  H    --   --      CH.sub.3                                                                            OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           172   Q-5                                                                               H  H    --   --      CH.sub.3                                                                            OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           173   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           174   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            175   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            176   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           177   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           178   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           179   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           __________________________________________________________________________

    ______________________________________                                         General Structure for Compounds 180- 205                                        ##STR41##                                                                      ##STR42##                                                                     Compound                                                                               Q      R.sub.1                                                                               R.sub.3                                                                               X       Y      Z                                  ______________________________________                                         180     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.3                                                                               CH.sub.3                                                                              CH                                 181     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             CH                                 182     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             CH                                 183     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              Cl      OCH.sub.3                                                                             CH                                 184     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                     NHCH.sub.3                                                                            N                                  185     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             N                                  186     Q-2    CH.sub.3                                                                              CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             N                                  187     Q-2    H      CH.sub.3                                                                              CH.sub.3                                                                               CH.sub.3                                                                              CH                                 188     Q-2    H      CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             CH                                 189     Q-2    H      CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             CH                                 190     Q-2    H      CH.sub.3                                                                              Cl      OCH.sub.3                                                                             CH                                 191     Q-2    H      CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             N                                  192     Q-2    H      CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             N                                  193     Q-2    H      CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                     NHCH.sub.3                                                                            N                                  194     Q-1    H      CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             CH                                 195     Q-1    H      CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             CH                                 196     Q-1    H      CH.sub.3                                                                              CH.sub.3                                                                               CH.sub.3                                                                              CH                                 197     Q-1    H      CH.sub.3                                                                              Cl      OCH.sub.3                                                                             CH                                 198     Q-1    H      CH.sub.3                                                                              CH.sub.3                                                                               OCH.sub.3                                                                             N                                  199     Q-1    H      CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                             N                                  200     Q-2    H      CH.sub.2 CH.sub.3                                                                     CH.sub.3                                                                               CH.sub.3                                                                              CH                                 201     Q-2    H      CH.sub.2 CH.sub.3                                                                     CH.sub.3                                                                               OCH.sub.3                                                                             CH                                 202     Q-2    H      CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              OCH.sub.3                                                                             CH                                 203     Q-2    H      CH.sub.2 CH.sub.3                                                                     Cl      OCH.sub.3                                                                             CH                                 204     Q-2    H      CH.sub.2 CH.sub.3                                                                     CH.sub.3                                                                               OCH.sub.3                                                                             N                                  205     Q-2    H      CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              OCH.sub.3                                                                             N                                  ______________________________________                                    

    ______________________________________                                         General Structure for Compounds 206- 207                                       Compound                                                                       ______________________________________                                         206                                                                                        ##STR43##                                                          207        sodium salt of compound 206                                         ______________________________________                                    

TEST A

Seeds of crabgrass (Digitaria spp.), giant foxtail (Setaria faberii) (in some cases), barnyardgrass (Echinochloa crus-galli), cheatgrass (Bromus secalinus), wild oats (Avena fatua), velvetleaf (Abutilon theo- phrasti), morningglory (Ipomoea spp.), cocklebur (Xanthium pensylvanicum), sorghum, corn, soybean, sugarbeet, cotton, rice, barley (in some cases), wheat and purple nutsedge (Cyperus rotundus) tubers were planted and treated preemergence with the test chemicals dissolved in a non-phytotoxic solvent. At the same time, these crop and weed species were treated with a soil/foliage application. At the time of treatment, the plants ranged in height from 2 to 18 cm. Treated plants and controls were maintained in a greenhouse for sixteen days, after which all species were compared to controls and visually rated for response to treatment. The ratings, summarized in Table A, are based on a numerical scale extending from 0=no injury, to 10=complete kill. The accompanying descriptive symbols have the following meanings:

C=chlorosis/necrosis;

B=burn;

D=defoliation;

E=emergence inhibition;

G=growth retardation;

H=formative effect;

U=unusual pigmentation;

X=axillary stimulation;

S=albinism; and

6Y=abscised buds or flowers.

    TABLE A       Cmpd. 1 Cmpd. 2 Cmpd. 3 Compound 4 Compound 5 Compound 6 Compound 7      Compound 8 Compound 9 Compound 10  Compound 11 Cmpd. 12 Rate kg/ha 0.05      0.05 0.05 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.05 0.01 0.05      0.01 0.05 0.01  0.05 0.01 0.01        POSTEMERGENCE Morningglory 3C,8G 10C 10C 10C 10C 10C 9C 1C,1H 1C 6C,9G 4      C,9H 1H 3H 0 5C,9G 2C,5G 10C 9C 2C,6G 2H 2G Cocklebur 3C,7H 9C 9C 9C 9C      10C 9C 1H 0 8G 2G 0 2H 0 9C 3C,9H 9C 9C 9C 5C,9G 0 Velvetleaf 2C,4G 10C      9C 9C 9C 9C 4C,9H 0 0 4C,8H 3C,5G 2G 0 0 4C,8G 1C 9C 4C,8G 5C,9H 4C,9H 0      Nutsedge 8G 9C 9C 4C,9G 3C,9G 9C 4C,9G 0 0 6G 0 0 0 0 4C,9G 3C,9G 9C 9C      4C,9G 3C,9G 0 Crabgrass 5G 5C,9G 9C 5C,9G 3C,8G 4C,8G 3C,5G 0 0 4C,8G      2C,5G 0 0 0 2G 0 3C,7G 2H 3C,5G 1H 0 Barnyardgrass 5C,9G 9C 5C,9G 9C 9C      9C 9C 4C,9H 0 5C,9H 3C,9H 1H 2H 0 9H 2C,5H 9H 3C,7H 5C,9H 2C,3H 0      Cheatgrass 0 7G 9C 3C,9G 6G 4G 0 0 0 6G 2G 0 0 0 7G 0 9C 3C,9G 9C 8G 0      Wild Oats 3C,8G 9C 9C 5C,9G 5C,9G 4C,9G 3C,9G 2G 0 5C,9G 4C,9G 0 0 0 0 0      5C,9G 2C,7H 9C 9H 0 Wheat 4C,9G 9C 9C 5C,9G 2C,9G 4C,9H 8G 3G 0 4C,9G      2C,9G 0 0 0 0 0 9G 3G 9G 5G 0 Corn 9C 9C 9C 5C,9G 3C,9H 5C,9G 9H 4C,9H      3C,7H 6C,9G 4C,9H 5H 5H 2G 7H 1C,3G 9C 3C,9H 5C,9G 3C,9H 0 Soybean 5C,9G      9C 9C 5C,9G 5C,9G 4C,9G 4C,9H 4C,8H 1C,1H 3C,7G 3G 2G 3H 0 5G 0 5C,9G      3C,8H 3C,7H 2H 1H Rice 6C,9G 9C 9C 9C 9C 6C,9G 9C 5C,9G 5G 9C 9C 2G 2G 0      4C,8G 0 9C 2C,7G 9C 5C,9G 0 Sorghum 6C,9H 9C 9C 5C,9G 6C,9G 9C 9C 4C,8H      3G 5C,9G 4C,9H 5G 0 0 5C,9H 3C,8H 9C 3C,9H 9C 4C,9H 0 Sugar Beets 6C,9H      9C 9C 8G 10C 9C 9C 4C,6G 0 5C,9H 4C,6H 2C,3H 3C,5H 0 10C 4C,9H 10C 10C      9C 9C 1C,1H Cotton 6C,9H 9C 9C 9C 9C 9C 4C,9G 4C,6G 3C,4G 3C,5G 3C,5G 2G      0 0 9C 3C,8H 9C 9C 9C 9H 1C Giant Foxtail    -- -- -- -- -- -- -- -- 0      -- -- -- -- -- -- -- -- -- Barley    -- -- -- -- -- -- -- -- 0 -- -- --      -- -- -- -- -- --  PREEMERGENCE Morningglory 3G 9H 9G 9G 9G 9G 9G 0 0 9G 7      G 0 0 0 9G 4C,8H 9G 8G 8G 3C,5H 0 Cocklebur 0 9H 9H 9H 9H 9H 9H 0 0 8G      7G 0 0 0 8H 2C,5G -- 9H 9H 8H 0 Velvetleaf 0 10C 10C 9C 9C 9C 4C,8G 0 0      4C,9G 0 0 0 0 7H 4G 9C 6C,9G 9C 3C,7H 0 Nutsedge 0 10E 10E 10E 4C,8G 10E      10E 0 0 0 0 0 0 0 10E 3G 10E 9G 10E 4G 0 Crabgrass 0 3C,8G 8G 5C,9G      5C,9G 4C,9G 7G 0 0 4C,8G 0 0 0 0 2C 0 4C,7G 2C,4G 2C,3G 0 0 Barnyardgrass       0 4C,9H 9H 5C,9H 5C,9H 4C,9H 4C,9H 0 0 9H 3G 0 0 0 3C,7G 0 4C,9H 2C,6G      3C,5G 0 0 Cheatgrass 0 7G 9H 9G 7G 5G 3G 0 0 5G 0 0 0 0 3C,7H 4G 10E      4C,9H 5C,9H 5G 0 Wild Oats 0 5C,9G 5C,9G 6C,9H 4C,8H 5C,9G 3C,7G 0 0      5C,9H 3C,6G 0 1C 0 2C,7G 0 9C 4C,9G 9C 3C,7G 0 Wheat 5G 10E 10E 10E      5C,9H 4C,9H 9G 4G 0 4C,9H 2C,6G 0 0 0 6G 0 4C,9G 7G 9G 5G 0 Corn 3C,8G      4C,9G 3C,9H 9H 5C,9H 3C,9G 8G 2G 0 9G 3C,7G 0 4G 0 3C,8H 0 9H 4C,9H      2C,9H 3C,7H 2G Soybean 5G 9H 9H 9H 4C,7G 3C,8H 4C,6G 0 0 2G 0 0 2G 0 3G      0 9H 4C,8H 2C,7G 2C,3G 2C Rice 1C 10E 10E 10E 10E 10E 10E 3G 0 10E 4C,8H      0 5G 0 10E 7G 10E 4C,9H 10E 3C,8G 0 Sorghum 3C,6G 5C,9H 10H 10E 5C,9H      10E 9H 0 0 10E 4C,9H 0 0 0 4C,9H 4C,8G 10E 5C,9H 9H 3C,8H 1C Sugar Beets      0 5C,9G 9C 5C,9G 5C,9G 5C,9G 5C,9G 0 0 5C,9G 4C,8G 0 4G 3H 9C 4C,8G      5C,9G 5C,9G 9C 5C,9G 3H Cotton 0 3C,9G 9C 3C,9G 3C,9G 3C,9G 3C,9G 0 0      2C,5G 0 0 0 0 9G 8G 9C 9G 9G 9G 0 Giant Foxtail    -- -- -- -- -- -- --      -- 0 -- -- -- -- -- -- -- -- -- Barley    -- -- -- -- -- -- -- -- 0 --      -- -- -- -- -- -- -- --        Cmpd. 13 Compound 14 Compound 15 Compound 16 Compound 17 Compound 18      Compound 19  Compound 20 Compound 21 Compound 22 Compound 23 Rate kg/ha      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05  0.01 0.05 0.01        POSTEMERGENCE Morningglory 10C 5C,9G 4G 3C,8H 0 10C 5C,9G 10C 10C 10C      9C 10C 4C,9G 10C 9C 4C,9G 3C,7H 4C,8H 3C,7H 10C 8G Cocklebur 10C 10C 10C      2C,4G 0 10C 8G 10C 10C 10C 10C 9C 7G 10C 9C 5C,9H 5H 5C,9G 3C,7H 10C 10C      Velvetleaf 9C 10C 10C 2C,4H 0 9C 3C,8G 9C 9C 10C 9C 9C 9C 9C 2C,7G 3C,6G      1H 3C,7H 3C,5H 10C 5C,9G Nutsedge 9C 9C 5C,9G 0 0 5C,9G 2C,8G 5C,9G      3C,9G 10C 10C 5C,9G 3C,8G 5C,9G 4C,9G 4G 3C,8G 5G 0 10C 10C Crabgrass 4G      2C,7G 1C 0 0 5G 0 3C,8G 3C,5G 9C 3C,7G 4C,8G 3C,4G 3C,7G 3C,3G 3C,5G 2G      3C,7H 3C,6G 5G 3G Giant Foxtail -- -- -- -- -- -- -- 9C 9C 9C 5C,9H 9C      5C,9G 5C,9H 4C,8G 9C 4C,9G 9C 4C,9H 5C,9G 3C,8G Barnyardgrass 5C,9H 9C      9C 3C,8H 3G 9C 3C,8H 9C 9C 9C 9C 9C 9C 9C 9C 9C 9C 9C 9C 9C 3C,9H      Cheatgrass 4C,9G 3G 0 0 0 0 0 5C,9G 3C,8G 9C 2C,8G 3C,7G 5G 5G 2G 0 0 2C      0 5G 2G Wild Oats 3C,5G 5C,9G 3C,9G 2C,9G 2C,2G 3C,9G 2C,5G 9C 5C,9G      5C,9G 4C,9G 9C 9C 3C,9G 3C,7G 2C 0 2C,6G 0 5G 2G Wheat 0 5C,9G 2C,9G 0 0      8G 5G 4C,9G 9G 9C 3C,9G 9C 5C,9G 3C,9G 9G 5G 0 8G 0 8G 6G Corn 9H 9C      5C,9H 1C,5G 2G 4G 2G 9C 5C,9G 10C 3C,9H 9C 4C,9H 4C,9H 3C,9H 10C 9C 10C      9C 9H 6H Barley -- -- -- -- -- -- -- 5C,9G 3C,8H 6C,9G 3C,8G 9C 4C,9G      2C,8G 3C,7G 0 0 2G 0 3C,9H 6G Soybean 9C 9C 9C 4C,9G 3H 3C,9G 2H,7G 9C      9C 9C 9C 9C 4C,9G 9C 4C,9G 5C,9G 4C,9G 9C 5C,9G 9C 9C Rice 2C,8G 9C 9C      5G 0 5C,9G 7G 9C 9C 9C 9C 9C 9C 9C 5C,9G 5C,9G 7G 9C 6G 9C 4C,9G Sorghum      9H 9C 5C,9H 3C,9H 0 9C 3C,9H 9C 9C 9C 9C 10C 9C 9C 9C 9C 4C,9G 9C 9C 9C      9C Sugar Beets 5C,9G 5C,9G 9C 3C,6G 2C,3G 9C 4C,8G 10C 5C,9G 10C 9C 10C      4C,8G 9C 4C,9G 3C,6H 3C,5G 9C 3C,8G 10C 10C Cotton 9C 9C 5C,9G 3C,9H 1H      2C,9G 8G 9C 5C,9G 9C 10C 9C 4C,9G 5C,9G 9C 4C,9H 4C,9H 4C,9H 3C,8H 9C 9C P      REEMERGENCE Morningglory 9G 9G 8G 5H 3H 9C 9H 9C 7H 9G 8G 8H 3C,7G 9G 7H 5      H 0 3C,8H 2H 9H 7H Cocklebur 9H 9H 9H 7H 0 9H 9H 9H 9H 9H 9H 8H -- 9H 9H      9H -- 9H 2C 9H 9H Velvetleaf 5C,9G 10C 9C 6G 0 9C 2C,4G 9C 3C,8G 9C 9C      9C 3C,7H 5C,9G 7G 7G 0 8H 5G 10C 9G Nutsedge 10E 10E 4C,9G 0 0 10E 3C,9G      10E 10E 10E 10E 9G 7G 10E 9G 0 0 0 0 10E 9G Crabgrass 3G 2C,7G 3G 0 0 4G      2G 4C,8G 3C,7G 8G 4G 5G 0 9C 2G 2C,5G 0 2C,5G 4G 0 0 Giant Foxtail -- --      -- -- -- -- -- 4C,9H 3C,8H 9H 3C,6G 9H 5G 4C,8G 4G 2C,5G 2G 3C,7G 3G      4C,9H 1C Barnyardgrass 3C,8H 5C,9H 3C,8H 1C 0 3C,9H 3C,3G 5C,9H 4C,9H      5C,9H 3C,9H 3C,8H 3C,6G 9H 3C,8H 3C,6G 0 3C,8G 0 5C,9H 3C,8H Cheatgrass      8G 6G 2G 0 0 0 0 4C,8H 3G 7H 6G 2G 0 3G 0 0 0 0 0 4G 0 Wild Oats 5G 9C      5C,9G 2C,5G 0 5C,9G 3C,6G 5C,9G 4C,9G 5C,9G 2C,9G 5C,9G 3C,8H 3C,9H      2C,5G 2G 0 2C 0 6G 0 Wheat 0 4C,9G 3C,8G 0 0 8G 3G 10H 3C,8H 10H 9G      5C,9H 3C,8G 3C,9H 7G 0 0 3G 0 4C,9G 4G Corn 8G 3C,9G 7G 6G 0 6G 2G 10H      4C,9H 4C,9H 8G 4C,9H 3C,7H 3C,9H 9H 4C,9H 2C,6G 9H 3C,8H 3C,8G 2C,5G      Barley -- -- -- -- -- -- -- 9G 3C,9G 3C,9G 9G 4C,9G 9G 3C,9G 8G 0 0 7G 0      3C,9G 2C,8G Soybean 3C,8H 3C,9H 2C,7G 2C,2H 1C 3C,7G 3C,3H 9H 4C,8H 9H      4C,8H 9H 3C,6H 3C,8H 3C,5G 3C,7H 0 3C,7H 2C,3G 3C,8H 3C,8H Rice 2C,9H      10E 3C,8G 5G 1C 10E 2C,8G 10E 9H 10E 10E 10E 4C,8H 10E 9H 8G 2G 9H 0 9H      4C,9G Sorghum 3C,9H 10E 3C,9H 3C,6G 0 10H 3C,9H 10H 6C,9H 10H 10H 5C,9H      6C,9H 10H 10H 5C,9H 3C,6G 4C,9H 3C,8H 10E 3C,9H Sugar Beets 10C 5C,9G      5C,9G 3C,7H 0 10E 5C,9G 10E 9C 5C,9G 5C,9G 9C 5G 9C 5C,9G 5G 3G 4C,7H 5G      5C,9G 5C,9G Cotton 9G 9G 9G 2C 0 9G 2C,5G 9C 2C,9G 4C,9G 4C,9G 9G 2C,8G      9G 8G 5G 0 2C,5G 1C 10C 9C         Compound 24 Compound 25 Compound 26 Compound 27 Compound 28 Compound      29 Compound 30 Compound 31 Compound 32 Compound 33 Compound 34 Rate      kg/ha 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05  0.01 0.05 0.01        POSTEMERGENCE Morningglory 5G 0  0 3C,5G 0 2C,6G 2G 10C 3C,8G 3C,9G      3C,7H 10C 4C,8H 10C 3C,8H 10C 10C 10C 10C  10C 5C,9G Cocklebur 10C 3H 2H      4C,8H 2H 10C 5C,9G 10C 9C 3H 0 9C 4C,9G 10C 9C 10C 10C 10C 9C 10C 5C,9G      Velvetleaf 5C,9G 0 0 2C,5G 0 9C 3C,7G 4C,9G 3C,9G 3C,7H 0 9C 7G 9C 4C,8H      10C 10C 10C 9C 10C 5C,9G Nutsedge 5C,9G 0 0 3C,6G 0 10C 3C,8G 10C 4C,9G      0 0 4C,8G 4G 7G 0 10C 9C 9C 5C,9G 5C,9G 5C,9G Crabgrass 0 0 0 3C,4H 0 2G      2G 3G 0 3C,5G 0 6C,9H 4C,6G 9C 3C,8G 5C,8G 7G 3C,7G 2G 2C,9G 2C,4G Giant      Foxtail 3C,7G 3C,8H 2H 4C,9H 3C,5G 4C,9G 4G 7G 2G 5C,9G 3C,7G 9C 10C 10C      9C 9C 9C 9C 4C,9H 10C 9C Barnyardgrass 3C,7G 5C,9H 0 5C,9H 2C,5G 4C,9H      4C,8H 3C,7H 1C,4G 3C,8H 2H 10C 9C 10C 9C 9C 9C 10C 9C 10C 4C,9H Cheatgras      s 2G 0 0 3G 0 4G 0 0 0 0 0 3G 0 3G 0 7G 5G 7G 5G 6G 2G Wild Oats 0 4C,8G      0 4C,9G 3C,4G 9G 3C,6G 2G 0 4C,9G 7G 4G 3G 7G 4G 4C,9G 9G 5C,9G 3C,7G 9C      4C,9G Wheat 5G 5C,9G 0 3C,9G 7G 5C,9G 2C,6G 4G 0 9G 7G 4G 0 2C,6G 3G 10C      6C,9G 9C 4C,9G 9C 3C,9G Corn 0 3C,9H 2H 9H 0 2G 0 0 0 4C,8H 5H 10C 10C      10C 9C 10C 2C,7H 3C,9H 3C,7H 4C,9H 1H Barley 3G 9G 2G 8G 0 9G 3G 2G 0 9C      9G 0 0 1C,4G 0 9C 8G 3C,9G 4C,9G 9C 2C,8G Soybean 9C 2H,4G 0 3C,8G 2H      5C,9G 4C,9H 3H,8G 3H,8G 3C,7H 4H 9C 5C,9G 9C 4C,9G 9C 9C 10C 5C,9G 9C      4C,9G Rice 3C,7G 9C 2G 9C 8G 9C 5C,9G 2C,8G 6G 9C 3C,8G 5C,9G 4C,9G 9C      4C,9G 9C 9C 9C 9C 9C 9C Sorghum 4C,9H 4C,9H 3G 5C,9G 3C,7H 9C 4C,9G      4C,9H 4C,9G 5C,9G 4C,9G 9C 9C 10C 9C 10C 9C 10C 10C 9C 4C,9H Sugar Beets      10C 5G 0 9C 2H 10C 9C 9C 9C 3C,7H 4H 10C 5C,9G 10C 9C 10C 10C 9C 5C,9G      10C 9C Cotton 4C,9G 0 0 3C,7G 0 9C 9H 9H 9G 5H 0 9C 9H 9C 9C 9C 10C 9C      9C 10C 9C PREEMERGENCE Morningglory 7H 0 0 2H 1H 6G 0 3C,9G 5H 5H 1C 9C      4C,4H 4C,8H 3C,5H 9C 8H 9C 9G 9H 8H Cocklebur 9H 0 0 2C 0 8H 6H 9H 3C,4H      0 0 9H 3C 9H 2C,5G 9H 8H 9H -- 8H 9H Velvetleaf 9C 3G 0 0 0 3C,8H 7G      5C,9H 2G 0 0 9C 9C 9C 0 10C 10C 4C,9G 9G 9H 3C,9G Nutsedge 3C,7G 0 0 0 0      5G 0 10E 0 0 0 4G 0 4G 0 10E 10E 10E 3C,5G 4C,8G 2C,3G Crabgrass 2G 0 0      0 0 0 0 0 0 0 0 3C,7G 3C,4G 3C,5G 0 7G 4G 3C,7G 2C,4G 3C,5G 1C Giant      Foxtail 3C,5G 3G 0 0 0 3C,6G 3C 3C,3H 3G 5G 0 9H 3G 3C,6G 1C 5C,9G 4C,7G      4C,8H 3C,4G 4C,8G 2G Barnyardgrass 3C,6G 0 0 2C 0 4C,9H 3C,3G 5C,9H      3C,3G 3C,5G 0 5C,9H 3C,7G 9C 3C,4H 9C 9H 4C,9H 2C,2H 1C,7H 0 Cheatgrass      0 0 0 0 0 0 0 3G 3G 0 0 3G 0 2G 0 7G 0 8G 2G 6G 0 Wild Oats 2C 0 0 0 0      3C,7G 2C 2C 0 3C,6G 0 2C 0 2C,4G 0 5C,9G 3C,8G 4C,9H 6C,9G 4C,9H 4C,8G      Wheat 5G 0 0 0 0 7G 2G 6G 0 9H 2G 2G 0 2G 0 10E 4C,9G 9C 4C,9G 4C,8G 8G      Corn 0 3G 0 0 0 2C 0 2G 0 2C,5G 0 5C,9H 9H 9H 0 3C,9H 3C,7G 3C,8H 1C,5G      4C,8H 2G Barley 2C,8G 5G 0 5G 3G 9G 6G 8G 5G 2C,8G 2G 5G 0 5G 0 5C,9G      4C,9G 5C,9G 9G 5C,9G 9G Soybean 3C,7H 0 0 0 0 2C,7G 2C,2H 3C,5G 3C,4G      2C,2H 0 3C,8H 3C,7H 3C,8H 2H 9H 3C,7H 9H 9H 9H 3C,7H Rice 3C,6H 5G 0      3C,5G 2C 9H 3C,7H 5C,9H 4C,8H 3C,8H 2C 9H 3C,6H 4C,9H 2C,4G 10E 10E 10E      10E 10E 3C,8H Sorghum 4C,8H 2C 0 3C,5G 2G 9H 2C,6G 5C,9H 5C,9H 3C,8H 1C      6C,9H 4C,8H 10H 4C,7G 6C,9H 9C 10H 7C,9H 6C,9H 4C,8H Sugar Beets 5C,9G 0      0 2H 3G 4C,8G 3C,7H 10C 3C,7G 3G 4H 10E 5H 5C,9G 5H 4C,8G 9C 9C 9C 9C      4C,8H Cotton 2C,7H -- 0 1C 0 4C,8G 2C,3G 3C,7G 2C,4G 0 2H 4C,9G 2C,2H      4C,8H 2C 9C 9G 9G 8G 4C,8G 2G        Compound 35 Compound 36 Compound 37 Compound 38 Compound 39 Compound      40 Compound 41 Compound 42  Compound 43 Compound 44 Rate kg/ha 0.05 0.01 0      .05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01  0.05 0.01        POSTEMERGENCE Morningglory 10C 10C 9C 10C 3C,8H 3C,5H 3C,8H 1C 10C 10C 1      0C 9C 4C,8H 2C,4G 2C,8G 2C,7G 3C,8H 3C,7H  3C,7H 3C,3H Cocklebur 10C 10C      9C 3C,8H 2C,2G 0 3C,7H 0 9C 9C 9C 9C 5C,9H 2C,4G 5C,9H 3C,8G 3G 0 2C,5G      2C Velvetleaf 10C 4C,9G 9C 9C 2C,4G 0 2C,5G 1C 9C 10C 10C 5C,9H 4C,8H      3C,5H 4C,8H 5G 7G 2C,5G 3C,6H 0 Nutsedge 10C 4C,9G 3C,7G 3G 0 0 0 0 9C      5C,9G 2C,8G 5G 0 0 3G 4G 0 0 0 0 Crabgrass 3C,7H 3G 9C 3C,7G 2C,3G 0 2G      0 5C,9G 3C,7G 3C,7G 4G 2G 0 0 0 3G 0 0 0 Giant Foxtail 9C 4C,9G 9C 9C      4C,8G 4G 3C,8H 2G 5C,9G 3C,7G 3C,7G 2G 5G 0 4G 0 2G 0 1C 0 Barnyardgrass      10C 10C 9C 10C 9C 3C,7H 5C,9G 4H 9C 9C 9C 3C,7H 2C,7H 3H 4C,9H 4G 4G 3G      3C,7H 2C,4G Cheatgrass 6G 2G 7G 3G 2C,6G 2G 2G 0 10C 9C 9C 4C,9G 3C,8G      4G 7G 0 8G 7G 0 0 Wild Oats 3C,9G 3C,6G 9C 9C 2C,6G 0 2C,5G 0 5C,9G 9G      4C,9G 3C,6G 7G 3G 2C,7G 0 4C,9G 5C,9G 0 0 Wheat 5C,9G 2C,8G 9C 5C,9G 0 0      4G 0 3C,9G 9G 9G 9G 4G 2G 2G 0 9G 9G 0 0 Corn 4G 0 9C 9C 4C,9G 3C,8H      3C,9H 3C,7H 3C,9G 2U,9G 3C,8H 1C,3G 0 0 2G 0 0 0 3C,7G 0 Barley 9C 6G 9C      4C,9G 0 0 0 0 4C,9G 9G 5G 2G 0 0 0 0 9G 9G 2C 0 Soybean 4C,9G 4C,9G      5C,9G 4C,9G 4C,9G 3C,3G 3C,8G 2C,4H 6C,9G 5C,9G 9C 4C,9G 4C,8H 3C,5H      2C,7G 1H 3H,8G 2H,5G 2C,7H 3H Rice 9C 5C,9G 9C 9C 5C,9G 4C,9G 5C,9G 5G      9C 5C,9G 9C 4C,9G 5C,9G 3C,5G 2C,9G 5G 4C,9G 4C,9G 4C,9G 4G Sorghum 9C      9C 9C 9C 4C,9G 4C,9G 4C,9G 2C,6G 3U,9G 9G 4C,9H 3C,8G 2C,6G 2C,4G 9G 7G      4C,8G 2C,5G 5C,9H 5G Sugar Beets 10C 10C 9C 10C 3C,7H 2H 3C,7H 3C,4H 10C      9C 10C 3C,8H 3C,6H 2C,3G 3C,8G 2C,6G 3C,7G 2C,5G 3C,7H 3C,6G Cotton 10C      10C 9C 9C 3C,8H 2C,3G 3C,7H 2C,2G 9C 4C,9G 4C,9G 4C,9H 4C,9H 2C,3G 2C,8G      5G 5G 0 3C,6G 1C PREEMERGENCE Morningglory 9C 8H 2C,9H 3C,7H 0 0 1C 0 9C 8      G 3C,8H 2C,3H 1C 2G 2C,4H 1H 3H 0 2C 5G Cocklebur 9H 7H 9H 3H -- 0 0 0      9H 8H 3C,7H 2C,3H 3C,3G -- 3C,7H 7H 8G 0 1H 0 Velvetleaf 9G 8G 9G 3C,5H      5G 0 0 0 3C,9G 4C,9G 3C,8H 3C,5H 1H 0 0 2G 0 0 7G 0 Nutsedge 10E 9G 5G 0      2G 0 3G 0 10E 8G 4G 0 0 0 0 0 0 0 0 0 Crabgrass 2C,5G 3C,4G 4C,9G 3C,6G      0 0 -- 0 3C,3G 2G 2C,5G 0 0 0 6G 0 0 0 0 0 Giant Foxtail 3C,6G 4G 4C,9H      3C,5G 0 0 0 0 4C,9H 3C,6G 3C,7G 2G 0 0 2C,7G 0 5G 0 3G 0 Barnyardgrass      4C,9H 3C,7G 3C,9H 3C,7H 1C 0 3G 0 5C,9H 4C,9H 3C,8H 2C,3G 0 0 9H 6G 0 0      3G 0 Cheatgrass 0 0 8G 0 0 0 2G 0 5C,9H 9H 9H 3C,6G 0 0 8G 4G 7G 3G 0 0      Wild Oats 3C,8G 3C,5G 6C,9H 3C,8G 0 0 0 0 4C,9H 3C,8H 3C,8G 3C,5G 0 0 2G      0 2C,6G 0 0 0 Wheat 5C,9H 7G 6C,9H 5G 0 0 0 0 5C,9H 3C,9G 3C,8G 5G 0 0      2G 0 6G 0 0 0 Corn 2C,8G 4G 10H 4C,9H 3C,7H 2C 2C,5G 0 3C,9H 2C,8G 3C,5G      2C,2G 2G 0 2G 0 2C,6G 0 3C,7H 0 Barley 9G 9G 9C 5C,9G 0 0 0 0 9G 9G      3C,9G 8G 2G 0 5G 0 9G 7G 0 0 Soybean 3C,8H 3C,7H 9H 3C,7H 3C,3H 1C 3C,3H      0 9H 3C,6H 4C,6H 3C,4H 3C,3H 1C 7G 0 1C 0 0 0 Rice 10E 10E 10E 3C,9H      3C,6H 3C,3G 2C,7G 2G 10E 5C,9H 4C,9H 2C,6G 0 0 8H 7G 9H 4G 3C,8H 2C,4G      Sorghum 10H 10H 10H 6C,9H 3C,8G 3C,4G 3C,8G 2C 4C,9G 4C,8H 4C,9G 3C,6G      3C,3G 0 8G 2C,7G 3C,6H 0 3C,8H 2C Sugar Beets 4C,9G 3C,8G 10C 4C,9G      3C,5G 7G 5H 3G 9G 8G 5C,9G 4C,8G 6G 3H 8G 0 9G 2G 7G 5G Cotton 9G 4C,9G      8G 1C 2C,4G 1C 2G 0 9G 9G 8G 2C,6G 2C,3G 0 5G 2G 0 0 2C 0        Compound 45 Compound 46 Compound 47 Compound 48 Compound 49 Compound      50 Compound 51 Compound 52 Compound 53 Compound 54 Compound 55 Rate      kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01  0.05 0.01 0.05 0.01        POSTEMERGENCE Morningglory 4C,9H 2C,5G 10C 10C 9C 4C,9H 4C,9H 2C,2H      4C,8G 2C,5G 2C,5H 0 4C,8H 1C 5C,9G 4C,9H 9C 10C  10C 10C 10C 8C Cocklebur       4C,9H 1C 10C 8H 7H 2G 1H 1H 4C,9H 5G 0 0 3C,6G 0 4C,9H 3C,4G 9C 9C 10C      10C 10C 9C Velvetleaf 3C,7H 3C,3G 10C 9C 5C,9G 3C,8G 3C,7H 3G 3C,8H 3H      2C,5G 0 2G 0 3C,8H 3C,4G 9C 9C 10C 9C 10C 9C Nutsedge 3G 0 2C,9G 4C,8G      7G 3G 4G 0 5G 0 0 0 8G 0 9G 2C,7G 9C 9C 9C 5C,9G 9C 9G Crabgrass 2G 0 7G      5G 4G 0 0 0 0 0 0 0 2C,2G 0 3C,7G 2C 8G 3G 6G 3G 3C,6G 2C,5G Giant      Foxtail 2G 0 5C,9G 3C,8G 5G 2G 0 0 3C,6G 0 2C,4G 0 6C,9H 3C,7H 9C 4C,8G      9C 3C,8G 5C,9G 3C,9G 9C 3C,8G Barnyardgrass 3C,9H 2C,5H 10C 5C,9G 3C,9H      3C,8H 3C,7H 1H 3C,8H 3H3C,7H 0 9C 3C,8H 9C 9H 9C 9C 10C 9C 9C 10C      Cheatgrass 3G 0 9G 8G 2C,6G 4G 2G 0 0 0 0 0 8G 0 3C,8G 5G 9C 9G 9C 4C,9G      9C 5C,9G Wild Oats 2G 0 2C,9G 9G 3C,8G 3G 2G 0 0 0 0 0 4C,9G 0 4C,9G      3C,7G 2G 0 3C,5G 0 5C,9G 3C,3G Wheat 2G 0 5C,9G 9G 8G 2G 2G 0 2G 0 0 0      8G 2G 8G 4G 9G 7G 3C,9G 9G 9G 9G Corn 2C,6G 0 2C,9G 9H 3C,8H 2G 1H 0 1H      0 2G 0 4C,9H 2C,5G 3C,8H 0 3H 0 2H 0 2H 0 Barley 0 0 3C,9G 9G 3C,8G 4G      2G 0 1C 0 0 0 3G 0 3C,7G 2G 3C,9G 2C,6G 8G 5G 9G 3C,7G Soybean 3C,8G      2C,6H 9C 5C,9G 4C,9G 3C,8G 2C,7G 2H 2H 1H 0 0 3C,7H 2C,5G 4C,9G 2C,8H 9C      5C,9G 9C 4C,9G 5C,9G 4C,8G Rice 5C,9G 5G 9C 9C 4C,9G 4C,9G 4C,9G 2G      4C,9G 4C,9G 6G 0 9C 5C,9G 9C 4C,9G 9C 5C,9G 9C 9C 5C,9G 5C,9G Sorghum      4C,9H 2C,8G 9C 5C,9G 4C,9G 4C,9G 4C,8G 6G 4C,9G 4C,9H 8G 4G 9C 4C,9H 9C      5C,9G 9C 10C 9C 9C 5C,9G 5C,9G Sugar Beets 5C,9G 3C,7H 10C 9C 9C 9C      4C,8H 2C,6G 3C,8H 2C,5G 3C,7G 0 9C 3C,7H 9C 4C,8H 9C 10C 10C 9C 9C 9C      Cotton 3C,8H 2C,4G 10C 2C,8G 8H 3C,8G 6H 0 7G 3G 2G 0 8H 7H 4C,9G 3C,8H      9C 9C 9C 5C,9G 9G 9G PREEMERGENCE Morningglory 4H 4H 9G 9G 9G 7G 2G 3G      8G 7G 0 0 5G 7G 8G 0 9C 9G 9G 9G 9G 8G Cocklebur 6H 4H 9H 8G 8H -- 0 --      9H 7H 8G -- 4H -- 7H 0 9H -- 9H 9H 9H 9H Velvetleaf 2G 3G 9C 9G 4C,9G 7H      0 -- 3H 0 7G -- 0 5G 5G 0 9C 9C 5C,9G 5C,9G 4C,9G 8G Nutsedge 0 0 4C,9G      0 4G 0 0 0 4G 0 0 0 0 0 5G 0 10E 10E 10E 10E 10E 9G Crabgrass 0 0 3G 0      2G 0 0 0 0 0 0 0 0 0 0 0 2G 0 3G 0 2G 0 Giant Foxtail 0 0 9H 7G 8G 2C 0      0 3C,4G 2G 0 0 4G 2G 6G 2G 9H 8H 9H 3C,8H 9H 3C,8G Barnyardgrass 4G 0 9H      3C,9H 8H 2C 0 0 3C,8H 2G 0 0 2G 2G 5G 0 9H 9H 9H 9H 9H 3C,8H Cheatgrass      0 0 7G 3G 6G 0 0 0 0 0 0 0 2G 0 5G 0 10H 9H 9H 10E 9H 8G Wild Oats 0 0      4C,9H 8H 2C,8G 2G 0 0 2G 0 0 0 0 0 2G 0 0 0 8G 2C,5G 8G 0 Wheat 0 0 10H      3C,9H 8G 3G 0 0 3G 0 0 0 2G 0 7G 0 9H 7H 10H 4C,9H 9G 2G Corn 3C,8H 0      10H 3C,9H 2C,9G 2C,6G 0 0 4G 0 0 0 2C,8G 0 3C,8H 2G 2C,7G 4G 7G 6G 3G      1C,2G Barley 0 0 9G 9H 9G 2C,7G 2G 0 8G 0 0 0 6G 0 8G 3G 9G 9G 9G 9G 9G      8G Soybean 2C,2H 0 9H 8H 3C,7H 7H 2C 0 4G 0 0 0 2C,5G 1H 8H 5H 9H 9H 9H      3C,8H 3C,8H 2C,6G Rice 3C,7H 0 10E 10E 5C,9H 6G 0 3G 3C,8H 4G 2C 0 9H 2G      9H 5H 10E 10E 10E 10E 10E 9H Sorghum 3C,8G 2C,4G 10H 5C,9H 5C,9H 2C,8G      2C -- 10H 3C,8H 2C,5G 0 2C,9H 2C,5G 3C,9H 3C,8G 5C,9H 9H 10H 5C,9H 10H      9H Sugar Beets 4G 4G 5C,9G 5C,9G 4C,9G 7G -- 2G 3C,8G 8G 4G 0 5G 5G 9G      8G 9C 9C 9C 5C,9G 9G 9G Cotton 5G 2C 9G 9G 9G 2C,5G 2G -- 2C,7G 1C 0 0      7G 0 2C,7G 2G 9G 9G 4C,9G 9G 9G 9G        Compound 56 Compound 57 Compound 58 Compound 59 Compound 60 Compound      61 Compound 62  Compound 63 CMPD 64* CMPD 65* CMPD 66 Rate kg/ha 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01  0.05 0.01 0.05 0.01        POSTEMERGENCE Morningglory 10C 10C 10C 2C,8G 1C,7G 0 10C 10C 3C,8G      1C,1H 1C,1H 0 0 0 10C 4C,8G 0 0 0 0 10C 10C Cocklebur 10C 4C,9G 10C 10C      0 0 10C 10C 2C,8G 2H 3H 0 0 0 4C,9H 3C,7H 0 0 0 0 10C 10C Velvetleaf 10C      3C,8G 10C 2C,9H 2G 0 10C 9C 3C,9G 4G 4H 0 0 0 4C,8H 3C,7H 0 0 0 0 10C 9C      Nutsedge 5C,9G 4C,9G 5C,9G 2C,9G 0 0 10C 10C 2C,5G 0 0 0 0 0 9G 2C,8G 0      0 0 0 6C,9G 5C,9G Crabgrass 6G 2G 7G 0 0 0 3C,9G 7G 0 0 0 0 0 0 3C,6G 5G      0 0 0 0 2C,6C 4G Giant Foxtail 4C,9G 7G 3C,9G 2C,7G 0 0 9C 9C 3C,8G 4G      5G 2G 2G 0 9C 2C,8G 0 0 0 0 9C 4C,9G Barnyardgrass 9C 9H 2C,9G 2C,5H 0 0      9C 9C 3C,7H 2H 2C,5G 3G 2C,5G 0 9C 3C,9G 0 0 0 0 9C 9C Cheatgrass 4C,9G      9G 8C 2C,9G 2G 0 9C 10C 9G 3G 6G 0 6G 0 5C,9G 9G 0 0 0 0 9C 4C,9G Wild      Oats 3G 0 2C,9G 2C,6G 0 0 9C 5C,9G 2C,7G 0 2C,5G 2G 2C,5G 0 3C,8G 2C,5G      0 0 0 0 2G 0 Wheat 8G 3G 1C,6G 0 0 0 9C 4C,9G 9G 0 9G 8G 6G 0 9G 7G 0 0      0 0 9G 8G Corn 0 0 1C,8H 3C,8H 0 0 9C 10C 3C,8H 0 2C,7G 3G 3G 0 5C,9G      3C,9G 0 0 0 0 4G 2G Barley 2G 0 5C,9G 3C,9G 0 0 9C 5C,9G 2C,4G 0 2C,5G      3G 4G 0 9G 8G 0 0 0 0 7G 3G Soybean 3C,8G 3C,5H 5C,8H 2C,6H 0 0 9C 9C 3G      2H 2C,6H 3H 0 0 3C,8H 3C,4H 0 0 0 0 9C 9C Rice 9C 5C,9G 5C,9G 2C,8G 3C 0      9C 9C 5C,9G 0 4G 2G 7G 0 6C,9G 4C,9G 0 0 0 0 9C 9C Sorghum 9C 5C,9G      3C,9G 3,9G 1C,5G 0 9C 9C 2C,9G 5G 4G 2G 7G 0 3C,9G 4C,9G 0 0 0 0 9C 9C      Sugar Beets 10C 9C 9C 10C 2C,4H 0 9C 9C 9C 3G 2C,4G 0 2C 0 9C 5C,9G 0 0      0 0 9C 10C Cotton 10C 3C,8G 10C 2C,8H 2G 0 10C 9C 3C,8G 0 0 0 0 0 4C,9G      3C,8H 0 0 0 0 10C 4C,9G PREEMERGENCE Morningglory 9G 9G 8H 3C,7H 0 0 9G      9G 0 0 0 0 0 0 3H 0 0 0 0 0 9H 2C,9H Cocklebur 9H 5H 2C,8H 2C,7H 0 0 9H      9H 2H 0 0 0 0 0 4G 1H 0 0 0 0 9H 7H Velvetleaf 8H 6H 2C,7H 2C,5H 0 0 9C      3C,9G 0 0 0 0 0 0 0 0 0 0 0 0 5C,9G 2C,7G Nutsedge 10E 4G 10E 9G 0 0 10E      10E 0 0 0 0 0 0 7G 0 0 0 0 0 10E 9G Crabgrass 2G 0 1C,5G 2C,4G 0 0 3C,7G      3G 0 0 0 0 0 0 3G 0 0 0 0 0 4G 0 Giant Foxtail 3C,7G 6G 2C,7H 2C,6G 0 0      5C,9H 3C,7G 0 0 0 0 0 0 3G 2G 0 0 0 0 9H 2C,8H Barnyardgrass 9H 8H 2C,6H      2C,4H 0 0 5C,9H 4C,9H 0 0 0 0 0 0 4G 2G 0 0 0 0 9H 3C,9H Cheatgrass 8H      6G 3C,9H 2C,9H 0 0 10E 9H 0 0 0 0 0 0 5G 0 0 0 0 0 9H 8G Wild Oats 0 0      2C,6G 2C,6G 0 0 4C,9H 3C,6G 0 0 0 0 0 0 2C 0 0 0 0 0 2G 0 Wheat 8G 5G 4G      0 0 0 10H 4,9H 0 0 0 0 0 0 3G 0 0 0 0 0 4C,9H 2C,8H Corn 1C 0 2C,7G      3C,4G 0 0 5C,9H 4C,9H 0 0 0 0 0 0 3C,3G 0 0 0 0 0 4C,8H 6G Barley 4C,8G      5G 6G 6G 0 0 4C,9G 3C,9G 0 0 0 0 0 0 3C,9G 4G 0 0 0 0 9G 2C,6G Soybean      7H 2H 2C,5G 1C,2G 0 0 9H 9H 0 0 0 0 0 0 1C 0 0 0 0 0 9H 9H Rice 10E 8H      3C,9H 2C,8H 0 0 10E 10E 0 0 0 0 0 0 4C,8H 3G 0 0 0 0 9H 9H Sorghum 9H      5C,9H 2C,9H 2C,8H 0 0 10H 4C,9H 0 0 0 0 0 0 4C,9H 3C,5G 0 0 0 0 10H      5C,9H Sugar Beets 4C,9G 8G 9C 4C,8G 1C 0 5C,9G 4C,9G 0 0 0 0 0 0 7G      3C,5G 0 0 0 0 5C,9G 4C,9G Cotton 9G 7G 2C,8G 2C,8G 0 0 9G 9G 0 0 0 0 0 0      3C,6G 5G 0 0 0 0 4C,9G 2C,8G      *It is noted that Compounds 64 and 65 were inactive at the levels tested.      However, it is believed that at higher levels, herbicidal activity would      be present.     CMPD 67 CMPD 68 CMPD 69 CMPD 70 CMPD 71 CMPD 72 CMPD 73 CMPD 74 CMPD 75      CMPD 76 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01  0.05 0.01        POSTEMERGENCE Cotton 9C 4C,9H 4C,9G 4C,9H 4C,8G 4C,9H 3C,8H 0 4C,9H      3C,8H 9C 4C,9G 4C,9H 4C,9H 9G 9G 9G 9G 9C 9C Morningglory 10C 10C 9C      5C,9G 10C 4C,9H 3C,8G 3C,7G 4C,9H 3C,8H 10C 4C,9G 10C 9C 4C,9G 3C,8H 9C      2C,9G 10C 7G Cocklebur 10C 9C 10C 5C,9G 9C 4C,9H 2G 0 4C,9H 2C,2H 10C      5C,9G 10C 4C,9G 4C,9G 3C,8H 5C,9G 3C,8H 10C 10C Nutsedge 5C,9G 4C,8G      5C,9G 7G 2C,8G 5G 0 0 4G 0 5C,9G 5C,9G 5C,9G 3C,9G 4C,9G 2C,5G 3C,9G      5C,9G 10C 10C Crabgrass 4G 3H 6G 3G 3H 2H 0 0 0 0 2H 0 0 2H 0 0 0 0      2C,7G 7G Barnyardgrass 9C 9C 9C 5C,9H 9C 4C,9H 5C,9H 5G 5C,9H 9C 10C 9C      4C,9H 3C,7H 3C,8H 4G 3C,8H 3C,5H 10C 9C Wild Oats 2C,6G 2G 4C,9G 2C,3G      3G 0 4C,8G 2G 3C,8G 3G 5C,9G 3C,7G 6C,9G 2C,2G 9C 3C,7G 2C,3G 0 2C,9G      2C,6G Wheat 9G 7G 9G 9G 6G 0 3C,8G 3G 3G 0 5C,9G 8G 4C,9G 2C,5G 4C,8G 3G      2C,3G 0 4C,9G 10C Corn 0 0 2H 0 0 0 5C,9G 6G 6G 3G 4C,9G 4G 3C,5G 3G 1C      0 0 0 6U,9C 3U,8G Soybean 9C 5C,9G 4C,9G 5C,9G 5C,9G 3C,7H 4C,9G 3C,7H      4C,9G 3C,8G 9C 5C,9G 5C,9G 4C,9G 4C,9G 4C,9G 3C,8G 4H 10C 9C Rice 9C 9C      9C 9C 9C 4C,9G 4C,9G 5G 8G 2C,5G 9C 5C,9G 5C,9G 3G 5C,9G 2C,8G 3C,8G 2G      6C,9G 9C Sorghum 9C 5C,9G 9C 4C,9G 9C 4C,9G 3C,9H 4C,8H 5C,9H 3C,9H 10C      9C 9C 4C,9H 9H 2C,5G 10C 9G 9C 3U,9G Cheatgrass 9C 4C,9G 10C 4C,9G 4C,9G      4C,9G 3C,8G 2C,5G 3C,6G 4G 9C 9C 9C 4C,9G 4C,9G 2C,7G 3C,8G 2C,5G 10C      10C Sugar Beets 10C 9C 10C 9C 9C 5C,9G 3C,7H 2C,2H 4C,8H 3C,6H 10C 10C      10C 3C,8H 3C,8H 3C,8G 4C,9G 1C,2G 10C 10C Velvetleaf 10C 4C,9H 9C 5C,9G      3C,7H 2C 0 0 4C,6H 0 10C 10C 10C 4C,9H 9C 3C,7H 5C,9G 3C,5G 10C 10C      Giant Foxtail 9C 5C,9G 9C 5C,9G 5C,9G 7G 4C,9H 3G 4C,9H 3C,7G 3C,8G 3G      3C,7H 2G 3G 2G 1C 0 4C,9G 2C,9G Barley 3G 0 2G 0 0 0 2G 0 5G 0 9G 4G 3G      0 3C,7G 0 0 0 3C,9G 9G PREEMERGENCE Cotton 3C,7H 6G 3C,8H 2C 2C,6G 2C 0      0 0 0 8G 3G 2G 0 1C 0 2G 0 9G 9G Morningglory 8H 2C,6H 9G 3H 8G 2C,2H 2G      0 3H 0 7H 4H 2G 0 0 0 3C,8H 6G 9G 8G Cocklebur 3C,7H 2C,5G 3C,7H 1C      3C,7H 2C 0 0 0 -- 8H 2C 0 0 0 0 2C,2H 1C 9H 9H Nutsedge 5G 5G 10E 0      2C,5G 3G 0 0 0 0 10E 3C,7G 5G 0 10E 0 3C,8G 0 10E 10E Crabgrass 0 0 2G 0      2G 0 0 0 0 0 0 0 0 0 0 0 0 0 7G 6G Barnyardgrass 3C,9H 2G 3C,9H 1C 3C,7H      0 2C,5G 0 0 0 9H 2C,5G 3C,7G 0 2G 0 3C,8H 0 9H 9H Wild Oats 2C 0 2C,4G 0      0 0 0 0 0 0 3C,7G 2G 3C,5G 0 0 0 0 0 7G 7G Wheat 3C,8H 5G 8G 6G 5G 0 0 0      0 0 8G 2G 7G 0 0 0 0 0 3C,9G 2C,9G Corn 4G 0 2G 2G 0 0 3G 0 2C,4G 0      3C,8H 3G 2G 0 0 0 0 0 9G 9G Soybean 9H 3C,7H 3C,9H 3C,6H 3C,7H 2C,4G 0 0      0 0 7H 3C,5H 3C,4H 1C,1H 1H 0 2C 0 9H 9H Rice 3C,9H 3C,7G 5C,9H 3C,7G 9H      7G 6G 0 0 0 10E 9H 9H 3G 7H 0 7H 6H 10E 10E Sorghum 3C,9H 3C,9H 5C,9H      3C,7H 3C,9H 2C,8H 2G 0 3C,5G 0 10H 9H 9H 3C,3G 3C,7G 0 9H 3C,7G 10C 10C      Cheatgrass 9G 8G 3C,9G 8G 9H 8G 5G 0 0 0 9H 3C,9H 9H 0 5G 0 8H 0 10E 10H      Sugar Beets 9G 7G 4C,8H 3C,8G 3C,7H 2C,5G 2G 0 3G 0 9G 9G 7G 1H 5H 0 5H      2G 9G 9G Velvetleaf 3C,7H 0 3C,5H 1C 2H 2C,2G 1C 0 0 0 5H 0 2G 0 2G 0 2G      4G 9G 9G Giant Foxtail 3C,8G 3G 3C,9H 2C,5G 9H 3C,5G 2C,2G 0 2G 0 3C,8H      2C,2G 3C,3G 0 0 0 2C 0 9H 8G Barley 2G 2G 3C,7G 0 2G 0 0 0 0 0 8G 5G 2G      0 0 0 0 0 9G 9G        CMPD 77 CMPD 78 CMPD 79  CMPD 80 CMPD 81 CMPD 82 CMPD 83 CMPD 84 CMPD      85 CMPD 86 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01  0.05 0.01        POSTEMERGENCE Cotton 9C 5C,9G 3C,9G 9G 10C 9C 9C 2C,8H 9C 2C,8H 9C      5C,9G 9C 9C 9C 4C,9G 9C 4C,9G 4C,9H 3C,4G Morningglory 10C 10C 10C 3C,8H      10C 9C 3C,8H 4C,8H 10C 4C,8H 10C 10C 10C 10C 10C 10C 10C 10C 3C,8H 3C,6H      Cocklebur 10C 10C 9C 3C,8H 10C 9C 5C,9H 4C,8H 10C 10C 10C 10C 10C 10C      10C 10C 10C 10C 4G 0 Nutsedge 10C 5C,9G 4C,9G 2C,9G 10C 4C,9G 8G 6G      3C,8G 0 9C 9C 9C 4C,8G 9C 9C 9C 5C,9G 3C,5G 0 Crabgrass 2C,6G 3G 6G 0 6G      2G 5G 0 2C,5G 0 6C,9G 4C,6G 4C,8G 4G 4C,9G 7G 3C,6G 2G 3C,5G 0 Barnyardgr      ass 9C 9C 9C 4C,9H 3C,9G 2C,8G 9C 2C,9H 10C 3C,9G 9C 9C 9C 9C 9C 9C 10C      9C 9C 5C,9H Wild Oats 3C,9G 2C,7G 3C,9G 3C,9G 6G 2C,6G 3C,7G 2C,5G 5C,9G      3C,8G 9C 3C,9G 5C,9G 4C,9G 9C 4C,9G 5C,9G 4C,9G 5C,9G 5C,9G Wheat 2C,9G      9C 3C,9G 9G 2C,9G 9G 4G 0 2G 0 9C 3C,9G 6C,9G 4C,9G 9C 4C,9G 4C,9G 8G      5C,9G 4C,9G Corn 4U,9G 2C,9G 3C,8H 1C,4G 3C,9G 2C,7H 6U,9C 3U,9G 6U,9C      3U,9C 10C 3C,9G 9C 9C 6C,9G 3C,9G 5C,9G 9G 9C 9G Soybean 6C,9G 5C,9G      5C,9G 3C,9G 3C,8H 2H,7G 5C,9H 4C,8H 4C,9G 3C,9G 5C,9G 5C,9G 9C 4C,9G      6C,9G 4C,9G 5C,9G 3C,9G 4C,9G 4C,9G Rice 9C 5C,9G 9C 3C,9G 5C,9G 2C,9G      9C 8G 4C,9G 8G 6C,9G 9C 9C 9C 9C 9C 9C 5C,9G 5C,9G 3C,8G Sorghum 9C 9C      10C 2C,9G 5C,9G 5C,9G 9C 2C,9G 9C 9C 9C 9C 9C 9C 9C 5C,9G 9C 9C 5C,9G      3C,8H Cheatgrass 10C 9C 10C 5C,9G 9C 9G 9G 5G 3C,9G 6G 9C 9C 9C 9C 9C 9C      9C 3C,9G 4C,8G 4C,8G Sugar Beets 10C 10C 10C 10C 10C 10C 10C 5C,9H 10C      3C,9H 9C 10C 10C 10C 10C 10C 10C 9C 10C 3C,7H Velvetleaf 10C 9C 10C      5C,9H 10C 5C,9H 5C,9H 3C,6H 9C 3C,8H 10C 9C 10C 9C 10C 10C 10C 9C 3C,5H      1C Giant Foxtail 9C 4C,9G 10C 3C,9G 9G 6G 9C 2C,8G 10C 9C 10C 9C 10C 10C      9C 9C 9C 9C 9C 3C,7H Barley 9C 9G 4C,9G 9G 9G 9G 2C,6G 5G 6G 2G 4C,9G      4C,9G 5C,9G 3C,9G 9C 4C,9G 4C,9G 3C,7G 2C 0 PREEMERGENCE Cotton 3C,9G 8G 9      G 5G 9G 8G 9G 0 3C,9G 0 9G 9G 9G 9G 9G 9G 9G 9G 4C,8G 7G Morningglory 9G      9G 9G 2C,7H 9G 9G 2C,8H 2C,6H 9G 2C,4H 9G 9G 9G 9G 9G 9G 9G 9G 8H 2H      Cocklebur 9H 8H 9H 2C,3H 9H -- 8H 2C,4G 9H 1C,2G 9G 9H 9H 9H 9H -- 9H 9H      4G -- Nutsedge 10E 9G 9G 6G 10E 9G 4C,9G 4G 9G 2G 10E 10E 10E 10E 10E      10E 10E 10E 3G 5G Crabgrass 3C,8G 2C,7G 10E 0 5G 0 3C,7H 0 3C,7H 0 8G 7G      4C,8G 4C,8H 10E 2G 8H 0 9G 0 Barnyardgrass 9H 3C,9H 3C,9H 3G 3C,8H 2C,7H      5C,9H 5G 9H 0 9H 9H 9H 9H 9H 9H 9H 9H 3C,9H 3G Wild Oats 3C,8G 2C,7G      2C,8H 2C,7G 2C,8G 7G 4G 8G 2C,4G 3C,9G 4C,8G 6C,9H 4C,8G 6C,9H 4C,9G      3C,9H 3C,5G 2C,3G 0 Wheat 10C 4C,9H 10H 8H 3C,9H 7G 5G 0 6G 0 4C,9H      3C,9G 5C,9H 8G 10H 4C,8G 2C,9H 3C,8H 3G 0 Corn 10C 9G 9G 2C,7G 9G 2C,7G      9G 8G 9G 9G 2U,9G 2U,9G 9H 9G 9H 9H 9H 9H 3C,9H 4C,8G Soybean 9H 8H 9H      2C,6G 3C,8H 2C,7G 4C,8H 3C,7H 9H 2C,6G 9H 9H 9H 9H 9H 9H 9H 9H 9H 2H      Rice 10E 10H 10E 9H 10E 10E 9H 3C,8H 10E 2C,8H 10E 10E 10E 10E 10E 10E      10E 10E 9H 7H Sorghum 10E 10E 9H 9H 10H 10H 10H 9H 10E 3C,8H 9H 4C,9H      10E 10H 10E 10E 10E 10H 3C,9H 4C,9G Cheatgrass 10H 9H 9H 8H 9H 9H 9H      1C,4G 9H 4G 9H 9H 9H 9H 9H 9H 9H 8H 7G 6G Sugar Beets 5C,9G 5C,9G 4C,9G      3C,8G 3C,9G 2C,6G 4C,9G 5G 9G 2C,6G 9G 9G 9G 9C 9C 9G 3C,9G 9G 4C,8G 4H      Velvetleaf 3C,9G 3C,9G 2C,8G 2C,7H 9G 9G 2C,7H 3C 3C,8H 2C 4C,9G 8G      5C,9G 8G 4C,9G 4C,9G 9C 7H 2C 2G Giant Foxtail 3C,9H 3C,9H 2C,9H 2C,5H      8G 5G 7G 2G 9H 5G 9H 9H 9H 9H 9H 9H 9H 10H 3C,8H 3G Barley 10C 9G 9C 8G      9G 9G 7G 6G 9G 6G 3C,9G 2C,9G 4C,9H 4C,9H 9H 9H 3C,9H 4C,9H 4C,8G      0        CMPD 87 CMPD 88 CMPD 89 CMPD 90 CMPD 91 CMPD 92 CMPD 93 CMPD 94 C      MPD 95  CMPD 96 CMPD 97 Rate kg/ha 0.05 0.01 0.05 0.05 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01        POSTEMERGENCE Cotton 4C,9H 4C,8H -- -- -- -- -- -- -- -- -- -- -- --      4C,9G 1C,5G 0  0 4C,9G 4C,9G 9C 4C,9H Morningglory 5C,9G 3C,9G 2C 0      3C,8H 2C,7G 2C,4H 0 2C,4G 2G 2C,7G 2H 3C,8H 2C,6H 5C,9G 5C,9G 0 0 10C      10C 10C 10C Cocklebur 9C 3C,8H 4C,9H 3C,8H 5C,9H 4C,8H 4C,9H 0 3C,8H      1C,5G 4C,8H 2C,7H 3C,8H 2C 4C,9H 3C,8H 4G 3G 10C 10C 10C 4C Nutsedge      4C,9G 3C,5G 2C,6G 6G 2C,8G 3G 0 0 0 0 0 0 0 0 6G 0 0 0 5C,9G 3C,8G 10C      9C Crabgrass 5C,9G 4G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 7G 2G 4C,8G 5G      Barnyardgrass 9C 9C 3C,6G 4G 3C,8H 0 2G 0 0 0 3C,6H 0 2C,7G 3G 4C,9H      2C,7H 0 0 10C 10C 10C 10C Wild Oats 6C,9G 4C,9G 2C,2G 2G 2C,5G 2C,3G      3C,5G 2G 0 0 0 0 4G 0 2G 0 0 0 9G 2C,5G 4C,9G 3C,6G Wheat 3C,9G 3C,7G 6G      3G 3C,9G 2C,7G 2C,4G 2G 0 0 0 0 2G 0 4G 3G 0 0 9G 2C,6G 3C,9G 8G Corn 9C      9C 2C,6H 2G 3C,8H 3G 0 0 0 0 3C,7H 0 2C,7H 0 0 0 0 0 2G 0 2C,7G 2G      Soybean 5C,9G 4C,9G 4C,9G 4C,8G 5C,9G 3C,9H 3C,7H 0 0 0 3C,9G 2C,6H      3C,8H 2C,7H 4C,9G 3C,7H 0 0 4C,9G 4C,9G 9C 9C Rice 4C,9G 4C,9G 3C,8G 7G      2C,8G 2C,5G 4G 0 2G 0 4G 0 4G 3G 2C,5G 0 0 0 9C 4C,8G 9C 5C,9G Sorghum      9C 9C 3C,8H 6G 3C,9H 2C,8H 2C,7H 0 3G 0 2C,8H 1C,5G 2C,8H 2C,7G 4C,9G      3C,9G 0 0 9C 9C 10C 10C Cheatgrass 6C,9G 2C,9G 2C,9G 2C,8G 9G 2C,9G 9G      4G 0 0 7G 0 5G 0 10C 4G 0 0 2C,5G 0 4C,9G 6G Sugar Beets 10C 5C,9G 10C      1C,3G 3C,9G 0 2C,5G 0 0 0 4C,8G 2C,7G 5C,8G 3C,7G 9C 2C,3H 0 0 4C,9G      2C,3G 10C 10C Velvetleaf 9C 3C,4H 3C,9H 2C,7G 4C,9G 2C,7G 2C,7G 5G 0 0      2C,4H 2G 3C,7H 2C,2H 4C,9H 2C,4H 3G 2G 10C 5C,9G 10C 10C Giant Foxtail      10C 9C 4G 0 5G 2G 2G 0 0 0 4G 0 6G 2G 2C,7G 2G 0 0 4C,9G 3C,9G 5C,9G 6G      Barley 3C,6G 0 5G 0 5G 5G 3G 0 0 0 2G 0 0 0 2G 0 0 0 9G 6G 9G 5G      PREEMERGENCE Cotton 5G 4G 0 0 0 0 0 0 0 0 0 0 2G 0 5G 0 0 0 2C,8G 6G 9G      9G Morningglory 9G 8H 0 0 2C,3G 0 0 0 0 0 0 0 0 0 3C,8G 5G 0 0 9G 8G 9G      9G Cocklebur 8H 8G -- 2G 3C,8H 0 0 0 0 -- 2C 0 0 -- 2C,4H 0 0 -- 9H      3C,8H 3G 5G Nutsedge 7G 4G 4G 0 2G 0 0 0 0 0 0 0 0 0 0 0 10E 4G 10E      3C,9G 10E 10E Crabgrass 5G -- 2G 0 2G 0 0 0 0 0 9G 8G 0 0 2C,5G 2G 0 0      2C,7G 5G 10E 2C,5G Barnyardgrass 9H 7H 0 0 2G 0 0 0 0 0 0 0 0 0 4C,9H 5G      0 0 9H 2C,7H 9H 9H Wild Oats 2C,4G 0 0 0 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 7G      0 3C,8G 2C,6G Wheat 5G 0 7G 0 4G 0 0 0 0 0 0 0 0 0 7G 0 0 0 9G 9G 10H 9H      Corn 9H 3C,9G 2C,3H 0 3C,6G 2G 0 0 0 0 0 0 1C 0 2C,3G 0 0 0 4C,7G 1C,3G      3C,8G 3G Soybean 9H 3C,6H 2C,3G 0 3C,5G 1C,3G 0 0 0 0 1C,2G 0 2C,4G 0      2C,3G 0 0 0 9G 3C,7H 9H 9H Rice 9H 5G 3C,8H 0 2C,3H 0 0 0 0 0 0 0 0 0 5G      0 6G 0 10E 8G 10E 9H Sorghum 10H 4C,9H 2C,9H 0 3C,7H 2C,3H 0 0 0 0 2C,5G      1C 3C,7H 0 4C,9H 3C,8H 4G 0 10E 6C,9G 10E 5C,9H Cheatgrass 9H 5G 8G 2G      8H 3G 0 0 0 0 0 0 0 0 8G 0 0 0 7G 7G 9G 7G Sugar Beets 4C,9G 3G 6G 0      2C,4G 4G 0 0 0 0 4G 2G 2H 0 4C,8G 5G 6G 0 4C,9G 8G 9G 9G Velvetleaf 7H      3G 0 0 2C,3H 0 0 0 0 0 0 0 2G 0 3G 0 0 0 4C,9G 2C,8G 5C,9G 7H Giant      Foxtail 4C,9H 4C,8G 0 0 3G 0 0 0 0 0 0 0 0 0 3C,8H 4G 0 0 2C,9G 8G 2C,7G      2C,5G Barley 9G 0 8G 0 2C,7H 2G 0 0 0 0 0 0 0 0 3G 0 0 0 9G 7G 9G      9G       CMPD 98 CMPD 99 CMPD 100 CMPD 101 CMPD 102 CMPD 103 CMPD 104      CMPD 105 CMPD 106 CMPD 107 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0      .01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE Cotton 4C,9G 3C,9H 9C 3C,9G 4C,9H 2C,7G 3C,9G 2C,4G      4C,9H 3C,8H 9C 4C,9H 9C 4C,9G 5C,9G 4C,9H 4C,9G 4C,9H 10C 5C,9G Morninggl      ory 9C 9C 10C 10C 3C,5G 2H 4C,9G 3C,8H 10C 5C,9G 10C 4C,9G 10C 10C 10C      3C,8G 10C 0 10C 2H Cocklebur 10C 5C,9G 10C 10C 3C,9H 6G 5C,9G 3C,8H 9C      4C,9G 10C 10C 10C 10C 9C 10C 10C 10C 10C 10C Nutsedge 4C,9G 4C,8G 10C 9C      3C,9G 3G 3C,8G 0 5C,9G 4C,9G 9C 5C,9G 9C 9C 5C,9G 8G 9C 4C,8G 5C,9G      3C,8G Crabgrass 1C 0 2G 0 0 0 2G 0 0 0 0 0 3G 0 3G 0 5G 0 3C,7G 2G      Barnyardgrass 9C 3C,8H 3C,9H 1C,4H 2H 0 2C,5H 0 3C,8H 1H 3C,9H 7H 10C 9C      9C 3C,8H 10C 5C,9H 10C 9C Wild Oats 5G 0 3C,7G 0 0 0 2C,5G 0 3C,6G 3G      2C,5G 2G 3C,9G 3C,7G 3C,7G 3C,5G 3C,9G 3C,8G 3C,9G 3C,8G Wheat 2C,7G 3G      2C,8G 7G 0 0 2C,7G 3G 5C,9G 7G 7G 2G 2C,9G 3C,9G 6C,9G 2C,8G 3C,9G 5C,9G      5C,9G 3C,9G Corn 0 0 10C 10C 3G 0 3C,9H 4G 4C,9H 2C,7G 1H 0 0 0 0 0 0 0      9C 3C,9G Soybean 4C,9G 4C,9G 9C 4C,9G 3H 0 3C,7H 2C,5H 5C,9G 4C,9G 3C,9G      8H 9C 9C 9C 5C,9G 5C,9G 5C,9G 9C 5C,9G Rice 4C,9G 5G 4C,9G 8G 2G 0 7G 0      8G 0 5C,9G 7G 9C 3C,9G 5C,9G 4C,9G 5C,9G 5C,9G 9C 5C,9G Sorghum 10C 9C      5C,9G 10C 4C,9G 7H 2C,9G 3C,8H 9C 4C,9H 9C 9C 9C 9C 9C 5C,9G 10C 3C,9H      9C 9C Cheatgrass 3C,7G 0 9C 3C,8G 2C,5G 0 8G 2G 4C,9G 3C,7G 8G 3G 7G 3G      7G 5G 5C,9G 5C,9H 10C 2C,8G Sugar Beets 10C 4C,8G 10C 9C 3C,5G 1C 10C      3C,7G 9C 3C,7G 10C 10C 10C 10C 10C 4C,9H 10C 10C 10C 9C Velvetleaf 4C,9H      4C,8H 10C 10C 3C,8H 3C,7G 4C,8H 3C,7H 9C 4C,9G 10C 5C,9G 10C 10C 10C      4C,8G 9C 4C,9H 10C 9C Giant Foxtail 3C,8G 2C,6G 2C,7G 3G 2G 0 2C,7G 2G      4C,9G 4G 6G 3G 3C,7H 3C,6G 4C,8G 7G 4C,8G 3C,8G 5C,9G 3C,8G Barley 2C,2G      0 9C 8G 2G 0 2C,6G 0 2C,9G 2C,6G 7G 2G 3C,9G 3C,8G 8G 6G 2C,9G 3C,8G      4C,9G 9G PREEMERGENCE Cotton 3C,8G 2C,4G 4H 6G 1C 0 0 0 8G 2C,3G 9G 2G      9H 5G 2C,8H 0 2C,4G 2G 9G  9G Morningglory 9H 4H 9G 6H 2G 0 3C,4H 0 8H      3C,4H 9G 6H 9G 2C,5G 3H 0 2C,5G 0 5G 2G Cocklebur 2C,7G 0 8H 8H 5G 0      2C,2G 0 8H 3C,3H 9G 9H -- 1H 8H 2H 2C,5G 3C,7H 9H 9H Nutsedge 10E 10E      10E 9G 9G 0 3G 0 10E 0 10E 10E 9G 10E 9G 0 8G 0 10E 10E Crabgrass 2C,3G      2G 10E 6G 5G 0 0 0 0 0 2G 0 4G 0 0 0 10H 0 8G 2C,5G Barnyard Grass 9H      3C,7H 7H 0 0 0 0 0 6H 2G 8H 4G 9H 2G 4C,9H 0 0 0 5C,9H 9H Wild Oats 2C 0      7G 5G 0 0 0 0 3C,8G 0 5G 0 7G 0 2C,6G 0 0 2G 8G 5G Wheat 7G 0 9G 8G 0 0      5G 0 9H 3C,8G 7G 2G 9H 5G 8H 0 5G 5G 9H 7G Corn 0 0 3C,9G 7G 0 0 0 0      3C,9H 3C,6G 0 0 3G 0 0 3G 0 0 9G 7G Soybean 3C,8H 3C,4G 3C,8H 6H 2C 0 2C      0 3C,6H 3C,5H 8H 3C,7H 9H 6H 3C,7H 3C,3H 9H 3C,4H 9H 3C,6H Rice 10H      3C,7G 9H 9H 6G 0 4G 0 8H 0 10H 3C,7G 9H 7G 10H 0 8H 3C,6G 10E 9H Sorghum      10H 10H 10H 9H 3C,8G 2G 2C,6G 0 10H 4C,8H 10E 9H 6C,9H 9H 9H 2C 4C,9H      3C,8H 10H 9H Cheatgrass 9G 2G 9G 8H 0 0 5G 0 8G 7G 8G 5G 8G 0 8G 0 8G 5G      10E 4C,9G Sugar Beets 4C,9G 8H 4C,9G 6H 2H 2G 7G 0 4C,9G 4C,8H 9G 9G      5C,9G 8G 5C,9G 7G 3C,8G 7H 9C 10C Velvetleaf 2C,7H 2C,3H 4C,9G 8G 3H 0      3C,5G 0 4C,8H 1H 7H 1H 4C,8G 3G 6H 2G 2C,2H 2H 5C,9G 8H Giant Foxtail      2C,9H 3G 4G 0 0 0 3G 0 8G 2G 7G 1C 3G 0 3G 0 0 0 9H 3C,7G Barley 2C,8G      7G 9G 8G 0 0 5G 0 9G 3C,7G 9G 6G 8G 4G 8G 3G 9G 3C,7H -- --        CMPD 108 CMPD 109 CMPD 110 CMPD 111 CMPD 112 CMPD 113 CMPD 114 CMPD      115 CMPD 116  CMPD 117 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE Cotton 5C,9G 10C 9C 5C,9G 6C,9G 3C,9G 4C,8H 3C,7H 4C,9H      4C,8G 1H 0 2C,3H 2G 4C,9G 9H 5C,9G  10C 5C,9G 4C,8G Morningglory 10C 9C      2C,7G 5G 10C 10C 4C,8H 3C,7G 10C 4C,9G 0 0 1H 0 10C 5C,9G 10C 10C 5C,9G      4C,9H Cocklebur 10C 10C 10C 10C 10C 10C 4C,9H 2C,4G 10C 4C,8H 1H 0 2H 2H      8G 2G 10C 2C,3H 4C,9H 3C,5H Nutsedge 3C,8G 2C,7G 4C,9G 6C,9G 5C,9G 3C,8G      2C,4G 0 3C,9G 0 0 0 4C,9G 0 10C 4C,8G 9C 3C,8G 9G 8G Crabgrass 3C,7G 5G      3C,6G 5G 3C,5G 3G 0 0 2G 0 2G 0 3C,6G 3G 6G 2G 3C,6G 2C 0 0 Barnyardgrass       9C 9C 10C 9C 9C 4C,9H 3C,7H 2C,5H 9C 3C,7G 5C,9H 3C,6G 9C 3C,8H 9C      5C,9G 9C 9C 2H 0 Wild oats 4C,9G 3C,7G 4C,9G 4C,9G 3C,9G 2C,3G 0 0 3C,5G      0 3C,5G 2G 9C 3C,6H 5C,9G 3G 3C,7G 3G 0 0 Wheat 9C 5C,9G 9C 2C,9G 3C,9G      3G 0 0 4G 0 9C 8G 9C 3C,7H 9G 2C,9G 5C,9G 9G 2G 0 Corn 4C,9G 4C,9H 3C,8H      3C,7H 3C,8H 2G 3C,7G 0 9G 3C,6G 2C,9G 2C,5H 4H 0 2G 0 6H 0 0 0 Soybean      5C,9G 9C 9C 4C,9G 4C,9G 3C,6G 4C,9G 3C,8G 4C,9G 4C,8G 2G 0 3C,8G 0 5C,9G      4C,9G 9C 5C,9G 4C,9G 3C,7H Rice 9C 9C 9C 9C 9C 4C,9G 3G 0 4G 0 9C 8G      5C,9G 9G 9C 9C 9C 3C,8G 2G 0 Sorghum 10C 9C 9C 9C 9C 4C,9H 3C,7H 0 3C,9G      3C,8H 4C,9G 3C,7H 9C 4C,9G 9C 9C 9C 9C 3C,3H 0 Cheatgrass 5C,9G 3C,8G      5C,9G 8G 4C,8G 6G 0 0 0 0 3C,9G 0 9C 3C,7G 8G 6G 3C,8G 3C,6G 0 0 Sugar      Beets 10C 10C 10C 9C 9C 9C 3C,5H 3C,8H 10C 4C,8H 3C,8G 3G 3C,7H 3C,6G 9C      9C 10C 9C 9C 3C,7G Velvetleaf 9C 10C 9C 4C,8H 9C 9C 3C,7H 0 4C,9G 3C,6H      4G 0 2H 0 9C 9C 10C 9C 3C,8H 3C,4H Giant foxtail 5C,9G 4C,8G 4C,8G 2C,6G      3C,8G 3G 2G 0 3C,7G 2C,2G 3C,8H 2G 9C 3C,8H 9C 4C,9G 4C,9H 3C,7G 0 0      Barley 3C,9G 8G 4C,9G 2C,8G 9G 5G 0 0 3G 0 2C,9G 9G 10C 2C,8G 3C,8G      3C,6G 3C,8G 3G 0 0 PREEMERGENCE Cotton 3C,8G 7G 8H 3G 8G 7G 0 0 2G 0 0 0 2      H 0 3C,5G 6G 3C,5G 0 2G 0 Morningglory 9H 3G 5G 1H 9G 7H 2C,3H 0 8G 0 0      0 0 0 7H 0 2C,6G 0 7H 0 Cocklebur 9H 9H -- 3C,8H 9H 8H 0 --  7H 2C,5G 0      -- 0 0 3G 0 -- 3G 3C,5G 1C Nutsedge 10E 4C,9G 10E 10E 10E 10E 10E 0 10E      0 0 0 0 0 9G 0 8G 0 4G 0 Crabgrass 4C,8G 3C,7G 4C,8G 2C,2G 3C,5G 3G 2G 0      2G 0 2G 0 7G 3G 4G 0 9G 0 0 0 Barnyardgrass 9H 3C,9H 5C,9H 2C,7H 9H      3C,9H 7H 0 9H 6H 4G 0 6G 0 8H 2G 3C,9H 2G 0 0 Wild Oats 5C,9G 3C,8G      4C,8H 3C,7G 3C,8G 3G 0 0 0 0 0 0 0 0 2C 0 1C 0 0 0 Wheat 9H 3C,9G 3C,9H      6G 3C,7G 3G 0 0 0 0 2G 0 7G 0 2G 0 3C,7H 0 0 0 Corn 3C,9H 3C,8G 3C,7G      2C,3G 3C,7G 2C,2G 3C,3G 0 2G 3G 2G 0 0 0 0 0 3G 0 0 0 Soybean 3C,8H      3C,7H 9H 3C,6G 4C,8H 3C,6H 2C,4H 0 3C,7G 3C,4G 0 0 0 0 3C,6H 2C 8H 3C,6H      3C,5G 2C Rice 10E 4C,9H 10E 10H 10E 9H 2C,5G 0 3C,7H 3G 2C,5G 0 2C,5G 0      9H 3C,5G 10H 5G 0 0 Sorghum 10E 4C,9H 10H 9H 5C,9H 5C,9H 3C,6G 0 8H      3C,5G 3C,5G 0 3C,7G 0 9H 3C,7G 10E 8G 0 0 Cheatgrass 10E 3C,8G 5C,9G 8H      9G 3C,7G 0 0 4G 0 0 0 0 0 7G 0 9H 2G 0 0 Sugar Beets 10C 4C,9G 9C 9G 9C      9C 5G 2G 3C,9H 7H 1H 0 4H 0 4C,9G 7H 4C,9G 6H 3C,7G 2H Velvetleaf 5C,9G      3C,5H 5C,9G 3C,7G 4C,8H 5H 2G 0 2C,2H 0 2G 0 0 0 3C,5H 0 3C,8H 1C 2C 0      Giant Foxtail 9H 3C,7G 3C,8G 3C,5G 3C,8G 3C,6G 1H 0 7G 0 2G 0 3G 0 7G 0      3C,8G 0 0 0 Barley -- 2C,8G 8G 7G -- 2C,5G 0 0 0 3G 9G 0 9G 2G 2C,9G 3G      9G 0 0 0        CMPD 118 CMPD 119 CMPD 120 CMPD 121 CMPD 122 CMPD 123 CMPD 124 CMPD      125 CMPD 126  CMPD 127 CMPD 128 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0      .05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05  0.01 0.05 0.01      0.05 0.01        POSTEMERGENCE Cotton 9H 8H 9C 9C 1C 0 10C 4C,9G 0 -- 4C,9H 4C,9H 4C,9H 3      C,8H 5C,9G 9C 9H -- 10C 3C,9G 2C,9H 2C,5H Morningglory 9C 3C,8H 10C 10C      3H 0 10C 10C 0 -- 10C 9C 4C,9G 4C,9H 10C 10C 4C,9G -- 10C 9C 6C,9G 4C,8H      Cocklebur 4C,9G 3C,7H 10C 10C 1H 0 10C 9C 2H -- 9C 4C,9H 5C,9G 4C,9H 10C      10C 4C,9G -- 10C 5C,9H 3C,9H 3C,4H Nutsedge 9C 4C,8G 5C,9G 4C,9G 0 0 9G      8G 0 -- 3C,8G 2C,5G 9G 3C,9G 10C 5C,9G 8G -- 2C,8G 8G 2C,6G 0 Crabgrass      0 0 3C,5G 2G 0 0 3C,5G 2G 0 -- 2C,5G 2G 3C,4G 2G 3C,8G 5G 0 -- 0 0 0 0      Barnyardgrass 4H 0 9C 9C 4H 0 9C 9C 1H -- 9C 4C,9H 5C,9H 4C,8H 5C,9H      3C,6H 0 -- 3C,9H 2C,7H 2C,5H 0 Wild Oats 0 0 4C,8G 3C,5G 3C,7G 0 4C,9G      3C,5G 2C,5G --  4C,9G 5G 4C,9G 7G 8G 4G 0 -- 2C,6G 2C 2C 0 Wheat 0 0 9C      4C,9G 8G 0 5C,9G 8G 6G -- 9G 8G 3C,9G 9G 8G 4G 0 -- 9G 9G 2C 0 Corn 0 0      2C,7H 3H 0 0 0 0 0 -- 0 0 0 0 3C,9G 9G 2H -- 3C,9G 3C,7H 2C,8H 2C,3G      Soybean 3C,7H 3C,7H 5C,9G 5C,9G 3C,4G 0 5C,9G 4C,9G 2G -- 4C,9G 3C,8G      5C,9G 4C,9G 4C,9G 4C,9G 3C,5G -- 3C,8H 3C,8G 3C,8H 2C,3H Rice 2G 0 9C 9C      8G 0 9C 9C 3G -- 9C 5C,9G 9C 5C,9G 5C,9G 3C,9G 0 -- 2C,9G 6G 4G 0      Sorghum 6H 0 9C 9C 4C,9H 0 9C 4C,9G 2C,5G -- 9C 4C,9G 5C,9G 3C,9G 5C,9G      3C,9G 3C,6G -- 5C,9G 2C,9G 9H 2C,7H Cheatgrass 0 0 5C,9G 4C,8G 3C,8G 0      4C,9G 4C,9G 3C,8G -- 9C 9G 6C,9G 3C,9G 9C 9C 5G -- 10C 3C,9G 5G 3G Sugar      Beets 9C 3C,7H 10C 9C 1H 0 10C 10C 0 -- 10C 4C,8H 9C 4C,9H 10C 10C 3C,8G      -- 10C 6C,9G 3C,9H 2C,3G Velvetleaf 4C,8H 3C,6H 10C 9C 1C 0 10C 9C 1C --      9C 3C,7H 9C 4C,8H 10C 10C 3C,6G -- 9C 9C 3C,7H 2C,4G Giant Foxtail 1C 2G      9C 9C 2C,5G 0 9C 4C,9G 0 -- 5C,9G 3C,7H 6C,9G 4C,8G 3C,7G 5G 0 -- 2C,9G      6G 3G 2G Barley 0 0 5C,9G 4C,9G 7G 0 4C,9G 3C,8G 8G -- 3C,8G 3C,6G 5C,9G      2C,9G 8G 5G 0 -- 9G 6G 4G 0 PREEMERGENCE Cotton 2G 0 4C,8G 6G 0 0 3C,7H      0 0 -- 5G 0 2G 0 9G 8G 0 -- 2C,8G 4G 0 0 Morningglory 8H 0 9G 3C,7H 0 0      3C,7H 3C,3H 0 -- 3C,8H 2C,6H 7H 1H 9G 9G 1H -- 9G 3C,9H 2C,3H 0 Cocklebur       3C,3H 0 9H 2C,2H 0 0 3C,8H 3C,3G 0 -- 3C,6H -- 2H 1H 9H 9H 7G -- 3C,8H      3C,7H 2H 0 Nutsedge 9G 0 10E 3C,9G 0 0 4C,8G 0 0 -- 9G 10E 3G 0 10E 10E      0 -- 10E 2C,9G 8G 0 Crabgrass 0 0 3C,4G 3C,5G 0 0 3C,6G 3G 0 -- 7G 0 0 0      5G 0 0 -- 2C 0 2G 0 Barnyardgrass 3G 0 4C,9H 3C,7H 0 0 4C,9H 4G 0 --      3C,9H 3C,8H 5G 0 9H 3C,7G 0 -- 4C,8H 2C,3G 5G 0 Wild Oats 0 0 3C,6G 0 0      0 2G 0 0 -- 3G 0 2G 0 6G 3G 0 -- 4C,7G 3G 0 0 Wheat 0 0 3C,9H 3G 0 0 8G      6G 0 -- 8G 0 3G 0 7G 2G 0 -- 8G 3G 0 0 Corn 7G 0 3C,6H 0 0 0 2H 0 0 --      1H 0 0 0 9H 2C,9G 0 -- 4C,8H 2C,3G 0 0 Soybean 2C,6H 0 4C,8H 3C,6H 0 0      3C,7H 0 0 -- 3C,5H 2C,3H 3C,6G 0 2C,7H 3C,2H 2G -- 3C,5G 2C 2C 0 Rice 4G      0 10E 3C,8H 0 0 3C,8H 4G 0 -- 9H 3C,8G 3C,6G 0 9H 9H 4G -- 9H 3C 0 0      Sorghum 3G 0 5C,9H 3C,8H 0 0 4C,9H 2C,6G 0 -- 5C,9H 3C,9H 3C,7G 2C 9H      5C,9H 2C -- 5C,9H 3C,8H 2C,3G 0 Cheatgrass 0 0 5C,9G 3C,9G 0 0 9H 7G 0      -- 5C,9G 8G 8G 0 9H 8G 0 -- 4C,9H 3C,8H 0 0 Sugar Beets 7G 0 9C 9C 3G 0      9C 4C,8H 2G -- 9C 5G 9G 4G 10C 9C 8G -- 3C,9G 3C,9G 0 0 Velvetleaf 3C,4G      0 4C,8H 3C,6H 0 0 3C,7H 1C 0 -- 5G 0 2C,3G 2H 5C,9G 4C,8H 0 -- 4C,8H      3C,6G 0 0 Giant Foxtail 0 0 4C,9H 3C,8G 0 0 3C,8H 0 0 -- 9H 2G 0 0 8G      2C,5G 0 -- 3C,8H 6G 0 0 Barley 4G 0 3C,9G 3C,8G 0 0 8G 0 0 -- 7G 3C,7G      7G -- 8G 8G 0 -- 8G 2G 0 0        CMPD 129 CMPD 130 CMPD 131 CMPD 132 CMPD 133 CMPD 134 CMPD 135 CMPD      136 CMPD 137  CMPD 138 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01  0.05 0.01        POSTEMERGENCE Cotton 3C,9H 2C,8H 2C,8H 3C,6H 10C 5C,9G 9C 10C 9C 7G 9C 3      C,8H 2C,3G 1C 8H 2C,2G 10C 4C,9G 3C,7G 0 Morningglory 3C,8H 2C,8G 6C,9G      4C,8H 10C 4C,9G 10C 9C 9C 7G 10C 9C 4C,8H 3C,4H 4C,8H 3C,8H 10C 4C,8G      10C 3C,7H Cocklebur 9C 4C,9H 10C 2C,3H 10C 10C 10C 10C 10C 5C,9G 10C 10C      3C,5H 3G 4C,8H 3C,5G 10C 10C 2H 0 Nutsedge 6G 2C,7G 3C,8G 2C,4G 9C 3C,8G      4C,9G 2C,9G 9C 3C,9G 9C 9G 0 2C,4G 3C,7G 3C,5G 3C,9G 3C,8G 0 0 Crabgrass      0 0 0 0 4C,8G 2G 4C,8G 3G 5C,9G 6G 3G 0 2G 0 3G 0 4G 0 0 0 Barnyardgrass      2G 3G 2C,6H 2C,6G 9C 9C 10C 9C 10C 10C 9C 5C,9H 3C,8H 3C,7H 9C 4C,9H 9C      3C,9H 9H 4C,9H Wild Oats 2G 0 2C,5G 3G 3C,9G 5G 4C,9G 3C,6G 4C,9G 4C,9G      4C,9G 2G 0 0 2C,3G 2G 0 0 0 0 Wheat 2G 0 2C,9G 2G 3C,9G 9G 3C,9G 9G      4C,9G 9C 9G 4G 2G 0 0 0 2G 0 7G 0 Corn 2C 0 3C,8H 2C,2H 10C 3C,9G 5C,9G      4G 3C,9H 2H 0 3G 3C,9G 3C,7H 9C 3C,8H 0 0 0 0 Soybean 2H 0 4C,8H 3C,4H      9C 9C 5C,9G 9C 9C 4C,9G 4C,9G 3C,8H 3G,8G 4H 4C,9G 4C,8H 3C,9G 1H 3C,5H      2H Rice 2C,5G 0 3C,9G 2C,4G 9C 9C 9C 9C 9C 5C,9G 9C 7G 3G 0 2C,3G 0      5C,9G 3C,6G 3C,7G 3G Sorghum 9G 3C,8H 2C,9G 2C,7H 10C 9C 9C 9C 10C 5C,9G      9C 3C,8H 3C,9H 3C,7H 9C 3C,9G 9C 9G 5C,9G 4C,9H Cheatgrass 2C,8G 5G 8G      8G 9C 9C 10C 9C 10C 9C 9C 9G 8G 6G 5C,9G 7G 8G 5G 3C,8G 6G Sugar Beets      3C,6G 2C,7G 3C,9G 3C,5H 9C 10C 10C 10C 10C 9C 9C 9C 8H 5H 9C 3C,7G 9C      3C,8G 3C,4H 2H Velvetleaf 2C,8G 2C,7G 5C,9H 3C,7G 10C 10C 10C 5C,9G 10C      10C 9C 5C,9G 2G 2G 3C,7G 1C 10C 3C,8G 3C,7H 2G Giant Foxtail 2G 3G 2C,7G      3G 9C 4C,9G 9C 3C,8G 9C 4C,8G 5C,9G 3C,7G 2C,8G 7G 9C 3C,7G 3C,9G 3C,7G      3C,7G 5G Barley 0 0 7G 0 4C,9G 5G 9C 7G 4C,9G 8G 7G 0 0 0 2G 0 0 0 0 0      PREEMERGENCE Cotton 2G 0 4G 0 9G 6G 8G 3H 9G 2G 7H 1H 0 0 0 0 6G 0 0 0      Morningglory 2C,6H 0 0 0 9G 3G 2C,3G 2G 7G 0 9G 7G 1H 0 3C,7H 0 9G 4G 0      0 Cocklebur 3C,8H 0 0 0 8H 9H 9H 2C,2H 8H 2C,8H 8H -- 4H -- 3C,5G 2C      3C,5H 2C,5G -- 0 Nutsedge 9G 0 0 0 10E 10E 9G 3C,9G 10E 10E 10E 9G 10E 0      7G 0 9G 0 0 0 Crabgrass 2G 0 0 0 5G 0 3C,9G 5G 8G 0 3G 0 0 -- 3C,7G 0 3G      0 0 0 Barnyardgrass 6G 0 3G 0 9H 5G 3C,9H 3C,7G 9H 8G 9H 7H 5G 0 4C,8H 0      9H 0 0 0 Wild Oats 2G 0 0 0 3C,6G 0 3C,5G 0 3C,7G 2C,3G 6G 0 0 0 0 0 0 0      0 0 Wheat 0 0 0 0 9H 0 3C,9H 0 3C,9H 5G 7G 0 0 0 0 0 3G 0 0 0 Corn 3G 0      0 0 3C,9H 2G 3C,8H 3G 3C,9H 3C,5G 3C,7G 5G 6H 0 3C,8H 2C 2G 0 0 0      Soybean 2C 0 0 0 9H 3C,4G 3C,7G 3C,5H 9H 3C,6H 3C,7H 3C,4H 0 0 3C,3G 0      3C,3H 2G 0 0 Rice 2C,8H 0 5G 0 10E 8G 10E 9H 10E 9H 10E 9H 2G 0 4G 0 9G      9G 0 0 Sorghum 3C,9H 0 2C,5G 2G 5C,9H 3C,8G 5C,9H 3C,9H 10H 3C,9H 10H      5C,9H 3C,7G 0 5C,9H 3C,6G 10H 9H 0 0 Cheatgrass 4G 0 3C,7G 2G 9H 8G 8G      8H 9H 8H 9H 8G 6G 0 8H 0 9G 0 0 0 Sugar Beets 3C,8G 0 9C 0 5C,9G 9C      5C,9G 7H 4C,9G 4C,9G 9G 8G 7G 2H 4C,8H 1H 9H 8H 4G 0 Velvetleaf 3G 0 0 0      8H 7G 2C,6H 2C,2H 7H 3G 7H 5G 0 2G 0 0 5H 0 0 0 Giant Foxtail 3G 0 2G 0      9H 6G 3C,9H 4G 9H 6G 9H 6G 2G 2G 3C,8G 0 9H 0 0 0 Barley 2G 0 7G 0 9G      2C,4G 3C,8G 2C,8G 9G 9G 9G 7G 0 0 4G 0 2C,3G 0 0 0        CMPD 139 CMPD 140 CMPD 141 CMPD 142 CMPD 143 CMPD 144 CMPD 145 CMPD      146 CMPD 147  CMPD 148 CMPD 149 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0      .05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05  0.01 0.05 0.01      0.05 0.01        POSTEMERGENCE Cotton 4C,9G 3C,8G 9C 3C,9G 5C,9H 4C,8H 10C 5G 5C,9G      4C,8H 3C,7G 2C,2G 4C,9H 4C,9H 10C 4C,8G 3C,8H 0  8H 0 9G 4C,8H Morningglo      ry 4C,9G 4C,8G 9C 5C,9G 9C 4C,8H 10C 5C,9G 10C 5C,9G 3C,8G 3C,6G 9C      5C,9H 10C 4C,8G 3C,5G 0 3C,4H 0 4C,9G 3C,8H Cocklebur 4C,9G 4C,9G 10C 8H      10C 4C,9H 9C 3C,7H 10C 9C 4C,8H 2H 10C 3C,9G 10C 4C,9H 5C,9G 2H 3C,3H 0      4C,9G 3C,8H Nutsedge 3C,5G 2C,4G 4C,9G 9G 2C,5G 3G 4C,9G 4C,9G 4C,8G      2C,5G 0 -- -- -- 4C,9G 4C,9G -- -- -- 0 -- 2G Crabgrass 5G 0 5G 0 0 0 3G      0 3G 3G 0 0 5G 0 5G 4G 2G 0 3G 0 5G 3G Barnyardgrass 9C 3C,8H 9C 5C,9H      4C,9H 3C,7H 4C,9H 3C,7H 9C 3C,8H 3C,6H 0 5C,9H 3C,7H 9C 4C,8H 4C,8H 2H      5C,9H 3C,7H 9C 3C,8H Wild Oats 2C 0 1C 0 1C 0 0 0 2C,5G 0 0 0 2G 0 0 0      1C 0 3C,7G 0 3C,8G 2G Wheat 9G 3G 5G 0 2G 0 4G 0 7G 3G 0 0 -- -- 7G --      3G 0 -- 0 -- -- Corn 0 0 3G 0 0 0 1C 0 3C,7G 2G 0 0 3C,9H 2C,5G 3C,7H 1H      2H 0 5C,9G 3C,3G 9C 3C,8H Soybean 4C,9G 4C,8G 5C,9G 3C,5H 4C,9G 1H 4C,9G      5C,9G 5C,9G 4C,9G 3C,6H 2C,2H 5C,9G 3C,9H 5C,9G 4C,8G 3C,8G 0 3C,7G 2G      5C,9G 3C,7G Rice 5C,9G 2C,5G 6C,9G 6G 5G 0 5C,9G 8G 9C 6C,9G 2C 0 9C      3C,8G 5C,9G 3C,5G 4C,9G 0 8G 2G 9C 5C,9G Sorghum 4C,9G 2C,5G 6C,9G 4C,9H      5C,9H 3C,6G 5C,9H 3C,9H 9C 6C,9G 3C,7G 2G 9C 5C,9G 9C 4C,9H 4C,9G 3G      4C,9H 3C,6G 9C 4C,9G Cheatgrass 5G 0 9C 3C,9G 9G 8G 3C,9G 8G 3C,9G 2G 0      0 3C,7G 2G 9C 9G 3C,5G 0 4C,9G 6G 8G 6G Sugar Beets 5C,9H 4C,9H 10C 9C      9C 9C 9C 9G 10C 9C 3C,8G 0 9C 9C 10C 5C,9H 3C,7G 3G 3C,7H 2H 9C 4C,8H      Velvetleaf 10C 3C,8H 10C 9C 9C 4C,7G 10C 9C 10C 4C,8H 3C,7G 0 6C,9G      3C,6G 10C 5C,9H 3C,6G 0 0 -- 4C,8G 2C Giant foxtail 5C,9G 3C,5G 3C,8G      3C,5G 3C,7G 3G 3C,7G 3C,5G 9C 5C,9G 3G 0 5C,9G 5C,9G5C,9G 3C,8G 3C,7G 0      4C,8G 3G 5C,9G 3C,8G Barley 2G 0 0 0 0 0 2C,3G 0 8G 0 0 0 7G 0 5G 0      3C,7G 0 0 0 6G 0 PREEMERGENCE Cotton 0 0 2C 0 1C 0 2C 0 3C,5G 0 0 0 1C 0 2      G 0 0 0 0 0 2C,2G 0 Morningglory 0 0 8H 0 3C,3H 0 2C,2H 0 8G 0 0 0 3C,3H      0 0 0 0 0 0 0 3C,5H 0 Cocklebur 0 0 8G 0 2C 0 2C 0 3C,3H 0 0 0 1C 0 0 0      0 -- 0 -- 2C 0 Nutsedge 0 0 9G 0 0 0 10E 0 0 0 0 0 0 0 8G 0 0 0 0 0 2G 0      Crabgrass 0 0 4G 0 0 0 2G 0 0 0 0 0 0 0 1C 0 0 0 0 0 0 0 Barnyardgrass 0      0 3C,7G 0 1C 0 3C,7H 0 7G 0 0 0 5G 0 3C,8H 0 2C 0 0 0 3C,7G 0 Wild Oats      0 0 0 0 0 0 1C 0 0 0 0 0 0 0 1C 0 0 0 0 0 0 0 Wheat 0 0 0 0 0 0 6G 0 6G      0 0 0 0 0 5G 0 0 0 0 0 2G 0 Corn 0 0 0 0 0 0 2C,3G 0 3C,7G 0 0 0 3C,5G 0      3C,4G 1C 0 0 0 0 3C,6G 1C Soybean 0 0 3C,3H 0 2G 0 3C,5H 0 3C,7G 3C,4H 0      0 3C,5G 0 2C,2H 0 0 0 0 0 3C,2H 2C Rice 0 0 9H 0 0 0 3C,9H 0 10E 2C,5G 0      0 4C,9H 0 9H 0 2C 0 0 0 3C,9H 2C,3G Sorghum 0 0 4C,8G 3C 4C,7G 0 3C,9H 0      9H 3C,9H 0 0 4C,9H 3C,7G 3C,9H 3C,5G 3C,3G 0 3C,6G 0 3C,9H 3C,8H      Cheatgrass 0 0 8G 0 2G 0 9H 0 4G 0 0 0 0 0 2C,8G 0 0 0 0 0 0 0 Sugar      Beets 0 0 9G 4G 4C,7H 0 9G 0 4C,9G 7H 0 0 4C 6H 9G 2H 4H 0 3G 4G 5H 3H      Velvetleaf 0 0 7H 0 2C 0 2H 0 3C,6H 0 0 0 2C 0 0 0 0 0 0 0 2C 0 Giant      Foxtail 0 0 3C,4G 0 3G 0 2C,5G 0 8G 0 0 0 3G 0 4C,9H 0 0 0 0 0 4C,8G 0      Barley 0 0 0 0 0 0 2C,3G 0 2C,4G 2G 0 0 2C 0 2C 0 2C 0 0 0 2G 0        CMPD 150 CMPD 151 CMPD 152 CMPD 153 CMPD 154 CMPD 155 CMPD 156 CMPD      157 CMPD 158 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05  0.01 0.05 0.01 0.05 0.01         POSTEMERGENCE Cotton 0 0 3C,7G 0 10C 9C 10C 10C 10C 3C,8H 10C 9C 2G      2H 2G 0 10C 10C Morningglory 2C,3G 0 4C,8H 0 10C 10C 10C 9C 4C,9H 2C,6G      10C 10C 4C,9G 3C,7H 2C,5G 0 9C 10C Cocklebur 2C 0 4C,8H 0 10C 10C 10C      10C 9C 4C,9H 10C 10C 7H 2H 3C,8H 2C,3H 10C 10C Nutsedge 0 0 0 0 4C,9G      4C,9G 4C,9G 9G 9G 2C,9G 9G 9G 0 0 0 0 9C 2C,9G Crabgrass 0 0 3C,5G 3G      3C,7G 3C,6G 3C,7G 3G 5G 3G 3C,6G 5G 3C,6G 2C,4G 5G 0 1H 0 Barnyardgrass      3C,9H 5G 9C 3C,9H 9C 9C 9C 4C,8H 4C,8H 3C,7H 3C,7H 3C,8H 6C,9H 3C,8H      3C,4G 2C,3H 9C 4C,9H Wild Oats 2C,9G 3C,4G 5C,9G 3C,8H 4C,9G 2C,6G 3C,7G      2C,3G 3C,8G 2C,5G 3C,5G 0 9C 4C,9G 2C,5G 9 3C,6G 2C,2H Wheat 9G 9G 9G 9G      2C,9G 9G 4C,9G 8G 8G 4G 7G 3G 3C,9G 9G 7G 4G 9G 5G Corn 3G 0 0 0 0 0 0 0      2G 2G 0 0 0 0 0 0 5G 2G Soybean 3C,7H 1H 3C,8G 3C,6G 5C,9G 9C 9C 9C      4C,9G 4C,9G 4C,9G 3C,9G 8G 3C,7G 3C,8G 2C,3H 9C 5C,9G Rice 3C,9G 5G      4C,9G 6G 5C,9G 5C,9G 5C,9G 6C,9H 5C,9G 5C,9G 4C,9G 2C,8G 6C,9G 4C,9G 6G      4G 9G 3C,8G Sorghum 3C,8H 3G 5C,9G 3C,9G 9C 9C 9C 6C,9G 4C,9G 5C,9H      5C,9G 5C,9H 5C,9G 3C,8H 3C,6G 2C,4G 2C,9G 5C,9G Cheatgrass 5G 0 8G 2C,5G      9G 8G 4C,9G 7G 8G 3C,5G 2C,5G 2G 3C,8G 2C,7G 3C,4G 2G 5C,9G 3C,6G Sugar      Beets 3C,7H 5H 4C,8G 4C,5G 10C 9C 9C 6C,9G 9C 4C,9G 5C,9G 3C,7H 3C,7H      3C,7H 3C,3G 0 10C 9C Velvetleaf 3G 0 1C 9 10C 5C,9G 10C 9C 4C,9H 3C,7H      4C,8H 3C,6H 2C,5G 3C,3G 2G 3G 10C 10C Giant Foxtail 2G 0 5C,9G 2C,5G      4C,8G 3C,7G 3C,8G 5G 3C,7G 3G 3C,7G 2C,5G 4C,9G 3C,8G 2C,7G 3G 2C,8G 4G      Barley 8G 7G 8G 6G 8G 8G 8G 5G 7G 5G 8G 5G 7G 4C,9G 4C,9G 5G 9G 3C,4G      PREEMERGENCE Cotton 0 0 1C 0 9G 8G 8G 3G 2G 4G 3C,7G 1C 0 0 0 0 5C,9G      4C,8G Morningglory 0 0 0 0 9G 6G 8H 7H 7H 0 4C,8H 5H 2C 1H 0 0 7H 6H      Cocklebur 0 0 6G 2H 9H -- -- -- 8H 8H 3C,8H 3C,5H 3H 3H 0 0 -- --      Nutsedge 0 0 0 0 10E 9G 10E 9G 3C,8G 0 10E 9G 0 0 0 0 9G 9G Crabgrass 0      0 0 0 8G 6G 7G 2G 3G 0 7G 3G 3G 0 3G 0 0 0 Barnyardgrass 0 0 2H 0 9H 8H      3C,8H 0 3C,7H 0 6H 3G 4G 0 2G 0 8G 6G Wild Oats 0 0 2C,5G 0 7G 3G 4C,8G      2C,3G 2C,3G 0 0 0 3C,6G 3G 0 0 2C,3G 2G Wheat 8G 0 3C,9H 0 9H 9G 4C,9H      8G 2C,6G 0 8G 0 2C,8H 5G 0 0 2C,8G 6G Corn 1C,1H 0 0 0 3G 0 0 0 0 0 0 0      0 0 0 0 3C,3G 0 Soybean 0 0 0 0 9H 8H 9H 3C,6H 3C,6H 2C,2H 3C,8H 3C,4H      1C,1H 0 0 0 3C,6H 5G Rice 7H 9 10H 0 10E 9H 9H 9H 9H 9G 10E 9H 9H 0 2G 0      5C,9H 8H Sorghum 3C,4G 0 9H 0 10H 9H 10H 9H 9H 3C,5G 9H 4C,9H 3C,9G      2C,5G 5G 0 5C,9H 9H Cheatgrass 0 0 0 0 8G 6G 9H 3C,7G 7G 0 5G 0 4G 0 0 0      9G 4G Sugar Beets 5G 0 5G 1H 9C 3C,7G 9G 3C,8H 4G 5G 7H 3H 5H 6G 0 0 9C      4C,9G Velvetleaf 0 0 0 0 5C,9G 4C,6H 4C,8H 3C,4H 3C,5H 1C 3C,5H 3G 2H 1H      0 0 9G 8H Giant Foxtail 0 0 5G 0 6G 2G 6G 0 5G 0 6G 2G 2C,5H 0 2H 0 7G 0      Barley 7H 0 4C,9G 0 9G 8G 9G 6G 8G 2G 8G 4G 9G 2G 2G 0 9H 4G        CMPD 159 CMPD 160 CMPD 161 CMPD 162 CMPD 163 CMPD 164 CMPD 165 CMPD      166 CMPD 167  CMPD 168 CMPD 169 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0      .05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01  0.05 0.01      0.05  0.01        POSTEMERGENCE Cotton 10C 4C,9G 3C,7H 1C 9C 3C,8G 6G 0 9C 5C,9G 10C 10C 1      0C 10C 10C 9C 4C,9H 3C,8G 3C,6G 0 10C 3C,7H Morning Glory 9C 9C 4C,8H 1H      10C 9C 1C 0 10C 10C 10C 10C 10C 10C 10C 10C 4C,8H 4C,8H 4C,8H 3C,7H 9C      4C,8H Cocklebur 10C 10C 1H 1H 10C 10C 7H 0 9C 2G 10C 9H 9C 6H 10C 10C      5C,9H 1H 1H 0 1H 0 Nutsedge 3C,8G 2C,9G 4G 9 2C,9G 9G 0 0 5C,9G 5C,9G      5C,9G 4C,9G 9C 5C,9G 9C 2C,9G 5G 0 0 0 3G 0 Crabgrass 4G 0 4G 0 5G 0 0 0      4C,9G 3C,6G 3C,7H 2C,5G 6C,9G 2C,8G 3C,7G 3G 3C,7G 2C,5G 4G 0 4C,9H      2C,8G Barnyard Grass 3C,8H 9C 4C,9H 3C,7H 9C 4C,9H 3C,5H 0 9C 9C 9C 9C      10C 9C 9C 9C 9C 4C,8G 10C 0 9C 9C Wild Oats 3C,8G 2C,5G 2C,9G 4C,9G 4G 0      0 0 6C,9G 5C,9G 9C 3C,8G 5C,9G 4C,9G 4C,9G 2C,6G 3C,6G 2C 3G 9 5C,9G      5C,9G Wheat 9G 2C,9G 7G 3G 5G 0 0 0 9C 9G 9C 3C,9G 9C 4C,9G 2C,9G 6G      4C,9G 2G 3G 0 9G 9G Corn 3C,8H 3G 2C,5H 0 2G 0 0 0 1H 0 3C,7H 1H 3HY,7G      3G 0 0 2C,4H 2H 10C 5H 2C,8H 3H Soybean 9C 4C,9G 3C,6H 2H 9C 9C 3H 0      4C,9G 6C,9G 9C 9C 9C 9C 5C,9G 4C,9G 5C,9G 4C,9G 5C,9G 2C,7G 3C,8H 5H      Rice 2C,8G 4G 4C,9G 4G 2C,9G 7G 2G 0 5C,9G 9C 9C 9C 9C 9C 9C 9C 9C 3C,6G      4C,9G 3G 9C 9C Sorghum 4C,9G 4C,9G 3C,9H 2C,5G 9C 5C,9G 7G 0 10C 9C 10C      9C 10C 9C 9C 9C 9C 4C,9H 4C,9G 2C,3G 9C 4C,9G Cheatgrass 9C 5C,9G 4C,9G      3C,8G 3C,9G 2C,8G 5G 0 5C,9G 2C,9G 9C 4C,9G 9C 4C,9G 3C,9G 6G 2C,8G      2C,5G 4G 9 4C,9G 9G Sugar Beets 9C 5C,9G 3C,7H 4H 4C,9G 3C,7H 2C,5G 0 9C      9C 9C 9C 10C 10C 9C 10C 10C 9C 9C 2C,5G 9C 3C,7H Velvetleaf 10C 10C      2C,2G 0 10C 5C,9G 2C,5G 0 10C 10C 10C 10C 10C 10C 10C 10C 5C,8H 3C,5H      2C,4G 0 9C 4C,8H Giant Foxtail 4C,9G 7G 4C,9G 3C,6G 3C,9G 3C,8G 3C,6G 0      9C 9C 9C 9C 9C 6C,9G 9C 9C 9C 4C,8H 9C 9 9C 9C Barley 2C,9G 3G 4C,9G      2C,5G 3C,9G 2C,5G 2C,5G 0 3C,9G 9G 4C,9G 3C,8G 4C,9G 9G 9G 7G 2G 0 0 0      9C 4C,9G PREEMERGENCE Cotton 8G 2C,4G 0 0 8G 2C,3G 2G 0 3C,8H 2G 4C,9G      2C,5G 5C,9G 9G 2C,8H 5G 3G 0 0 0 3G 0 Morning Glory 9H 5H 2C,3G 9 9G      3C,8H 5G 0 8H 5H 9C 3C,9H 9C 9C 9G 3C,8H 2H 1H 0 0 8H 0 Cocklebur 9H      3C,3H 2H 0 3C,8H 3C,8H 2C,4G 0 0 0 5G 0 6G 3G 7H 3H 2G 1H 0 0 0 0      Nutsedge 10E 5G 0 0 7G 3C,8G 0 0 10E 8G 9G 10E 10E 10E 10E 10E 0 0 0 0 0      0 Crabgrass 4G 0 0 0 5G 0 0 0 4C,8G 2C,8G 4C,7G 3C,6G 4C,9G 3C,6G 2C,6G      3C,6G 0 0 0 0 4C,8G 0 Barnyard Grass 3C,8H 0 2C 0 4C,9H 4C,9H 3G 0 3C,8H      2C,4G 9H 4C,8H 9H 9H 9H 3C,9H 2C,6G 3G 0 0 4C,9H 3G Wild Oats 4C,8H      2C,4G 6G 0 0 2G 0 0 3C,9H 2C,3G 4C,9H 2C 4C,8G 2C,6G 2C,8G 1C 0 0 0 0      2C,8H 2G Wheat 4C,9H 8H 4G 0 8G 2G 0 0 3C,9H 8G 4C,9H 2C,8H 4C,9H 2C,8H      9H 7H 7G 0 0 0 9H 4G Corn 3C,7H 2G 0 0 3C,7G 2C,5G 0 0 0 0 3C,9H 0 4C,9H      4G 2G 0 6H 0 2C,3G 0 4C,9H 0 Soybean 3C,7H 3C,3H 0 0 4C,8H 3C,6H 0 0 8H      7H 9H 7H 9H 9H 9H 3C,8H 2C,6H 2C,2H 2G 0 3G 0 Rice 10E 7G 3C,6G 0 5C,9H      4C,9H 6G 0 10E 9H 10E 9H 10E 10E 10E 10E 8H 2C,5G 0 0 10E 9H Sorghum      4C,9H 3C,7H 3C,6G 0 9H 4C,9H 3G 0 5C,9H 9H 10E 5C,9H 10H 4C,9H 10E 10E      4C,9H 2C,4G 2C,5G 0 10H 9H Cheatgrass 9H 8G 6G 0 3C,9G 8G 0 0 9H 8G 9H      9H 9H 9H 9G 7G 3G 0 0 0 9H 0 Sugar Beets 5C,9G 3C,8G 6H 0 9G 3C,7G 3G 0      5C,9G 8G 5C,9G 8H 5C,9G 9G 4C,9G 9G 6G 0 0 0 0 0 Velvetleaf 8H 3G 2H 0      3C,7G 2H 2G 0 8H 3C,5H 5C,9H 2C,5H 5C,9G 2C,8H 5C,9G 3G 0 0 0 0 2G 0      Giant Foxtail 4C,8H 5G 2C,5G 0 4C,9G 3C,9H 2G 0 4C,9H 2C,5G 4C,9H 3C,8H      9H 4C,9H 9H 2C,6G 2C,5G 0 0 0 9H 3C,8G Barley 3C,9G 2G 2C,8G 0 3C,9G 4G      0 0 9G 2C,7G 3C,9G 4G 9G 9G 9G 2C,8G 7G 0 0 0 2C,9H 2C        CMPD 170 CMPD 171 CMPD 172 CMPD 173 CMPD 174 CMPD 175 CMPD 176 CMPD      177 CMPD 178 CMPD 179 CMPD 180 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01  0.05 0.01      0.05 0.01        POSTEMERGENCE Cotton 9C 4C,9G 5C,9H 4C,9H 0 -- 3C,9G 10C 5C,9G 3G 9C      4C,9G 9C 10C 9C 10C 9C 4C,9H 10C 4C,9H 10C 4C,8H Morningglory 10C 9C      5C,9H 3C,6H 0 -- 0 0 3C,8H 2C,4H 5C,9G 4C,8H 10C 9C 10C 5C,9G 10C 2C,7G      10C 5C,9G 3C,8H 6C,9G Cocklebur 10C 10C 10C 4C,9H 2G -- 8G 2C,6G 4C,9G      2G 10C 4C,8H 10C 10C 10C 10C 10C 9C 10C 10C 9C 5C,9H Nutsedge 10C 4C,9G      8G 3C,7G 3G -- 0 0 0 0 2C,8G 0 9G 9G 9G 3C,9G 8G 2C,4G 9C 3C,9G 5C,9G      2C,9G Crabgrass 4C,8G 2C,6G 2G 0 0 -- 0 0 0 0 3G 0 3C,8G 5G 3C,7G 2G 3G      0 5G 0 6G 4G Barnyardgrass 9C 9C 4G 2H 0 -- 2C,5H 0 7H 3G 9H 5G 9C 4C,9H      5C,9H 3C,9H 9H 3C,7H4C,9H3C,7H 10C 3C,7H Wild Oats 5C,9G 3C,8G 2C,5G 0 0      -- 0 0 0 0 3C,8G 5G 4C,9G 9G 5C,9G 3C,7G 4C,9G 4C,9G3C,5G 2C,3G 3C,8G      2C,7G Wheat 9G 6G 4G 0 0 -- 5G 0 0 0 3G 0 9G 9G 9G 9G 9G 9G 9G 5G 2C,9G      9G Corn 3C,7H 0 0 0 0 -- 0 0 2G 0 0 0 2H 0 1H 0 0 0 1H 0 4U,8G 2C,7G      Soybean 9C 9C 3C,9G 4C,8G 0 -- 0 0 4C,9G 7H 5C,9G 4C,9G 9C 9C 9C 5C,9G      5C,9G 4C,9G 3C,8H 2C,5H 5C,9G 5C,8H Rice 9C 4C,9G 4C,9G 2C,6G 0 -- 0 0      7G 0 9G 4G 9C 9C 9C 5C,9G 4C,9G 4C,9G 4C,9G 4C,9G 5C,9G 6C,8G Sorghum 9C      9C 4C,9H 3C,8G 0 -- 3G 0 2G 0 3C,9G 3C,7G 5C,9G 4C,9G 5C,9G 3C,9G 3C,9G      3C,8G 3C,9G 4C,9H 10C 3U,8G Cheatgrass 9C 3C,9G 2C,8G 8G 0 -- 3G 0 0 0      3G 0 6G 4G 8G 0 0 0 3G 0 5C,9G 4C,8G Sugar Beets 10C 5C,9G 9C 5C,9H 3G      -- 3H 2G 9C 4C,8H 9C 10C 10C 10C 10C 9C 10C 10C 10C 9C 9C 9C Velvetleaf      10C 10C 5C,9H 4C,8H 0 -- 3G 2C,3G 3C,7H 0 4C,9H 3C,6H 10C 10C 10C 6C,9G      10C 4C,9H 10C 4C,9G 9C 6C,9H Giant Foxtail 9C 4C,9G 5G 2H 0 -- 2C,6G 0      2G 0 3C,6G 3G 4C,9G 3C,7G 4C,9G 3C,6G 2C,4G 3G 3C,7H 3C,6G 10C 3C,9G      Barley 3C,8G 7G 2C,4G 0 0 -- 0 0 0 0 6G 0 3C,9G 9G 3C,9G 3C,9G 9G 7G 9G      5G 6C,9G 3C,8G PREEMERGENCE Cotton 4C,8H 3C,8G 2C,6G 0 0 -- 2G 0 3G 0 2G 0       2C,9G 8G 3C,6G 1C 2G 0 9G 2C,6G 2C,6G 0 Morningglory 9H 8H 8H 3C,3H 0      -- 0 0 5H 0 6H 1H 9H 4G 7G 0 2H 0 3C,8G 3C,7H 7H 3G Cocklebur 9H 8H --      2C,2H 0 -- 3G 0 2C,6H 0 2C,5G 0 9H 7H -- 3C,4G 2C,3H 0 9H 8H -- 3C      Nutsedge 10E 8G 0 0 0 -- 0 0 0 0 0 0 9G 5G 8G 3 2C,5G 0 10E10E 7G 0      Crabgrass 3C,7G 0 0 0 0 -- 0 0 0 0 0 0 9G 0 2C 0 0 0 2G 0 0 2G Barnyardgr      ass 9H 6H 3G 0 0 -- 0 0 2H 0 0 0 9G 1H 3H 0 1C 0 8H 7H 0 0 Wild Oats      3C,9G 3G 1C 0 0 -- 0 0 0 0 0 0 3C,7G 2C,5G 3C,5G 0 3C,4G 0 2C,5G 0 2C,4G      0 Wheat 3C,9G 5G 0 0 0 -- 0 0 0 0 0 0 9H 9H 9H 0 6G 0 8H 3G 2C,8H 4G      Corn 3C,8H 2G 1C,2G 0 0 -- 0 0 6G 0 0 0 5G 0 0 0 0 0 0 0 9H 0 Soybean 9H      8H 2C,6G 0 0 -- 0 0 2C,5G 0 3C,6H 1C,1H 9H 3C,6H 3C,7H 2C,4G 2C,5G 0      3C,7H 5G 2C,8H 5G Rice 5C,9H 2C,8G 4G 2G 0 -- 2G 0 8H 0 8G 2G 10E 10H 9H      1C 2C,3G 0 10E 9H 3C,9H 2C Sorghum 5C,9H 9H 3C,9G 3G 0 -- 4G 0 2G 0      2C,8H 2G 4C,9H 9H 9H 3C,5G 3C,7G 0 9H 9H 3C,9H 3C,6G Cheatgrass 5C,9G 8G      5G 0 0 -- 0 0 0 0 0 0 5G 0 4G 0 0 0 0 0 2C,8H 2G Sugar Beets 5C,9G 4C,9G      5C,9G 5G 0 -- 7G 5G 4G 0 7H 2G 9G 9G 9G 7G 4C,9G 3C,6H 9G 9G 4C,8G 3G      Velvetleaf 5C,9G 5G 3C,7H 2C,2G 0 -- 0 0 2G 0 0 0 4C,9G 3H 6G 3C,3H      3C,3H 0 3C,7H 3C,3H 4C,7H 2H Giant Foxtail 5C,9H 4C,8H 3G 0 0 -- 2G 0 0      0 0 0 2C,5G 0 4G 1C 0 0 5G 3G 0 2G Barley 3C,9G 8G 5G 0 0 -- 5G 0 0 0 8G      0 9G 2C,6H 3C,9G 0 2C,8G 0 9G 4G 2C,9H 4G        CMPD 181 CMPD 182 CMPD 183 CMPD 184 CMPD 185 CMPD 186 CMPD 187 CMPD      188 CMPD 189 CMPD 190 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0      .05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01  0.05 0.01 0.05      0.01      POSTEMERGENCE Cotton 10C 9C 10C 10C 10C 4C,8H 4C,8H 3C,7H      3C,8H 2C,8H 2C,8H 3C,8H 2C,7H 2C,6H 9C 5C,9H 10C 5C,9G  3C,9H 8H Morning      Glory 10C 10C 10C 10C 10C 2C,8H 10C 5C,9H 5C,9G 4C,8H 4C,9G 3C,8H 4C,9H      4C,8H 10C 10C 10C 10C 4C,9G 3C,5G Cocklebur 10C 10C 10C 10C 10C 3C,7H      2C,9H 7G 5C,9G 5C,9H 4C,9H 4C,8H 3C,8H 2C,7H 10C 10C 10C 10C 3C,8G 6H      Nutsedge 9C 6C,8G 10C 9C 9C 9G 3G 2G 2C,8G 3G 6G 3C 2C,9G 2C,7G 9C 9C      10C 9C 9G 3C,9G Crabgrass 2C,7G 4G 2C,9G 5G 2C,4G 2G 6G 2G 2G 0 0 0 0 0      2G 0 5G 0 0 0 Barnyardgrass 9C 4C,9G 10C 10C 9C 5C,8G 9C 5C,9G 10C 10C      10C 3C,8H 2C,7G 3G 9C 4C,9H 10C 4C,9H 3C,5G 1H Wild Oats 2C,8G 7G 2C,6G      2G 2C,8G 0 3C,9G 2C,8G 3C,9G 2C,5G 2C,7G 2C,8G 0 0 2C,4G 0 2G 0 0 0      Wheat 9G 8G 2C,9G 7G 2C,9G 3G 3C,9G 2C,8G 9G 2C,6G 9G 9G 0 0 2C,5G 0 8G      0 0 0 Corn 6U,9G 3U,8G 10C 6U,9G6U,9G 3C,7G 4U,9C 2U,9G 5U,9C 2U,9G 10C      4U,9C 3C,7G 3C,3G 9C 5C,9G 9C 4C,9G 2C,5G 1H Soybean 6C,9G 6C,9G 6C,9G      9C 4C,8H 2C,6H 5C,8H 4C,9H 4C,9H 4C,7H 4C,9H 3C,8H 2C,8G 7H 5C,9G 4C,9G      4C,9G 3C,9G 1H 0 Rice 3C,7G 3G 5C,8G 2C,8G 3C,8G 3G 9C 9C 9C 4C,9G 9C      4C,9G 4G 0 7G 0 4C,9G 2G 0 0 Sorghum 6C,9G 3C,8G 6C,9G 5C,9G 6C,9G 2C,8G      10C 5C,9G 9C 3C,9G 5C,9G 4C,9G 2C,8G 2C,6G 9C 3C,9G 5C,9G 9G 9G 3C,6G      Cheatgrass 10C 9C 10C 9C 9C 3C,8G 5C,9G 3C,9G 5C,9G 5C,9G 9C 4C,9G 2C,8G      7G 9C 4C,8G 5C,9G 9C 7G 0 Sugar Beets 10C 10C 10C 9C 6C,9G 5C,9G 2C,7G 0      4C,9G 5C,9H 9C 5C,9G 9C 3C,7H 9C 10C 9C 10C 9C 3C,7G Velvetleaf 10C 10C      10C 10C 10C 6C,9H 5C,9G 4C,8H 4C,9H 3C,8H 4C,8H 3C,5H 4C,8H 4C,7H 10C      10C 10C 9C 3C,8G 0 Giant Foxtail 9C 4C,9G 10C 6C,9G 3C,9G 2C,7G 9C 5C,9G      10C 5C,9G 9C 3C,9G 6G 2G 3C,8G 3G 4C,9G 6G 0 0 Barley 2C,8G 7G 8G 5G 8G      2C,4G 4C,9G 3C,9G 4C,9G 2C,8G 3C,9G 2C,8G 2C,6G 3G 2G 0 7G 0 0 0      PREEMERGENCE Cotton 3C,7G 3G 3C,9G 3C,8G 2C,8G 4G 1C,8G 0 1C,3G 2G 1C,4G 0       0 0 1C 0 9G 9G 2C,7H 3G Morningglory 9G 6G 9H 9C 9H 3C,8H 9G 2C,7G      2C,8H 2C,5G 3C,8H 2G 0 0 2C,2H 0 9G 8G 3H 0 Cocklebur 8H 2G 2C,9H -- 8H      4C,8G 8G 0 3C,7G -- 8H 0 0 0 2C,5G 1C 9H 9H 2C 0 Nutsedge 9G 0 10E 9G      10E 3C,8G 0 0 5G 0 0 0 0 0 0 0 10E 9G 5G 0 Crabgrass 0 3G 2C,4G 6G 2C 0      2C 0 0 0 0 0 0 0 0 0 3G 0 0 0 Barnyardgrass 3C,7G 0 9H 2C,7H 9H 7G 3C,9H      0 2C,4G 0 2C,4G 0 0 0 0 0 3C,9H 5G 7H 0 Wild Oats 2C,6G 0 2C,7G 3G 2C,4G      0 2C,8G 2C 2C,4G 3G 2C,7G 3G 0 0 0 0 3C,4G 0 2G 0 Wheat 2C,8G 7G 2C,8H      7G2C,8H4G 2C,9H 7G 2C,8H 6G 8H 5G 0 0 0 0 5G 0 0 0 Corn 2C,9H 3C,7H 9H      2C,9H 9H 9H 9H 3C,8G 9H 2C,8G 9H 3C,9G 0 0 3C,4G 0 5C,9H 3C,7G 3C,6G 0      Soybean 3C,8H 2C,4G 2C,8H 3C,8H 2,7H 3H 3C,7H 2C,5G 1C,6G 4G 2C,8H 1C,3G      2G 0 5G 2C,2H 9H 6H 3H 0 Rice 2C,7G 0 3C,8H 2C,6G 2C,9H 3C,8H 10E 7G 10E      2C,7G 10H 2C,4G 2C 0 0 2G 8H 0 7G 0 Sorghum 3C,7H 3C,7G 10H 2C,9H 10H      10H 9C 3C,9H 10C 3C,9H 10C 4C,9G 0 0 3C,7G 3C,3G 9G 9H 2C,8G 3C,5G      Cheatgrass 3C,9H 3G 9H 2C,9H 2C,9H 9H 9H 2C,9H 9H 6G 9H 6G 0 0 7G 0 9H      7G 7G 0 Sugar Beets 4C,9G 2C,8G 3C,9G 4C,9G 4C,8G 4C,8H 5G 5G 5G 0 3C,7G      1C,3G 0 0 7H 2H 9H 9G 7H 0 Velvetleaf 4C,8H 7G 4C,9H 2C,8H 4C,8H 2C,4G      3C,7H 0 0 0 4G 0 4G 2H 2C 2G 4C,9G 3G 0 0 Giant Foxtail 3G 3G 2C,9H      3C,9H 2C,7G 2C 2C,8H 0 2C,5G 0 2C,5G 0 0 0 0 0 9G 0 2G 0 Barley 2C,8G      2C,5G 8G 8G 8G 5G 9H 7G 9G 2C,8H 4C,9G 2C,8G 0 0 0 0 3C,9G 2G 0 0        CMPD 191 CMPD 192 CMPD 193 CMPD 194 CMPD 196 CMPD 196 CMPD 197 CMPD      198* CMPD 199 CMPD 200 CMPD 201 Rate kg/ha 0.05 0.01 0.05 0.01 0.05 0.01 0      .05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01  0.05 0.01      0.05 0.01        POSTEMERGENCE Cotton 6H 0 1H 0 7H 3G 4C,8H 2C,4H 4C,9G 2C,9G 0 0 5H 0      0 0 0 0 3C,9G 3C,8H 5C,9G 5C,9G Morningglory 3C,6H 0 8H 5G 4C,9H 3C,7H      4C,9G 4C,8H 9C 3C,8H 1H 0 0 0 0 0 0 0 4C,9G 4C,9G 10C 10C Cocklebur      3C,7H 0 7H 0 5G 2G 4C,9H 3C,5G 5C,5G 4C,9H 2C,3G 0 0 0 0 0 0 0 5C,9G      4C,9G 10C 10C Nutsedge 7G 0 0 0 0 0 2G 0 8G 3C,5G 0 -- 0 0 0 0 0 0 0 0      3C,9G 3C,7G Crabgrass 0 0 0 0 3C,5G 4G 0 0 0 3G 0 0 0 0 0 0 0 0 0 0 0 0      Barnyardgrass 9H 3H 5C,9H 4H 9C 3C,8H 3H 0 5H 3C,5H 0 0 0 0 0 0 0 0 2G 0      3C,9H 6H Wild oats 0 0 0 0 4C,8G 3C,6G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 1C 0      Wheat 0 0 0 0 9G 3C,7G 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 2G 0 Corn 2C,9G      3C,8H 3C,9G 5H 4U,9G 3C,9G 9G 7H 1C 1C 0 0 0 0 0 0 0 0 2G 0 4C,9G 3C,9H      Soybean 3C,7H 0 3C,5H 1H 5C,9G 4C,8G 8H 4H 4C,9G 3C,7H 0 0 0 0 0 0 0 0      3C,8G 3C,4H 4C,8G 3C,8H Rice 6G 5G 5C,9G 7G 9C 9C 7G 4G 3G 2G 4G 0 0 0 0      0 0 0 0 0 3G 0 Sorghum 3C,9H 4G 3C,8H 2G 9C 3C,9G 3C,8H 2G 4C,9G 4C,9H 0      0 0 0 0 0 0 0 3C,6G 3G 9G 4C,9G Cheatgrass 8G 2G 7G 0 5C,9G 9G 5C,9G 5G      2C,8G 8G 0 0 0 0 0 0 0 0 6G 3G 4C,9G 7G Sugar Beets 7H 3G 3C,8H 4H 6G 3H      4C,8G 2C,3G 9C 5C,8H 0 0 0 0 0 0 2G 0 9C 5C,9G 10C 10C Velvetleaf 0 0 1C      0 4C,7H 6G 1C 0 3C,7H 3C,3G 0 0 0 0 0 0 0 0 9C 3C,8H 10C 10C Giant      foxtail 0 0 0 0 5C,9G 3C,7G 1H 0 0 1H 0 0 0 0 0 0 0 0 0 0 3G 0 Barley 0      0 0 0 2G 0 2G 0 0 0 0 0 0 0 0 0 0 0 0 0 2C,2G 0 PREEMERGENCE Cotton 0 0      0 0 1C 0 0 0 3C,5G 0 0 0 0 0 0 0 0 0  2G 0 3C,6G 0 Morningglory 2H 4H 0      0 3H 0 0 0 6H 0 0 0 0 0 0 0 0 0 0 0 3C,8G 2C Cocklebur 0 0 0 0 1C -- 0 0      0 2C 0 0 0 0 0 0 0 0 0 0 3C,6H 2C,6H Nutsedge 0 0 0 0 0 0 0 0 0 0 0 0 0      0 0 0 0 0 0 0 9G 5G Crabgrass 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0      0 Barnyardgrass 0 0 0 0 0 0 0 0 1C 0 0 0 0 0 0 0 0 0 0 0 3C,7H 3C,2G      Wild oats 0 0 0 0 2C,4G 0 0 0 0 0 0 0 0 0 0 0 0 0 2G 0 2G 0 Wheat 0 0 0      0 3C,8G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Corn 2C,6G 0 5G 0 3C,8H 0 0 0      0 0 0 0 0 0 0 0 0 0 0 0 4C,8G 3C,5G Soybean 0 0 0 0 3C,8H 2G 0 0 3C,5G      1C 0 0 0 0 0 0 0 0 0 0 2C,3H 1C,2H Rice 0 0 5G 0 8G 0 0 0 2C,4G 0 0 0 0      0 0 0 0 0 0 0 5G 0 Sorghum 6G 0 3C,3G 0 9H 3C,3G 0 0 3C,7G 3G 0 0 0 0 0      0 0 0 2C,3G 0 4C,9H 3C,6G Cheatgrass 0 0 0 0 6G 0 0 0 7G 3G 0 0 0 0 0 0      0 0 5G 0 8G 3C,5G Sugar Beets 0 0 2H 0 3H 2H 0 0 4C,8G 5G 0 0 0 0 0 0 0      0 3C,8G 0 5C,9G 3C,8G Velvetleaf 0 0 0 0 0 0 0 0 2C 0 0 0 0 0 0 0 0 0 0      0 3C,5H 3C Giant foxtail 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 2G 0      Barley 0 0 0 0 7H 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 2G 0      *It is noted that Compound 198 was inactive at the levels tested. However      it is believed that at higher levels, herbicidal activity would be      present.     CMPD 202 CMPD 203 CMPD 204 CMPD 205 CMPD 206 Rate kg/ha 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE Cotton 9C 10C 9C 9H 3C,8G 3C,5G 4C,9H 4C,9H 9C 4C,9H      Morningglory 10C 10C 4C,9G 3C,8H 5C,9G 3C,8G 4C,9G 3C,8H 10C 9C Cocklebur       10C 10C 5C,9G 3C,8G 5C,9G 3C,8H 4C,9H 3C,8H 10C 4C,9G Nutsedge 9C 10C      2C,8G 8G 0 0 5C 0 Crabgrass 0 0 0 0 0 0 2G 0 Barnyardgrass 3C,9H 6H      1C,2H 0 2C,8H 5H 3C,8H 2C,7H 4C,9G 3C,7H Wild oats 0 0 0 0 2G 0 1C 0 4G      0 Wheat 2G 0 0 0 0 0 0 0 5G 0 Corn 10C 4C,9G 2C,4G 0 3G 0 0 0 4C,9G      3C,7H Soybeans 5C,9G 4C,9G 3H 1H 4C,9G 3C,8G 4C,9G 3C,5G 3C,4H 1C,1H      Rice 7G 2G 0 0 6G 1C 9G 2C,4G Sorghum 4C,9G 4C,9G 3C,8G 2G 3C,7G 1C      3C,9H 3G 3C,7G 5G Cheatgrass 9C 9G 6G 0 8G 5G 5C,9G 7G0 0 Sugar Beets      10C 9C 3C,9H 4C,9G 4C,9G 9C 9C 3C,8H 10C 9C Velvetleaf 10C 10C 5C,9H      3C,8M 4C,8H 3C,6H 3C,8H 3C,5H 10C 4C,8H Giant Foxtail 3G 2G 1C 0 2C,5G 0      3C,4G 0 5C,9G 4C,9G Barley 0 0 0 0 0 0 0 0 0 0 Purple nutsedge      2C,8G -- Large crabgrass         2C,8G 4G Rice dry seeded         7G 3G      PREEMERGENCE Cotton 3C,9G 7H 6G 0 1C 0 2G 0 9G 2C,4G Morningglory 9G 7H      2C,2H 0 0 0 3C,6H 0 7G 6H Cocklebur 8H 7H 2C,2H 0 0 0 2C 6G 3C,6H 6G      Nutsedge 10E 10E 7G 0 0 0 0 0 Crabgrass 0 0 0 0 0 0 0 0 Barnyardgrass      3C,8H 1H 1C 0 3G 0 3C,4G 0 5G 2G Wild oats 3G 0 0 0 0 0 0 0 0 0 Wheat 4G      0 0 0 0 0 0 0 0 0 Corn 3C,9G 3C,8G 2C,3G 0 3C,5G 0 3C,7G 1C 3C,6G 2G      Soybeans 4C,8H 3H 1C 0 1C 0 2C,2H 1H 0 0 Rice 8G 2G 2G 0 6G 0 9H 3G      Sorghum 3C,9H 3C,8H 2C,6G 0 3C,9H 3C,3G 4C,9G 3C,3G 2C,3G 0 Cheatgrass      9G 6G 3G 0 4G 0 8H 0 0 0 Sugar Beets 5C,9G 8G 3C,8G 3H 3C,8H 2H 4C,9G 3H      4C,9G 3C,7G Velvetleaf 3C,8G 3C,3G 2G 0 0 0 1C 0 3C,6H 3C,3H Giant      Foxtail 2G 0 0 0 2G 0 0 0 2C,8G 3G Barley 2C,4G 0 2G 0 0 0 2C,2G 0 0 0      Purple nutsedge         7G -- Large crabgrass         2C 0 Rice dry      seeded         2C,7G 0

TEST B Postmergence

Two round pans (25 cm diameter by 12.5 cm deep) were filled with Sassafras sandy loam soil. One pan was planted with blackgrass, (Alopecurus myosuroides), sugar beets, nutsedge (Cyperus rotundus) tubers, rape (Brassica napus), crabgrass (Digitaria sanguinalis), sicklepod (Cassia obtusifolia), teaweed (Sida spinosa), jimsonweed (Datura stramonium), velvetleaf (Abutilon theorphrasti), and giant foxtail (Setaria faberii). The other pan was planted with wheat, barley, cotton, rice, corn, soybean, wild oats (Avena fatua), cocklebur (Xanthium pennsylvania), morningglory (Ipomoea hederacea), johnsongrass (Sorghum halepense) and barnyard-grass (Echinochloa crusgalli). The plants were grown for approximately fourteen days, the sprayed post-emergence with the chemicals dissolved in a non-phytotoxic solvent.

Preemergence

Two round pans (25 cm diameter by 12.5 cm deep) were filled with Sassafras sandy loam soil. One pan was planted with blackgrass, sugar beets, nutsedge, rape, crabgrass, sicklepod, teaweed, jimsonweed, velvetleaf, and giant foxtail. The other pan was planted with wheat, barley, cotton, rice, corn, soybeans, wild oats, cocklebur, morningglory, johnsongrass, and barnyardgrass. The two pans were sprayed preemergence with the chemicals dissolved in a nonphytotoxic solvent.

Treated plants and controls were maintained in the greenhouse for 28 days, then all treated plants were compared to controls and visually rated for plant response. Response ratings are based on a scale of 0 to 100 where 0=no effect, and 100=complete control. A dash (-) response means no test.

Response ratings are contained in Table B.

    TABLE B        Compound 2 Compound 3 Compound 4 Compound 5 Rate g/ha 62 16 16 4 4 1      .25 62 16 16 16 4 4 4 1 1 .25 .25 62 16 4 1 62 16 4 1        POSTEMERGENCE Corn 100 100 100 100 100 60 40 100 100 100 100 100 90      100 80 70 60 0 100 100 80 40 100 90 60 40 Wheat 100 100 100 60 100 40 0      100 100 30 70 40 0 20 0 0 0 0 100 100 40 0 70 40 0 0 Barley -- -- -- --      -- -- -- -- -- -- -- -- -- -- -- -- --  -- -- -- -- -- -- -- -- -- Rice      100 100 100 90 70 50 30 100 100 80 100 90 60 100 50 30 30 0 100 100 60      30 100 90 30 0 Soybean 100 100 100 100 90 90 60 100 100 100 100 100 90      90 80 70 80 0 100 100 100 60 90 90 60 40 Cotton 100 100 60 70 20 40 0      100 100 100 100 100 80 100 70 40 30 0 100 90 70 30 100 90 60 30 Sugar      beet 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100      0 100 100 100 100 100 100 100 90 Rape 100 100 100 100 100 100 100 100      100 100 100 100 100 100 100 100 100 0 100 100 100 100 100 100 100 100      Crabgrass 100 80 100 50 60 40 0 100 90 50 70 70 30 30 50 0 30 0 100 80      50 30 70 50 40 30 Johnsongrass 100 100 100 100 90 60 40 100 100 100 100      100 70 90 70 30 30 0 100 100 70 30 100 100 80 40 Blackgrass 100 100 100      100 90 50 30 100 100 100 100 100 60 100 80 30 70 0 100 100 60 30 100 100      60 30 Barnyardgrass 100 100 100 100 100 60 40 100 100 100 100 100 70 100      100 30 40 0 100 100 60 30 100 100 80 40 Nutsedge 100 100 100 100 80 90      80 100 100 100 100 100 100 100 100 100 100 0 100 90 50 30 100 100 80 70      Giant Foxtail 100 100 100 90 90 50 30 100 100 80 60 60 30 30 30 0 0 0      100 90 60 30 100 80 30 0 Wild Oats 90 100 80 60 70 40 0 100 100 50 100      40 0 80 0 0 0 0 100 90 30 0 70 40 0 0 Cocklebur 100 100 90 70 60 30 0      100 100 90 100 100 70 90 60 60 30 0 100 90 50 30 100 100 60 30 Morningglo      ry 100 100 90 100 70 90 60 100 100 100 100 100 100 100 100 80 70 0 100      100 80 50 100 90 80 60 Teaweed 100 100 90 70 30 40 0 100 100 60 90 80 30      60 50 0 30 0 100 80 60 40 90 70 50 30 Sicklepod 100 100 100 90 70 60 0      100 100 100 100 100 100 100 90 100 80 0 100 80 60 30 70 60 40 30      Jimsonweed 100 100 100 90 70 70 40 100 100 90 100 90 60 100 70 30 40 0      100 100 70 40 100 90 60 30 Velvetleaf 100 100 100 100 80 80 50 100 100      90 100 100 80 100 90 50 50 0 100 100 100 60 100 100 60 30        Rate g/ha 250 62 62 16 16 4 1 250 62 62 16 16 16 4 4 1 1  250 62 16 4      250 62 16 4        PREEMERGENCE Corn 100 100 100 80 90 20 0 100 100 100 70 70 100 20 40 0 0          100 100 90 60 100 100 90 30 Wheat 100 90 100 80 100 30 0 100 100 100      20 0 40 0 0 0 0  100 100 90 70 100 100 50 0 Barley -- -- -- -- -- -- --      -- -- -- -- -- -- -- -- -- --  -- -- -- -- -- -- -- -- Rice 100 100 100      100 100 90 70 100 100 100 100 100 100 100 100 90 0  100 100 100 100 100      100 100 100 Soybean 100 100 100 80 100 40 20 100 100 100 70 70 90 40 40      0 0  100 100 90 60 100 90 80 60 Cotton 100 80 100 80 80 30 0 100 100 100      70 70 100 30 0 0 0  100 90 60 30 100 80 50 30 Sugar beet 100 100 100 100      100 100 30 100 100 100 100 100 100 100 90 80 0  100 100 100 90 100 100      100 80 Rape 100 100 100 90 100 20 0 100 100 100 90 90 100 90 80 20 0      100 100 100 50 100 100 80 60 Crabgrass 100 100 100 90 90 30 0 100 90 100      60 30 80 30 0 0 0  100 90 50 30 90 70 50 30 Johnsongrass 100 100 100 100      100 90 30 100 100 100 90 70 100 80 30 50 0  100 100 100 70 100 100 100      100 Blackgrass 100 90 100 100 100 70 20 100 100 100 100 90 100 100 70 50      0  100 100 100 90 100 100 100 90 Barnyardgrass 100 100 100 90 100 80 20      100 100 100 80 50 100 30 0 0 0  100 100 100 60 100 100 90 70 Nutsedge      100 100 100 100 100 70 20 100 100 100 100 90 100 90 50 50 0  100 90 80      60 100 100 100 90 Giant Foxtail 100 100 100 90 100 80 50 100 100 100 80      30 100 50 0 0 0  100 100 100 60 100 100 90 60 Wild Oats 100 90 100 90 90      20 0 100 100 100 70 90 80 0 40 0 0  100 90 70 70 90 80 50 30 Cocklebur      100 90 100 80 90 20 0 100 100 100 50 80 80 50 40 20 0  100 100 80 50 100      90 70 50 Morningglory 100 50 100 40 70 0 0 100 100 100 40 80 100 30 40 0      0  100 90 50 30 100 80 70 30 Teaweed 100 100 100 80 90 50 20 100 100 100      80 70 90 70 30 0 0  100 90 70 30 90 70 50 30 Sicklepod 100 90 100 80 80      60 20 100 90 100 90 50 90 80 30 20 0  100 90 60 30 90 70 50 50 Jimsonweed       100 100 100 90 90 60 20 100 100 100 100 80 100 80 30 50 0  100 90 80 50      100 90 60 30 Velvetleaf 100 100 100 100 100 60 0 100 100 100 100 80 100      90 30 60 0  100 100 80 50 100 90 60 30        Compound 8 Compound 13 Compound 14 Compound 16 Compound 20 Compound 21 C      ompound 22 Compound 23 Rate g/ha 62 16 4 1 62 16 4 1 16 4 1 .25 62 16 4      1 62 16 4 62 16 4 62 16 4 62 16 4 1        POSTEMERGENCE Corn 100 80 50 30 100 100 70 40 100 80 60 40 0 0 0 0       100 90 40 100 90 70 100 100 70 50 30 0 0 Wheat 30 0 0 0 30 0 0 0 30 0 0      0 0 0 0 0 90 60 20 0 0 0 70 20 0 40 0 0 0  Barley -- -- -- -- -- -- --      -- -- -- -- -- -- -- -- -- -- -- -- 0 0 0 0 0 0 -- -- -- -- Rice 90 70 0      0 90 30 0 0 60 30 0 0 60 0 0 0 95 90 85 80 20 0 90 50 20 70 40 0 0      Soybean 100 80 70 0 100 100 100 70 100 100 70 60 100 70 40 0 95 90 80      100 90 50 100 100 80 100 100 80 60 Cotton 100 90 60 40 100 100 90 50 100      70 50 30 90 70 50 30 100 100 90 60 0 0 80 70 20 100 100 70 40 Sugar beet      100 100 100 90 100 100 100 100 100 100 90 70 100 100 90 70 95 90 90 90      80 0 100 90 70 100 100 100 100 Rape 100 100 100 90 100 100 100 100      100100 90 60 100 100 90 60 100 100 100 100 90 30 100 100 70 100 100 100      100 Crabgrass 90 50 30 0 90 60 50 30 30 0 0 0 30 0 0 0 60 30 20 40 0 0      60 30 0 60 40 30 0 Johnsongrass 90 50 0 0 100 90 60 30 100 80 60 30 90      70 30 0 100 100 85 100 70 20 100 100 70 100 100 80 60 Blackgrass 100 90      30 0 100 70 40 0 70 30 0 0 70 30 0 0 100 95 85 80 60 0 100 70 50 100 70      30 0 Barnyardgrass 90 50 0 0 100 90 60 30 100 80 50 30 90 50 0 0 100 95      80 100 70 30 100 100 50 100 100 80 60 Nutsedge 100 70 70 40 100 100 90      80 90 70 50 30 90 70 60 40 100 80 60 0 0 0 0 0 0 100 100 70 50 Giant      Foxtail 90 50 0 0 100 80 30 0 70 30 0 0 0 0 0 0 90 85 60 100 60 20 100      100 50 70 50 30 0 Wild Oats 30 0 0 0 60 30 0 0 40 0 0 0 0 0 0 0 85 70 30      0 0 0 60 20 0 40 0 0 0 Cocklebur 100 90 50 30 100 70 50 30 100 90 60 30      90 80 50 30 100 95 85 60 0 0 100 60 20 100 100 100 100 Morningglory 100      90 60 30 100 100 100 50 90 70 50 30 90 80 60 30 100 100 90 50 0 50 70 60      20 100 80 60 30 Teaweed 100 70 30 30 100 90 60 40 90 50 30 0 70 30 30 0      90 95 90 40 20 0 70 50 20 90 70 50 30 Sicklepod 90 50 30 0 100 100 80 40      80 50 0 0 50 30 0 0 70 25 30 50 0 0 80 50 20 100 70 50 30 Jimsonweed 100      100 60 30 100 100 60 30 90 90 50 30 100 80 50 30 95 90 30 80 70 20 90 70      50 100 100 70 50 Velvetleaf 100 100 70 50 100 100 100 70 100 90 50 30      100 80 30 0 100 100 90 30 0 0 70 30 20 100 100 100 90 Green Foxtail                    70 20 0 100 80 50 Cheatgrass                    0 0 0 0 0      0 Wild Buckwheat                    100 80 0 80 80 50 Viola            40 20 0 80 -- 20 Lambsquarter                    90 50 0 80 60      50    Rate g/ha 250 62 16 4 250 62 16 4 62 16 4 1 250 62 16 4 250 62 16      250 62 16 250 62 16 250 62 16 4        PREEMERGENCE Corn 100 90 30 0 100  90 90 20 90 70 50 30 80 50 30 0 100 9      5 90 90 60 20 90 80 0 70 50 30 0 Wheat 80 30 0 0 30 0 0 0 80 40 0 0 90      40 0 0 95 95 80 40 0 0 50 0 0 80 60 40 0 Barley -- -- -- -- -- -- -- --      -- -- -- -- -- -- -- -- -- -- -- 0 0 0 60 20 0 -- -- -- -- Rice 100 100      100 20 100 100 100 70 100 100 70 40 100 100 90 60 100 100 100 -- -- --      -- -- -- 100 100 80 50 Soybean 100 80 40 0 100 100 90 70 100 90 70 60      100 80 60 30 95 95 85 80 80 30 90 80 30 100 80 60 40 Cotton 100 60 20 0      100 80 80 20 80 70 50 30 90 70 50 30 95 90 80 90 20 0 90 80 20 90 70 40      0 Sugar beet 100 100 100 50 100 100 100 90 100 100 100 80 100 100 100      100 10095 90 90 70 50 80 70 80 100 100 100 80 Rape 100 100 90 40 100 100      90 90 100 100 60 60 100 90 60 0 100 95 80 80 60 0 90 80 70 100 90 70 50      Crabgrass 80 70 40 20 90 70 50 0 90 70 50 30 90 70 50 40 90 30 10 90 0 0      70 70 20 90 70 50 30 Johnsongrass 100 90 60 20 100 100 100 60 100 80 50      30 100 80 50 30 95 95 90 100 80 0 100 90 80 100 90 80 60 Blackgrass 100      90 70 30 100 90 80 50 100 90 60 30 100 90 60 30 100 95 80 100 50 0 90 70      70 100 100 80 50 Barnyardgrass 100 90 20 0 100 100 90 60 100 70 50 0 100      80 40 0 100 95 90 100 50 0 100 90 50 100 80 60 40 Nutsedge 100 100 80 60      100 100 100 90 100 100 90 80 100 100 100 90 100 100 100 0 0 0 0 0 0 100      100 80 60 Giant Foxtail 100 90 -- 0 100 90 70 50 100 60 40 0 80 60 30 0      100 95 90 90 70 0 100 90 70 100 100 90 70 Wild Oats 100 90 80 0 -- -- --      -- 80 40 0 0 90 40 0 0 90 85 65 60 20 0 50 50 20 70 50 30 0 Cocklebur      100 80 20 0 100 70 80 20 10090 70 50 100 80 70 30 95 90 90 30 20 0 -- 30      0 90 80 70 50 Morningglory 100 60 20 0 100 90 80 30 90 70 50 30 100 80      50 30 95 90 80 70 20 0 80 60 20 70 50 30 0 Teaweed 100 90 90 20 100 90      90 20 90 80 50 30 90 80 50 30 90 80 50 80 30 0 70 40 0 90 70 50 --      Sicklepod 100 90 30 0 100 100 80 20 90 70 50 30 90 70 50 30 90 50 10 50      0 0 70 30 0 90 70 40 0 Jimsonweed 100 100 80 30 100 100 90 50 90 70 50      30 90 70 50 30 100 90 60 60 0 0 70 30 0 100 80 60 40 Velvetleaf 100 100      60 20 100 100 90 80 90 70 50 30 90 70 50 30 100 95 70 30 0 0 60 30 0 100      80 60 40 Green Foxtail                    90 90 30 100 90 50 Cheatgrass                        50 0 0 60 0 0 Wild Buckwheat                    100 50      50 90 60 20 Viola                    100 -- 20 90 50 30 Lambsquarter                     90 70 0 90 60 0        Compound 24 Compound 27 Compound 28 Compound 31 Compound 32 Compound      33 Compound 34 Rate g/ha 62 16 4 1 250 62 16 4 250 62 16  62 16 4 1 62      16 4 1 62 16 4  62 16 4 1        POSTEMERGENCE Corn 0 0 0 0 0 0 0 0 0 0 0  100 70 50  30 80 40 0 0 80      40 30  70 30 0 0 Wheat 30 0 0 0 40 20 0 0 30 0 0  0 0 0 0 80 60 40 20 90      70 30  60 30 0 0 Barley -- -- -- -- -- -- -- --     -- -- -- -- -- -- --      -- -- -- --  -- -- -- -- Rice 30 0 0 0 90 70 50 30 50 30 0  70 30 0 0      100 70 50 30 80 70 30  90 70 50 30 Soybean 100 100 80 60 90 80 70 50 80      60 40  100 90 70 40 100 100 90 70 90 90 70  90 90 80 60 Cotton 100 90 70      40 100 90 60 30 100 70 30  80 60 30 0 100 100 100 80 90 90 50  90 80 50      30 Sugar beet 100 100 100 90 100 100 100 100 100 100 100  100 100 60 30      100 100 70 50 100 100 80  100 100 70 50 Rape 100 100 100 100 100 100 100      100 100 100 100  100 100 100 100 100 100 100 100 100 100 100  100 100      100 100 Crabgrass 30 0 0 0 70 50 30 0 50 30 0  90 70 50 30 90 70 50 30      60 30 0  80 50 30 0 Johnsongrass 100 70 50 30 100 90 70 50 90 70 50  100      100 60 30 100 100 100 80 100 100 60  100 90 70 30 Blackgrass 100 100 70      40 90 60 30 0 100 90 70  100 100 60 30 100 100 90 70 90 70 30  100 70 30      0 Barnyardgrass 80 60 30 0 100 90 70 50 90 60 30  100 100 70 30 100 100      100 90 100 70 50  100 70 50 0 Nutsedge 100 90 70 50 100 100 70 50 70 50      30  30 0 0 0 100 100 100 90 100 60 50  90 70 50 30 Giant Foxtail 70 30 0      0 70 50 30 0 80 60 30  100 100 70 40 100 90 70 50 90 70 50  90 70 60 0      Wild Oats 30 0 0 0 60 40 20 0 30 0 0  70 40 20 0 80 60 40 20 80 40 30      70 50 30 0 Cocklebur 100 100 100 90 100 90 70 50 90 70 50  90 70 50 30      100 100 100 70 100 80 60  90 70 30 0 Morningglory 100 90 70 50 90 80 70      50 100 100 70  90 70 50 30 100 100 90 70 100 100 50  90 80 60 40 Teaweed      70 50 30 0 80 60 40 20 80 60 40  80 60 30 0 100 80 60 30 80 50 30  80 50      30 0 Sicklepod 70 50 30 0 80 60 30 0 50 30 0  80 60 30 0 100 100 90 80      90 50 30  90 50 30 0 Jimsonweed 100 70 50 30 100 70 50 30 100 80 60  100      80 60 40 100 90 80 70 90 80 60  100 80 70 50 Velvetleaf 100 100 70 50      100 100 80 50 100 80 50  100 80 60 40 100 100 100 90 100 100 90  100 100      80 60 Green Foxtail Cheatgrass Wild Buckwheat Viola Lambsquarter        Rate g/ha 250 62 16 4 250 62 16 4 250 62 16 4 250 62 16 4 250 62 16 4      250 62 16 4 250 62 16 4        PREEMERGENCE Corn 30 0 0 0 0 0 0 0 0 0 0 0 90 60 0 0 90 80 70  40 40 0 0       0 60 0 0 0 Wheat 70 30 0 0 70 50 30 0 70 30 0 0 60 30 0 0 80 60 40 20      90 40 0 0 70 30 0 0 Barley -- -- -- -- -- -- -- -- 70 30 0 0 -- -- -- --      -- -- -- -- --  -- -- -- -- -- -- -- Rice 90 70 50 30 100 90 70 50 100      90 60 30 100 100 90 70 100 100 100 100 100100 30 0 100 100 40 0 Soybean      90 70 50 30 70 50 30 0 90 60 30 0 90 70 50 30 100 80 60 40 90 60 30 0 90      50 0 0 Cotton 70 50 30 0 50 30 0 0 70 30 0 0 80 40 0 0 90 70 50 30 80 60      30 0 60 30 0 0 Sugar beet 100 100 90 80 100 90 70 50 90 70 50 30 100 90      70 50 100 100 90 70 100 80 40 0 100 90 70 50 Rape 100 90 70 50 90 70 50      30 90 70 50 30 90 70 50 20 100 90 70 50 90 70 50 30 90 70 40 0 Crabgrass      90 60 30 0 80 70 60 30 70 50 30 0 90 60 30 0 90 80 70 60 70 50 30 0 70      50 40 30 Johnsongrass 90 80 70 50 90 80 70 40 100 90 70 50 100 80 60 40      100 100 90 70 100 90 70 50 90 70 40 0 Blackgrass 90 80 70 40 90 70 50 30      90 70 50 30 100 90 70 50 90 80 70 50 90 70 30 0 100 80 40 0 Barnyardgrass       90 80 60 30 90 60 30 0 90 70 50 30 90 80 60 30 100 90 70 40 100 70 30 0      90 40 0 0 Nutsedge 100 80 60 40 90 70 50 30 100 70 50 30 80 60 40 20 100      90 80 70 90 70 50 30 90 70 50 30 Giant Foxtail 100 90 70 40 90 60 40 0      90 70 50 30 100 80 60 30 100 100 80 60 100 80 50 30 90 50 0 0 Wild Oats      70 40 30 0 80 60 30 0 30 0 0 0 60 30 0 0 90 70 50 30 80 30 0 0 70 30 0 0      Cocklebur 90 70 50 30 80 60 40 0 90 70 50 30 90 70 50 30 90 70 50 30 90      60 30 0 90 50 30 0 Morningglory 80 60 40 20 30 0 0 0 90 60 30 0 80 60 40      20 100 90 60 30 90 60 30 0 80 50 30 0 Teaweed 90 70 50 30 90 70 50 30       70 50 30 0 100 80 60 40 60 30 0 0 80 50 30 0 Sicklepod 90 70 40 0 90 70      40 0 40 0 0 0 80 60 40 0 100 80 40 0 90 60 30 0 70 30 0 0 Jimsonweed 90      70 50 30 90 70 50 30 90 70 50 30 90 70 50 30 90 80 70 50 90 70 50 30 90      70 50 30 Velvetleaf 90 70 50 30 90 70 50 30 90 70 50 30 90 70 50 30 90      80 70 50 80 60 40 20 80 70 50 30 Green Foxtail         90 70 50 30      Cheatgrass         60 30 0 0 Wild Buckwheat         90 70 50 30 Viola           90 70 50 30 Lambsquarter         100 70 50 30        Compound 35 Compound 36 Compound 39 Compound 40 Compound 46 Compound      53 Compound 54 Rate g/ha 62 16 4 1 62 16 4 1 62 16 4 1 62 16 4 1  62 16      4 1 62 16 4 1 62 16 4 1        POSTEMERGENCE Corn 30 0 0 0 90 70 30 0 100 100 70 30 80 20 0 0  100 80 5      0 0 0 0 0 0 0 0 0 0 Wheat 40 0 0 0 80 50 30 0 100 100 80 50 90 80 20 0      80 70 20 0 60 30 0 0 80 60 40 20 Barley -- -- -- -- -- -- -- -- 100 80      40 0 20 0 0 0 90 80 50 0 60 30 0 0 60 30 0 0 Rice 100 70 30 0 90 70 50      30 100 100 80 30 90 60 30 0 100 100 70 20 90 60 30 0 90 60 30 0 Soybean      90 80 60 50 100 80 60 40 100 100 90 70 100 80 80 50 100 90 80 60 100 90      80 70 100 90 70 50 Cotton 100 80 40 0 90 70 40 0 70 30 30 0 70 60 30 0      100 60 50 0 90 60 20 0 90 70 20 0 Sugar beet 100 100 100 70 100 100 100      70 100 90 40 20 70 50 0 0 100 100 60 20 100 100 100 90 100 100 90 70      Rape 100 100 100 100 0 0 0 0 100 100 100 80 100 100 70 50 100 100 90 50      100 100 100 100 100 100 100 90 Crabgrass 60 30 0 0 90 60 30 0 90 50 20 0      40 0 0 0 60 30 0 0 70 50 30 0 60 30 0 0 Johnsongrass 100 100 70 40 100      90 60 30 100 100 70 50 80 50 20 0 90 100 80 20 100 90 70 50 100 90 70 50      Blackgrass 100 80 30 0 100 100 70 30 90 100 70 60 80 50 20 0 100 90 60 0      100 90 60 30 100 90 70 50 Barnyardgrass 100 100 70 30 100 90 70 30 100      100 90 60 90 60 20 0 100 100 80 20 100 100 90 60 100 90 70 50 Nutsedge      90 70 50 30 0 0 0 0 70 80 30 0 50 0 0 0 30 -- -- 0 -- -- -- -- -- -- --      -- Giant Foxtail 90 80 50 30 90 70 50 30 90 40 20 0 60 30 0 0 100 80 40      0 100 90 70 50 90 70 50 30 Wild Oats 50 0 0 0 90 60 30 0 100 100 90 40      100 40 0 0 90 90 30 0 30 0 0 0 30 0 0 0 Cocklebur 100 90 50 30 30 0 0 0      100 100 100 30 100 90 80 0 100 70 20 0 100 90 70 50 100 90 70 50      Morningglory 100 90 50 30 100 90 70 50 100 100 90 30 100 100 70 30 100      100 80 60 100 100 90 60 100 70 50 30 Teaweed 90 60 30 0 70 50 30 0 90 50      20 0 60 50 30 0 80 60 40 0 90 70 50 30 90 70 50 30 Sicklepod 90 40 0 0      90 60 30 0 100 100 50 0 100 30 30 20 100 90 70 0 100 100 70 50 100 70 50      30 Jimsonweed 100 80 50 30 80 60 40 0 100 100 70 50 90 70 50 0 100 90 80      20 100 90 70 50 100 90 70 50 Velvetleaf 100 100 70 30 80 60 40 0 100 90      60 20 100 80 60 0 100 90 60 20 100 100 80 60 100 90 70 50 Green Foxtail             100 70 50 0 60 30 20 0 100 80 60 0 90 70 50 30 90 70 50 30      Cheatgrass         100 100 60 50 80 70 50 0 40 20 0 0 100 90 70 50 100      70 50 30 Wild Buckwheat         100 90 70 0 70 0 0 0 100 100 80 0 100 90      70 50 90 70 50 30 Viola         70 80 80 30 80 -- -- -- 90 70 30 30 100      90 70 50 90 70 50 30 Lambsquarter         100 90 50 20 90 70 20 0 100      100 80 50 100 90 70 50 100 90 70 50        Rate g/ha 250 62 16 4 250 62 16 4 250 62 16 4 250 62 16 4 250 62 16 4      250 62 16 4 250 62 16 4        PREEMERGENCE Corn 30 0 0 0 70 30 0 0 100 80 70 20 80 20 0 0  90 80 0 0 0       0 0 0 0 0 0 0 Wheat 80 60 30 0 60 30 0 0 90 70 60 0 80 60 0 0 90 70 40      20 70 40 20 0 80 50 30 0 Barley -- -- -- -- -- -- -- -- 90 80 20 0 0 0 0      0 90 90 50 0 60 40 20 0 50 30 0 0 Rice 100 100 100 70 100 100 100 90 100      100 90 60 100 80 50 0 100 100 90 80 90 80 70 30 90 70 50 30 Soybean 90      80 70 30 80 40 0 0 100 100 60 60 100 50 30 0 90 80 40 0 90 80 60 30 80      60 30 0 Cotton 90 70 50 30 40 0 0 0 80 70 20 0 30 0 0 0 90 70 40 0 60 50      30 0 80 40 0 0 Sugar beet 100 100 90 70 100 90 70 50 100 100 60 20 90 80      60 0 100 90 70 50 100 90 80 70 100 90 80 70 Rape 100 90 60 30 80 60 40 0      100 100 90 20 100 90 40 0 100 100 80 50 100 90 70 50 90 80 70 50      Crabgrass 80 60 50 30 100 70 50 30 100 90 70 20 100 80 20 0 90 50 30 0      90 70 50 30 70 50 30 0 Johnsongrass 100 100 90 70 100 90 70 40 100 100      90 80 100 100 90 80 100 70 50 30 90 80 70 30 90 70 50 30 Blackgrass 100      100 90 50 100 100 80 60 100 90 90 50 100 90 70 50 90 90 50 30 100 70 50      30 90 80 70 50 Barnyardgrass 100 90 80 50 100 80 40 0 100 90 70 30 100      90 80 0 90 70 40 0 90 80 70 30 90 80 70 40 Nutsedge 100 100 70 50 70 50      30 0 100 --  -- -- -- -- 0 -- 90 70 50 30 90 80 70 50 100 90 70 50 Giant      Foxtail 100 90 80 50 100 90 70 40 100 90 70 30 100 90 70 0 90 80 50 30      90 80 70 30 90 80 70 40 Wild Oats 80 60 30 0 70 40 0 0 90 90 60 20 90 30      0 0 70 60 30 0 40 20 0 0 40 0 0 0 Cocklebur 90 80 50 40 -- 0 0 0 100 80      70 0 90 -- -- -- 40 0 0 0 90 70 50 30 90 70 50 30 Morningglory 90 80 60      30 80 60 30 0 100 90 40 0 90 70 20 0 90 80 70 50 90 80 70 60 90 80 70 50      Teaweed 90 70 40 0 90 70 50 20 100 90 60 30 90 90 50 0 90 70 50 30 90 70      50 30 90 70 50 30 Sicklepod 50 30 0 0 90 70 50 30 100 80 30 0 80 0 0 0      50 30 0 0 90 80 70 60 90 70 50 30 Jimsonweed 100 80 50 30 90 70 40 20      100 90 70 50 100 40 20 0 90 70 50 30 90 80 70 50 100 70 50 30 Velvetleaf      90 80 50 30 90 70 50 20 100 90 50 20 90 30 0 0 90 70 50 30 90 70 50 30      90 70 50 30 Green Foxtail         100 90 80 70 100 100 40 0 90 80 50 30      90 70 50 30 90 80 70 50 Cheatgrass         100 100 90 70 100 90 70 60 90      80 30 20 90 80 70 30 90 80 70 50 Wild Buckwheat         100 90 80 70 100      70 60 20 100 80 60 30 90 80 70 50 90 80 70 50 Viola         100 100 90      20 90 80 20 0 100 100 100 90 100 90 70 50 100 100 90 70 Lambsquarter          100 100 90 60 100 100 80 70 100 100 70 50 90 70 50 30 90 80 70      50      Compound 55 Compound 56 Compound 206 Rate g/ha 62 16 4 1 62 16 4 1       62 16 4 1        POSTEMERGENCE Corn 0 0 0 0 0 0 0 0 60 30 0 0 Wheat 90 60 30 0 40 20 0      0 30 0 0 0 Barley 70 40 0 0 20 0 0 0 0 0 0 0 Rice 90 60 30 0 80 60 30 0         Soybean 90 80 70 50 70 30 0 0 30 0 0 0 Cotton 90 60 0 0 40 0 0 0 80      70 60 30 Sugar beet 100 100 90 70 100 90 70 50 100 100 90 70 Rape 100      100 100 80 100 100 90 80 100 100 90 70 Crabgrass 80 60 40 20 50 30 0 0        Johnsongrass 100 90 70 50 90 70 50 30 50 30 0 0 Blackgrass 100 90 70      50 90 70 50 30 70 50 30 0 Barnyardgrass 100 100 70 50 90 70 50 30 100 60      30 0 Nutsedge -- -- -- -- -- -- -- --     Giant Foxtail 90 80 70 30 90      60 30 0 50 30 0 0 Wild Oats 70 30 0 0 0 0 0 0 0 0 0 0 Cocklebur 100 90      70 50 90 70 50 30 90 60 30 0 Morningglory 100 80 60 30 100 60 30 0      Teaweed 90 70 50 30 90 70 50 30     Sicklepod 100 70 50 30 70 50 30 0 70      50 30 0 Jimsonweed 90 80 60 30 90 70 50 30 100 70 50 30 Velvetleaf 100      90 70 40 100 70 50 30 100 100 90 70 Green Foxtail 90 70 50 30 90 70 50      30 80 50 30 0 Cheatgrass 100 90 70 50 90 70 50 30 0 0 0 0 Wild Buckwheat      100 90 80 60 90 70 50 30 70 50 30 0 Viola 100 90 70 50 -- 70 50 30      Lambsquarter 100 90 70 50 90 70 50 30 100 90 70 50 Large crabgrass        50 30 0 0 Prikley sida         80 70 50 30 Rice dry seeded         70      50 30 0 Ivy morningglory         90 80 70 50 Purple nutsedge         70      30 0 0 Chickweed spp.         100 90 60 30        Rate g/ha 250 62 16 4 250 62 16 4 250 62 16 4        PREEMERGENCE Corn 0 0 0 0 0 0 0 0 100 30 0 0 Wheat 80 40 0 0 80 40 0 0      0 0 0 0 Barley 80 30 0 0 0 0 0 0 0 0 0 -- Rice 100 70 50 30 90 80 70 40         Soybean 90 70 30 0 80 60 30 0 0 0 0 0 Cotton 90 60 30 0 70 0 0 0 30 0      0 0 Sugar beet 100 90 80 70 100 90 80 70 90 70 50 -- Rape 90 80 70 40      100 90 80 70 90 90 60 -- Crabgrass 70 50 30 0 70 50 30 0     Johnsongrass       90 80 70 50 100 90 80 6080 50 30 0 Blackgrass 100 100 90 80 90 80 70 50      60 30 0 -- Barnyardgrass 90 80 70 40 100 80 70 50 70 30 0 0 Nutsedge 90      80 70 50 90 80 70 50     Giant Foxtail 90 80 60 30 90 80 70 40 80 70 50      30 Wild Oats 50 30 0 0 30 0 0 0 0 0 0 -- Cocklebur 100 70 50 30 100 70      50 30 40 20 0 0 Morningglory 100 90 60 30 90 70 50 30     Teaweed 90 70      50 30 90 70 50 30     Sicklepod 90 70 50 30 100 70 50 3030 20 0 0      Jimsonweed 90 70 50 30 90 70 50 30 70 50 30 0 Velvetleaf 90 70 50 30 90      70 60 50 90 70 50 -- Green Foxtail 90 80 70 50 90 80 70 50 100 50 30 0      Cheatgrass 90 80 70 40 90 80 70 50 0 0 0 -- Wild Buckwheat 90 80 70 50      90 70 60 40 80 50 30 -- Viola 100 100 90 70 100 100 90 80     Lambsquarte      r 90 70 50 30 90 70 50 30 90 70 50 30 Large crabgrass         60 30 0 0      Prikley sida         70 50 30 20 Rice dry seeded         80 60 40 20 Ivy      morningglory         80 50 30 0 Purple nutsedge         30 0 0 0      Chickweed spp.         60 30 0 --

TEST C

The Corn and Sorghum Herbicide Test included the following species in both the preemergence and postemergence evaluations:

    ______________________________________                                                  SPECIES                                                               Category   Common Name  Scientific Name                                        ______________________________________                                         Crops      Corn         Zea mays                                                          Soybean      Glycine max                                                       Sorghum      Sorghum bicolor                                        Grasses    Green foxtail                                                                               Setaria viridis                                                   Giant foxtail                                                                               Setaria faberii                                                   Johnsongrass Sorghum halepense                                                 Barnyardgrass                                                                               Echinochloa crus-galli                                            Fall panicum Panicum dichotomiflorum                                           Crabgrass    Digitaria sanguinalis                                             Nutsedge     Cyperus rotundus                                       Broadleaves                                                                               Cocklebur    Xanthium pensylvanicum                                            Morningglory Ipomoea hederacea                                                 Velvetleaf   Abutilon theophrasti                                              Jimsonweed   Datura stramonium                                                 Lambsquarters                                                                               Chenopodium album                                                 Pigweed      Amaranthus retroflexus                                            Smartweed    Polygonum persicaris                                   ______________________________________                                    

Postemergence

Postemergence plants were grown in Sassafras sandy loam soil. Corn and soybeans were grown in separate 25 cm diameter containers. Sorghum and the seven grass weed species were grown in two 18 cm diameter containers, 4 species per container. The seven broadleaf weed species were also grown in two 18 cm diameter containers, 4 species in one container, 3 species in the second container. One additional planting of corn in an 18 cm diameter container was made. The soil surface of this additional container of corn was covered with the absorbent, perlite, before spray treatment so that test chemicals would enter the plant only via the foliage. The plants were grown 10-21 days, dependent upon the species and then sprayed postemergence with the test chemicals dissolved in a non-phytotoxic solvent.

PREEMERGENCE

Preemergence plantings were grown in fertilized Tama slit loam soil. These plants are identical to those described in the postemergence section, with the exception of the corn planting having perlite covering the soil surface. These plantings were made the day of or the day before the spraying the test chemicals dissolved in a non-phytotoxic solvent.

EVALUATION

Treated plants and controls were maintained in the greenhouse for 2 to 4 weeks. Visual planting response ratings were made on a percentage scale of 0 to 100 in comparison with a control where 0=no injury, and 100=death.

    TABLE C       Compound 35 Compound 53 Compound 163 Compound 165 RATE RATE GM 0004      0008 0016 0031 0062 0125 0250 0004 0008 0016 0031 0062 0125 0250 0004      0008 0016 0031 0062 0125 0250 0004 0008 0016        POSTEMERGENCE CORN 0 0 0 0 25 45 -- 0 0 0 0 25 45 -- 0 0 0 20 55 65 -- 0       20 45 SOYBEAN 45 70 85 100 100 100 -- 100 100 100 100 100 100 -- 100      100 100 100 100 100 -- 100 100 100 GREEN FXTL 45 55 70 85 95 100 -- 30      40 55 75 85 95 -- 60 80 90 100 100 100 -- 25 70 75 GIANT FXTL 40 45 60      75 95 100 -- 35 50 75 90 100 100 -- 60 80 95 100 100 100 -- 40 90 95      PANICUM 90 100 100 100 100 100 -- 80 100 100 100 100 100 -- 90 100 100      100 100 100 -- 100 100 100 CRABGRASS 0 0 0 30 45 55 -- 0 0 0 30 45 60 --      0 25 40 85 100 100 -- 20 40 60 BARNYARDGRASS 85 95 100 100 100 100 -- 75      100 100 100 100 100 -- 80 100 100 100 100 100 -- 100 100 100 JOHNSONGRASS       100 100 100 100 100 100 -- 95 100 100 100 100 100 -- 100 100 100 100      100 100 -- 100 100 100 SORGHUM 100 100 100 100 100 100 -- 95 100 100 100      100 100 -- 100 100 100 100 100 100 -- 100 100 100 NUTSEDGE 30 50 85 90      100 100 -- 70 95 100 100 100 100 -- 60 75 90 100 100 100 -- 100 100 100      VELVETLEAF 25 55 75 90 100 100 -- 65 95 100 100 100 100 -- 100 100 100      100 100 100 -- 90 100 100 COCKLEBUR 100 100 100 100 100 100 -- 75 90 100      100 100 100 -- 0 30 60 80 100 100 -- 25 50 80 SMARTWEED 60 80 85 90 100      100 -- 55 75 90 100 100 100 -- 60 80 100 100 100 100 -- 65 80 90      LAMBSQUARTER 0 30 60 75 85 100 -- 25 50 70 90 95 100 -- 65 80 100 100      100 100 -- 40 70 85 PIGWEED 50 85 100 100 100 100 -- 70 95 100 100 100      100 -- 65 95 100 100 100 100 -- 95 100 100 MORNINGGLORY 60 75 95 100 100      100 -- 60 80 90 100 100 100 -- 85 95 100 100 100 100 -- 80 95 100      JIMSONWEED 65 100 100 100 100 100 -- 70 95 100 100 100 100 -- 90 100 100      100 100 100 -- 80 95 100 PREEMERGENCE CORN -- -- 0 0 0 0 35 -- -- 0 0 0      20 40 -- -- 0 0 0 0 20 -- 0 0 SOYBEAN -- -- 0 20 30 45 65 -- --  0 35 60      80 100 -- -- 20 30 40 60 80 -- 20 35 GREEN FXTL -- -- 55 85 95 95 100 --      -- 35 50 70 90 95 -- -- 25 60 75 100 100 -- 20 50 GIANT FXTL -- -- 55 85      95 100 100 -- -- 35 50 65 85 95 -- -- 20 40 70 100 100 -- 30 70 PANICUM      -- -- 80 100 100 100 100 -- -- 65 85 100 100 100 -- -- 30 70 95 100 100      -- 50 85 CRABGRASS -- -- 0 20 25 60 70 -- -- 0 0 0 30 40 -- -- 0 25 55      70 100 -- 0 30 BARNYARDGRASS -- -- 85 100 100 100 100 -- -- 30 70 85 100      100 -- -- 0 35 65 100 100 -- 0 20 JOHNSONGRASS -- -- 100 100 100 100 100      -- -- 70 100 100 100 100 -- -- 40 95 100 100 100 -- 40 85 SORGHUM -- --      100 100 100 100 100 -- -- 80 100 100 100 100 -- -- 70 95 100 100 100 --      40 75 NUTSEDGE -- -- 60 95 100 100 100 -- -- 70 85 100 100 -- -- -- 60      80 95 100 100 -- 30 60 VELVETLEAF -- -- 0 0 0 35 60 -- -- 0 0 30 45 --      -- -- 0 0 25 45 80 -- 0 0 COCKLEBUR -- -- 0 0 0 30 65 -- -- 0 0 0 0 --      -- -- 0 0 30 55 70 -- 0 0 SMARTWEED -- -- 0 0 30 80 100 -- -- 30 60 80      100 -- -- -- 0 35 60 85 100 -- 25 50 LAMBSQUARTER -- -- 0 50 80 100 100      -- -- 25 60 85 100 -- -- --  20 60 95 100 100 -- 20 55 PIGWEED -- -- 0      35 70 95 100 -- -- 0 40 75 95 -- -- -- 30 70 100 100 100 -- 30 65      MORNINGGLORY -- -- 0 0 0 30 55 -- -- 0 0 25 35 -- -- -- 0 0 20 35 70 --      0 0 JIMSONWEED -- -- 0 35 45 70 100 -- -- 0 30 55 80 -- -- -- 0 30 70 90      100 -- 0 0        Compound 165 Compound 166 RATE RATE GM 0031 0062 0125 0250 0004 0008      0016 0031 0062 0125 0250        POSTEMERGENCE CORN 85 100 -- -- 0 0 0 0 0 25 60 SOYBEAN 100 100 -- --      95 100 100 100 100 100 100 GREEN FXTL 95 95 -- -- 70 80 85 90 95 100 100      GIANT FXTL 100 100 -- -- 70 85 95 100 100 100 100 PANICUM 70 100 -- --      90 95 100 100 100 100 100 CRABGRASS 70 100 -- -- 0 0 20 40 50 65 80      BARNYARDGRASS 100 100 -- -- 95 100 100 100 100 100 100 JOHNSONGRASS 70      100 -- -- 100 100 100 100 100 100 100 SORGHUM 100 100 -- -- 100 100 100      100 100 100 100 NUTSEDGE 100 100 -- -- 85 100 100 100 109 100 100      VELVETLEAF 100 100 -- -- 80 90 100 100 100 100 100 COCKLEBUR 100 100 --      -- 95 100 100 100 100 100 100 SMARTWEED 100 100 -- -- 45 80 90 95 100      100 100 LAMBSQUARTER 100 100 -- -- 65 65 85 95 95 100 100 PIGWEED 100      100 -- -- 90 70 100 100 100 100 100 MORNINGGLORY 100 100 -- -- 95 100      100 100 100 100 100 JIMSONWEED 100 100 -- -- 85 95 100 100 100 100 100      PREEMERGENCE CORN 0 0 15 -- -- 0 0 0  0 0 45 SOYBEAN 60 85 100 -- -- 0 0      30 50 65 70 GREEN FXTL 85 100 100 -- -- 0 65 85 100 100 100 GIANT FXTL      90 100 100 -- -- 0 45 85 100 100 100 PANICUM 100 100 100 -- -- 20 75 100      100 100 100 CRABGRASS 65 90 100 -- -- 0 20 35 50 65 70 BARNYARDGRASS 50      90 100 -- -- 0 75 100 100 100 100 JOHNSONGRASS 100 100 100 -- -- 70 100      100 100 100 100 SORGHUM 100 100 100 -- -- 70 100 100 100 100 100      NUTSEDGE 80 100 100 -- -- 25 85 100 100 100 100 VELVETLEAF 25 50 85 --      -- 0 0 0 35 60 80 COCKLEBUR 0 35 70 -- -- 0 0 0 0 30 65 SMARTWEED 75 95      100 -- -- 30 0 20 30 50 100 LAMBSQUARTER 70 90 100 -- -- 25 25 75 100      100 100 PIGWEED 90 100 100 -- -- 45 30 80 100 100 100 MORNINGGLORY 20 40      85 -- -- 0 0 0 20 65 75 JIMSONWEED 30 70 90 -- -- 0 25 50 75 95 100

TEST D

Sixteen cm diameter Wagner pots, equipped with a stoppered drain opening near the bottom of the side wall, were partially filled with Woodstown sandy loam. About 1500 mls of water were added to each pot to bring the water level to a point 3 cm above the soil surface. Japonica and Indica rice seedlings were hand transplanted into the pots. Also, a number of barnyardgrass (Echinochloa crus-galli) seeds were added to each pot. At the same time, seedlings or tubers of the following species were transplanted into the muddy soil: water plantain (Alisma trivale), Scirpus (Scirpus mucranatus), and Cyperus (Cyperus difformis). The weed species selected for this test are of economic importance in major rice-growing areas. The chemical treatments were applied directly to the paddy water after being formulated in a nonphytotoxic solvent within hours after transplanting of two additional species: water chestnut (Eleocharis spp.) and arrowhead (Sagittaria latifolia). Shortly after treatment, the drain hole was opened to drop the water level by two cm. Water was then added to restore the water level to its original height. The following day the draining and refilling process was repeated. The pots were then maintained in the greenhouse.

Rates of application and plant response ratings made 21 days after treatment are summarized in Table D. Response ratings are based on a scale of 0 to 100 where 0=no effect and 100=complete control.

                  TABLE D                                                          ______________________________________                                                  Compound 188 Compound 189                                             Rate g/ha  0016   0008    0004  0016  0008 0004                                ______________________________________                                         Japonica Rice                                                                             0      0       0     15    15   0                                   Indica Rice                                                                               0      0       0     15    0    0                                   Barnyardgrass                                                                             77     22      0     95    77   30                                  Water Chestnut                                                                            82     87      85    90    85   70                                  Arrowhead  95     90      80    92    95   87                                  Scirpus    77     80      60    87    85   67                                  Cyperus    82     55      32    95    95   92                                  Water Plantain                                                                            75     75      60    85    72   67                                  ______________________________________                                    

TEST E

The weed species used in this test are all of major economic importance in soybean-growing regions. The following species are included in the screen:

    ______________________________________                                                                    GROWTH STAGE                                                                   AT APPLICA-                                                                    TION (POST-                                                                    EMERGENCE                                           Plant Species                                                                             Scientific Name PHASE)                                              ______________________________________                                         Grass Weeds:                                                                   barnyardgrass                                                                             Echinochloa crus-galli                                                                         2-3     leaves                                      giant foxtail                                                                             Setaria faberi  2-3     leaves                                      green foxtail                                                                             Setaria viridis 2-3     leaves                                      johnsongrass                                                                              Sorghum halepense                                                                              2-3     leaves                                      fall panicum                                                                              Panicum dichotomiflorum                                                                        2-3     leaves                                      broadleaf  Brachiaria platyphylla                                                                         2-3     leaves                                      signalgrass                                                                    large crabgrass                                                                           Digitaria sanguinalis                                                                          2-3     leaves                                      Broadleaf Weeds:                                                               velvetleaf Abutilon theophrasti                                                                           2-3     leaves                                      jimsonweed Datura stramonium                                                                              1-2     true leaves                                 hemp sesbania                                                                             Sesbania exaltata                                                                              1st     true leaf                                   sicklepod  Cassia obtusifolia                                                                             1st     true leaf                                   cocklebur  Xanthium pensylvanicum                                                                         2nd     true leaf                                   morningglory                                                                              Ipomoea hederacea                                                                              1-2     true leaves                                 ladysthumb Polygonum persicaria                                                                           3-4     leaves                                      smartweed                                                                      pigweed    Amaranthus retroflexus                                                                         4-5     leaves                                      lambsquarters                                                                             Chenopodium album                                                                              4-5     leaves                                      teaweed    Sida spinosa    2-3     leaves                                      black nightshade                                                                          Solanum nigrum  2nd     true leaf                                   purple nutsedge                                                                           Cyperus rotundus                                                                               5-6     leaves                                      corn       Zea mays        2-3     leaves                                      soybeans   Glycine max     1st     trifoliate                                  ______________________________________                                    

For the preemergence phase of the test, crop and weed species are planted in a Tama slit loam soil (approximately 3% organic matter). Approximate planting depths are: corn and soybeans--3 to 4 cm; morningglory, cocklebur, and nutsedge--2.5 to 3 cm; velvetleaf, sicklepod, and sesbania--2 cm; all other species--0.5 cm.

For the postemergence phase of the test, crop and weed species are planted in a Sassafras sandy loam soil (approximately 1% organic matter) one to three weeks before application so that they will be present as young plants at the time of treatment. Alternatively, for postemergence tests, plants are grown in a 50:50 mixture of commercially available potting mix and Sassafras soil. Approximate planting depths are: corn and soybeans--3 to 4 cm; morningglory, cocklebur, and nutsedge--2.5 to 3 cm; velvetleaf, sicklepod, and sesbania--2 cm; all other species--0.5 cm.

Treated plants and controls were maintained in a greenhouse for 3 to 4 weeks, after which all species were compared to controls and visually rated for response to treatment. The ratings, summarized in Table E, are based on a numerical scale extending from 0=no injury to 100=complete kill.

                  TABLE E                                                          ______________________________________                                         Postemergence                                                                  Rate = gm/h 0004   0008    0016 0032  0064 0125                                ______________________________________                                                   CMPD 206                                                              Soil type  Mix    Mix     Mix  Mix   Mix  Mix                                 Soybeans    0      0       10   15    20   25                                  Corn        40     70      90   100   100  100                                 Velvetleaf  50     75      100  100   100  100                                 Jimsonweed  30     40      40   50    85   95                                  Sicklepod   10     20      30   40    40   50                                  Hemp sesbania                                                                              20     40      50   75    85   95                                  Cocklebur   50     60      80   100   100  100                                 Ivy morningglory                                                                           75     85      90   95    100  100                                 Redroot pigweed                                                                            20     40      45   50    50   60                                  Lambsquarter                                                                               50     50      60   90    90   90                                  Prickly sida                                                                               30     45      50   65    75   85                                  Barnyardgrass                                                                              20     30      50   75    95   100                                 Giant foxtail                                                                              0      0       20   30    50   80                                  Green foxtail                                                                              0      30      40   50    60   70                                  Johnsongrass                                                                               20     30      40   50    60   70                                  Fall panicum                                                                               0      0       20   30    40   50                                  Large crabgrass                                                                            0      0       0    0     0    0                                   Brdlf sgnlgrass                                                                            20     30      40   50    50   70                                  Purple nutsedge                                                                            0      20      30   40    50   80                                  Lady smartweed                                                                             0      0       0    20    30   50                                  Black nightshad                                                                            50     60      70   95    100  100                                           CMPD 207                                                              Soil type  Mix    Mix     Mix  Mix   Mix  Mix                                 Soybeans    0      0       0    0     10   15                                  Corn        10     20      50   75    80   80                                  Velvetleaf  50     75      95   100   100  100                                 Jimsonweed  30     40      50   60    80   100                                 Sicklepod   0      20      30   40    50   80                                  Hemp sesbania                                                                              20     40      50   60    70   80                                  Cocklebur   50     60      70   100   100  100                                 Ivy morningglory                                                                           50     75      80   80    95   95                                  Redroot pigweed                                                                            20     30      50   60    70   95                                  Lambsquarter                                                                               50     50      70   80    80   95                                  Prickly sida                                                                               30     40      50   60    75   90                                  Barnyardgrass                                                                              0      0       20   40    65   100                                 Giant foxtail                                                                              0      30      40   50    60   80                                  Green foxtail                                                                              0      30      30   40    50   60                                  Johnsongrass                                                                               20     30      40   50    60   70                                  Fall panicum                                                                               0      0       0    0     0    0                                   Large crabgrass                                                                            0      0       0    0     0    0                                   Brdlf sgnlgrass                                                                            0      0       20   50    60   70                                  Purple nutsedge                                                                            0      20      30   40    100  80                                  Lady smartweed                                                                             0      20      30   40    50   65                                  Black nightshad                                                                            50     80      100  100   100  100                                 ______________________________________                                     

What is claimed is:
 1. A compound of the formula: ##STR44## wherein J is ##STR45## W is O, S or NR_(X) ; R_(X) is H, OH, C₁ -C₃ alkyl, C₁ -C₃ alkoxy, allyloxy, propargyloxy, C₁ -C₃ haloalkyl, C₁ -C₃ haloalkoxy or NR_(Y) R_(Z) ;R_(Y) is H or C₁ -C₃ alkyl; R_(Z) is C₁ -C₃ alkyl; G is O, S, SO or SO₂ ; m is 0 or 1; n is 0, 1 or 2; R is H or CH₃ ; E is a single bond, CH₂ or O; Q is ##STR46## R₁ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR_(a) R_(b), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, SCN, CO₂ R_(c), C₁ -C₃ haloalkoxy, C₁ -C₃ haloalkylthio, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ haloalkoxy, C₁ -C₂ alkylthio, C₁ -C₂ haloalkylthio or CN; R₂ is H, C₁ -C₃ alkyl, allyl or phenyl; R₃ is H, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, CH₂ -(C₂ -C₅ alkenyl), CH₂ (C₂ -C₅ haloalkenyl), CH₂ (C₂ -C₅ alkynyl), CH₂ (C₂ -C₅ haloalkynyl), C₆ H₅ or C₁ -C₄ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, C₁ -C₂ alkylsulfinyl or C₁ -C₂ alkylsulfonyl; R₄ is H, halogen, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, C₂ -C₆ alkenyl, C₂ -C₆ haloalkenyl, C₂ -C₆ alkynyl, C₃ -C₆ haloalkynyl, C₆ H₅, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, OCH₂ CH₂ O-(C₁ -C₂ alkyl) or di(C₁ -C₃ alkyl)amino; R₅ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, allyl or propargyl; R_(a) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy; R_(b) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or R_(a) and R_(b) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --; R_(c) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ haloalkyl, C₁ -C₂ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or C₂ -C₄ alkoxyalkyl; A is ##STR47## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₄ haloalkoxy, C₁ -C₄ haloalkyl, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₃ -C₅ cycloalkyl; Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₄ haloalkoxy, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₂ -C₅ alkylsulfinylalkyl, C₂ -C₅ alkylsulfonyalkyl, C₁ -C₄ haloalkyl, C₂ -C₄ alkynyl, azido, cyano ##STR48## or --N(OCH₃)CH₃ ; p is 2 or 3; L₁ and L₂ are independently O or S; R₆ is H or CH₃ ; R₇ and R₈ are independently C₁ -C₃ alkyl; and X₃ is CH₃ or OCH₃ ;and their agriculturally suitable salts; provided that (a) when J is J-9 and n is O, then Q is Q-1 or Q-2; (b) when E is O, then J is J-1; (c) when W is S, then A is A-1, R is H, and Y is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.sub..tbd.CH, OCH₂ CH₂ OCH₃, CH(OCH₃)₂ or ##STR49## (d) when the total number of carbon atoms in X and Y is greater than 4, then the carbon content of R₁, R₃, R₄ and R₅ must each be less than or equal to 2; (e) when J is J-1 and m is 0, then n is 0; and (f) when n is 0 and m is 1, then Q is Q-1 or Q-2.
 2. A compound of claim 1 where E is a single bond.
 3. A compound of claim 1 where E is CH₂.
 4. A compound of claim 1 where E is O.
 5. A compound of claim 2 where m is O; and W is O.
 6. A compound of claim 5 whereX is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, cyclopropyl, CH₂ F, CF₃, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and Y is H, C₁ -C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH₂ SCH₃, ##STR50##
 7. A compound of claim 6 whereR₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; and n is O.
 8. A compound of claim 7 whereR₃ is H, C₁ -C₃ alkyl, C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; and R₄ is H, C₁ -C₃ alkyl, C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, N(CH₃)₂, allyl, propargyl or C₁ -C₂ alkyl substituted with 1-3 atoms of F, Cl, or Br.
 9. A compound of claim 8 where J is J-1.
 10. A compound of claim 9 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 11. A compound of claim 10 where Q is Q₁.
 12. A compound of claim 10 where Q is Q₂.
 13. A compound of claim 10 where Q is Q₃.
 14. A compound of claim 10 where Q is Q₄.
 15. A compound of claim 10 where Q is Q₅.
 16. A compound of claim 10 where Q is Q₆.
 17. A compound of claim 10 where Q is Q₇.
 18. A compound of claim 8 where J is J-2.
 19. A compound of claim 18 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 20. A compound of claim 19 where Q is Q₁.
 21. A compound of claim 8 where J is J-3.
 22. A compound of claim 21 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 23. A compound of claim 22 where Q is Q₁.
 24. A compound of claim 8 where J is J-4.
 25. A compound of claim 24 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 26. A compound of claim 25 where Q is Q₁.
 27. A compound of claim 8 where J is J-5.
 28. A compound of claim 27 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 29. A compound of claim 28 where Q is Q₁.
 30. A compound of claim 8 where J is J-6.
 31. A compound of claim 30 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 32. A compound of claim 31 where Q is Q₁.
 33. A compound of claim 8 where J is J-7.
 34. A compound of claim 33 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 35. A compound of claim 34 where Q is Q₁.
 36. A compound of claim 8 where J is J-8.
 37. A compound of claim 36 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 38. A compound of claim 37 where Q is Q₁.
 39. A compound of claim 37 where Q is Q₂.
 40. A compound of claim 37 where Q is Q₃.
 41. A compound of claim 37 where Q is Q₄.
 42. A compound of claim 37 where Q is Q₅.
 43. A compound of claim 37 where Q is Q₆.
 44. A compound of claim 37 where Q is Q₇.
 45. A compound of claim 8 where J is J-9.
 46. A compound of claim 45 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 47. A compound of claim 46 where Q is Q₁.
 48. A compound of claim 8 where J is J-10.
 49. A compound of claim 48 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 50. A compound of claim 49 where Q is Q₁.
 51. A compound of claim 8 where J is J-11.
 52. A compound of claim 51 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 53. A compound of claim 52 where Q is Q₁.
 54. A compound of claim 8 where J is J-12.
 55. A compound of claim 54 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 56. A compound of claim 55 where Q is Q₁.
 57. A compound of claim 8 where J is J-13.
 58. A compound of claim 57 whereA is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 59. A compound of claim 58 where Q is Q₁.
 60. A compound of claim 3 wherem is 0; n is 0; J is J-1, J-2, J-3, J-8, J-10 or J-11; W is O; R is H; R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; R₃ is H, C₁ -C₃ alkyl, CH₂ CH₂ OCH₃, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; R₄ is H or C₁ -C₃ alkyl; A is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 61. A compound of claim 4 wherem is O; R is H; R₁ is H; R₃ is H or C₁ -C₃ alkyl; R₄ is H or C₁ -C₃ alkyl; A is A-1; X is CH₃, OCH₃, OCH₂ CH₃ or cyclopropyl; and Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.
 62. The compound of claim 1 which is N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide.
 63. The compound of claim 1 which is N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide, sodium salt.
 64. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 1 and at least one of the following: surfactant, solid or liquid diluent.
 65. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 2 and at least one of the following: surfactant, solid or liquid diluent.
 66. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 3 and at least one of the following: surfactant, solid or liquid diluent.
 67. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 4 and at least one of the following: surfactant, solid or liquid diluent.
 68. A compositon suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 5 and at least one of the following: surfactant, solid or liquid diluent.
 69. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 6 and at least one of the following: surfactant, solid or liquid diluent.
 70. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 62 and at least one of the following: surfactant, solid or liquid diluent.
 71. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 63 and at least one of the following: surfactant, solid or liquid diluent.
 72. A composition suitable for controlling the growth of undesired vegetation in soybean which comprises an effective amount of the compound of claim 62 and at least one of the following: surfactant, solid or liquid diluent.
 73. A composition suitable for controlling the growth of undesired vegetation in soybean which comprises an effective amount of the compound of claim 63 and at least one of the following: surfactant, solid or liquid diluent.
 74. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 1. 75. A method for controlling the growth of undesired vegetation which comprises applyng to the locus to be protected an effective amount of a compound of claim
 2. 76. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 3. 77. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 4. 78. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 5. 79. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 6. 80. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 62. 81. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 63. 82. A method for controlling the growth of undesired vegetation in soybean which comprises applying to the soybean field an effective amount of the compound of claim
 62. 83. A method for controlling the growth of undesired vegetation in soybean which comprises applying to the soybean field an effective amount of the compound of claim
 63. 